OA12709A - Pharmaceutical formulations for the controlled release of 4-amino-6,7-dimethoxa-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-YL)-5-(2-pyridyl)quinzoline. - Google Patents

Pharmaceutical formulations for the controlled release of 4-amino-6,7-dimethoxa-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-YL)-5-(2-pyridyl)quinzoline. Download PDF

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Publication number
OA12709A
OA12709A OA1200400094A OA1200400094A OA12709A OA 12709 A OA12709 A OA 12709A OA 1200400094 A OA1200400094 A OA 1200400094A OA 1200400094 A OA1200400094 A OA 1200400094A OA 12709 A OA12709 A OA 12709A
Authority
OA
OAPI
Prior art keywords
formulation
amino
pyridyl
dimethoxy
methanesulfonamido
Prior art date
Application number
OA1200400094A
Other languages
English (en)
Inventor
John Douglas Davis
Michael John Humphrey
Ross James Macrae
Janet Sarah Smith
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of OA12709A publication Critical patent/OA12709A/en

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
OA1200400094A 2001-10-11 2002-09-30 Pharmaceutical formulations for the controlled release of 4-amino-6,7-dimethoxa-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-YL)-5-(2-pyridyl)quinzoline. OA12709A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0124455.7A GB0124455D0 (en) 2001-10-11 2001-10-11 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
OA12709A true OA12709A (en) 2006-06-26

Family

ID=9923660

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200400094A OA12709A (en) 2001-10-11 2002-09-30 Pharmaceutical formulations for the controlled release of 4-amino-6,7-dimethoxa-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-YL)-5-(2-pyridyl)quinzoline.

Country Status (33)

Country Link
EP (1) EP1434570B8 (is)
JP (1) JP4131471B2 (is)
KR (1) KR20050032510A (is)
CN (1) CN1568180A (is)
AP (1) AP2004003001A0 (is)
AR (1) AR036782A1 (is)
AT (1) ATE303135T1 (is)
BR (1) BR0213196A (is)
CA (1) CA2461168A1 (is)
CO (1) CO5560534A2 (is)
DE (1) DE60205925T2 (is)
DK (1) DK1434570T3 (is)
DO (1) DOP2002000464A (is)
EA (1) EA006168B1 (is)
ES (1) ES2246017T3 (is)
GB (1) GB0124455D0 (is)
GT (1) GT200200184A (is)
HR (1) HRP20040261A2 (is)
HU (1) HUP0600064A3 (is)
IL (1) IL160969A0 (is)
IS (1) IS7179A (is)
MA (1) MA27075A1 (is)
MX (1) MXPA04003293A (is)
NO (1) NO20041520L (is)
OA (1) OA12709A (is)
PA (1) PA8556001A1 (is)
PE (1) PE20030551A1 (is)
PL (1) PL369666A1 (is)
PY (1) PY0223360A (is)
SV (1) SV2004001279A (is)
UY (1) UY27477A1 (is)
WO (1) WO2003032956A1 (is)
ZA (1) ZA200401976B (is)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0317663D0 (en) * 2003-07-29 2003-09-03 Astrazeneca Ab Pharmaceutical composition
KR102474467B1 (ko) 2013-03-14 2022-12-05 암젠 인크 복소환식 화합물 및 그들의 용도
KR101943592B1 (ko) 2017-08-31 2019-01-30 조현우 데이터 마이닝 기법을 이용한 전자가계부 시스템

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69008526T2 (de) * 1990-07-02 1994-08-18 Bend Res Inc Asymmetrische mikroporöse Kügelchen für regulierbare Freigabe.
FR2752737B1 (fr) * 1996-08-29 1998-10-02 Synthelabo Comprime a liberation controlee de chlorhydrate d'alfuzosine
GB9700504D0 (en) * 1997-01-11 1997-02-26 Pfizer Ltd Pharmaceutical compounds
IL141235A (en) * 2000-02-09 2012-04-30 Novartis Int Pharm Ltd Combined use of an alpha-adrenoceptor antagonist and a muscarinic antagonist in the preparation of a drug for the treatment of non-malignant prostatic hyperplasia
JP3857919B2 (ja) * 2000-03-03 2006-12-13 ファイザー・インク 4−アミノ−6,7−ジメトキシ−2−(5−メタンスルホンアミド−1,2,3,4−テトラヒドロイソキノル−2−イル)−5−(2−ピリジル)キナゾリンメシラートおよび多形

Also Published As

Publication number Publication date
AP2004003001A0 (en) 2004-03-31
CO5560534A2 (es) 2005-09-30
GB0124455D0 (en) 2001-12-05
GT200200184A (es) 2003-05-23
KR20050032510A (ko) 2005-04-07
EA200400431A1 (ru) 2004-08-26
BR0213196A (pt) 2004-08-31
UY27477A1 (es) 2003-05-30
EP1434570B1 (en) 2005-08-31
CA2461168A1 (en) 2003-04-24
DE60205925T2 (de) 2006-06-08
IL160969A0 (en) 2004-08-31
WO2003032956A1 (en) 2003-04-24
IS7179A (is) 2004-03-11
ZA200401976B (en) 2004-07-12
JP4131471B2 (ja) 2008-08-13
EA006168B1 (ru) 2005-10-27
ES2246017T3 (es) 2006-02-01
SV2004001279A (es) 2004-02-19
HUP0600064A2 (en) 2006-06-28
AR036782A1 (es) 2004-10-06
EP1434570A1 (en) 2004-07-07
ATE303135T1 (de) 2005-09-15
PE20030551A1 (es) 2003-06-26
MA27075A1 (fr) 2004-12-20
NO20041520L (no) 2004-04-05
DE60205925D1 (de) 2005-10-06
PL369666A1 (en) 2005-05-02
PY0223360A (es) 2004-04-01
DOP2002000464A (es) 2003-04-15
HUP0600064A3 (en) 2007-02-28
DK1434570T3 (da) 2005-11-07
JP2005507909A (ja) 2005-03-24
EP1434570B8 (en) 2005-10-26
CN1568180A (zh) 2005-01-19
PA8556001A1 (es) 2003-07-28
HRP20040261A2 (en) 2004-08-31
MXPA04003293A (es) 2004-07-23

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