IS7186A - Kínuklídínafleiður, aðferðir til framleiðslu þeirra og notkun þeirra sem M2 og/eða M3 múskarín viðtakahindra - Google Patents

Kínuklídínafleiður, aðferðir til framleiðslu þeirra og notkun þeirra sem M2 og/eða M3 múskarín viðtakahindra

Info

Publication number
IS7186A
IS7186A IS7186A IS7186A IS7186A IS 7186 A IS7186 A IS 7186A IS 7186 A IS7186 A IS 7186A IS 7186 A IS7186 A IS 7186A IS 7186 A IS7186 A IS 7186A
Authority
IS
Iceland
Prior art keywords
production methods
muscarinic receptor
receptor inhibitors
quinuclidine derivatives
quinuclidine
Prior art date
Application number
IS7186A
Other languages
English (en)
Inventor
Guyaux Michel
U. Dinesh Chimmanamada
Mioskowski Charles
Quere Luc
Starck Jean-Philippe
Talaga Patrice
Wagner Alain
Zanda Matteo
Original Assignee
Ucb, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb, S.A. filed Critical Ucb, S.A.
Publication of IS7186A publication Critical patent/IS7186A/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS7186A 2001-10-17 2004-03-18 Kínuklídínafleiður, aðferðir til framleiðslu þeirra og notkun þeirra sem M2 og/eða M3 múskarín viðtakahindra IS7186A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01124727 2001-10-17
PCT/EP2002/010644 WO2003033495A1 (en) 2001-10-17 2002-09-23 Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors

Publications (1)

Publication Number Publication Date
IS7186A true IS7186A (is) 2004-03-18

Family

ID=8178984

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7186A IS7186A (is) 2001-10-17 2004-03-18 Kínuklídínafleiður, aðferðir til framleiðslu þeirra og notkun þeirra sem M2 og/eða M3 múskarín viðtakahindra

Country Status (19)

Country Link
US (1) US7361668B2 (is)
EP (1) EP1438309A1 (is)
JP (1) JP2005512974A (is)
KR (1) KR20050030169A (is)
CN (1) CN1571787A (is)
BG (1) BG108683A (is)
BR (1) BR0212983A (is)
CA (1) CA2462980A1 (is)
CZ (1) CZ2004501A3 (is)
HU (1) HUP0401849A3 (is)
IL (1) IL160896A0 (is)
IS (1) IS7186A (is)
MX (1) MXPA04002983A (is)
NO (1) NO20042023L (is)
NZ (1) NZ532283A (is)
PL (1) PL370087A1 (is)
RU (1) RU2004110717A (is)
WO (1) WO2003033495A1 (is)
ZA (1) ZA200402060B (is)

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WO2009152392A2 (en) * 2008-06-11 2009-12-17 University Of Toledo Muscarinic agonists for neurological disorders and methods of making the same
PL2391366T3 (pl) 2009-01-29 2013-04-30 Novartis Ag Podstawione benzimidazole do leczenia gwiaździaków
US8389526B2 (en) 2009-08-07 2013-03-05 Novartis Ag 3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
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WO2012116237A2 (en) 2011-02-23 2012-08-30 Intellikine, Llc Heterocyclic compounds and uses thereof
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Also Published As

Publication number Publication date
BR0212983A (pt) 2004-10-13
IL160896A0 (en) 2004-08-31
NO20042023L (no) 2004-05-14
US20050020660A1 (en) 2005-01-27
RU2004110717A (ru) 2005-10-20
EP1438309A1 (en) 2004-07-21
US7361668B2 (en) 2008-04-22
BG108683A (en) 2005-04-30
MXPA04002983A (es) 2004-07-15
KR20050030169A (ko) 2005-03-29
ZA200402060B (en) 2005-03-15
HUP0401849A2 (hu) 2004-12-28
HUP0401849A3 (en) 2007-05-02
CA2462980A1 (en) 2003-04-24
NZ532283A (en) 2005-06-24
PL370087A1 (en) 2005-05-16
CN1571787A (zh) 2005-01-26
JP2005512974A (ja) 2005-05-12
CZ2004501A3 (cs) 2004-09-15
WO2003033495A1 (en) 2003-04-24

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