IS6421A - Nikótínamíð bensósambræddar-heterósýklýl afleiðurnytsamlegar sem valvísir latar á PDE4 samsætuensím - Google Patents

Nikótínamíð bensósambræddar-heterósýklýl afleiðurnytsamlegar sem valvísir latar á PDE4 samsætuensím

Info

Publication number
IS6421A
IS6421A IS6421A IS6421A IS6421A IS 6421 A IS6421 A IS 6421A IS 6421 A IS6421 A IS 6421A IS 6421 A IS6421 A IS 6421A IS 6421 A IS6421 A IS 6421A
Authority
IS
Iceland
Prior art keywords
benzosubstituted
pde4
nicotinamide
selective inhibitor
derivative useful
Prior art date
Application number
IS6421A
Other languages
English (en)
Inventor
Marfat Anthony
James Chambers Robert
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of IS6421A publication Critical patent/IS6421A/is

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Medicinal Chemistry (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
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  • Heart & Thoracic Surgery (AREA)
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  • Cardiology (AREA)
  • Diabetes (AREA)
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IS6421A 2000-01-31 2002-06-13 Nikótínamíð bensósambræddar-heterósýklýl afleiðurnytsamlegar sem valvísir latar á PDE4 samsætuensím IS6421A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928400P 2000-01-31 2000-01-31
PCT/IB2001/000124 WO2001057036A1 (en) 2000-01-31 2001-01-30 Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
IS6421A true IS6421A (is) 2002-06-13

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IS6421A IS6421A (is) 2000-01-31 2002-06-13 Nikótínamíð bensósambræddar-heterósýklýl afleiðurnytsamlegar sem valvísir latar á PDE4 samsætuensím

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UY (1) UY26569A1 (is)
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Families Citing this family (43)

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US7417038B1 (en) * 1998-10-15 2008-08-26 Imperial Innovations Limited Methods of treating cachexia
WO2001054666A1 (en) * 2000-01-28 2001-08-02 Alza Corporation Liposomes containing an entrapped compound in supersaturated solution
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