NO20042023L - Kinuklidinderivater fremgangsmate for flemstilling av disse og anvendelse av disse som m2- og/eller m3-muskarinreseptor-inhibitorer - Google Patents

Kinuklidinderivater fremgangsmate for flemstilling av disse og anvendelse av disse som m2- og/eller m3-muskarinreseptor-inhibitorer

Info

Publication number
NO20042023L
NO20042023L NO20042023A NO20042023A NO20042023L NO 20042023 L NO20042023 L NO 20042023L NO 20042023 A NO20042023 A NO 20042023A NO 20042023 A NO20042023 A NO 20042023A NO 20042023 L NO20042023 L NO 20042023L
Authority
NO
Norway
Prior art keywords
kinuclidine
multiplying
receptor inhibitors
derivatives process
muscarin receptor
Prior art date
Application number
NO20042023A
Other languages
English (en)
Norwegian (no)
Inventor
Michel Guyaux
Chimmanamnada U Dinesh
Charles Mioskowski
Luc Quere
Jean-Philippe Starck
Patrice Talaga
Alain Wagner
Matteo ZANDA
Original Assignee
Ucb Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Sa filed Critical Ucb Sa
Publication of NO20042023L publication Critical patent/NO20042023L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20042023A 2001-10-17 2004-05-14 Kinuklidinderivater fremgangsmate for flemstilling av disse og anvendelse av disse som m2- og/eller m3-muskarinreseptor-inhibitorer NO20042023L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01124727 2001-10-17
PCT/EP2002/010644 WO2003033495A1 (en) 2001-10-17 2002-09-23 Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors

Publications (1)

Publication Number Publication Date
NO20042023L true NO20042023L (no) 2004-05-14

Family

ID=8178984

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20042023A NO20042023L (no) 2001-10-17 2004-05-14 Kinuklidinderivater fremgangsmate for flemstilling av disse og anvendelse av disse som m2- og/eller m3-muskarinreseptor-inhibitorer

Country Status (19)

Country Link
US (1) US7361668B2 (is)
EP (1) EP1438309A1 (is)
JP (1) JP2005512974A (is)
KR (1) KR20050030169A (is)
CN (1) CN1571787A (is)
BG (1) BG108683A (is)
BR (1) BR0212983A (is)
CA (1) CA2462980A1 (is)
CZ (1) CZ2004501A3 (is)
HU (1) HUP0401849A3 (is)
IL (1) IL160896A0 (is)
IS (1) IS7186A (is)
MX (1) MXPA04002983A (is)
NO (1) NO20042023L (is)
NZ (1) NZ532283A (is)
PL (1) PL370087A1 (is)
RU (1) RU2004110717A (is)
WO (1) WO2003033495A1 (is)
ZA (1) ZA200402060B (is)

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UY28871A1 (es) 2004-04-27 2005-11-30 Glaxo Group Ltd Antagonistas del receptor de acetilcolina muscarinico
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US8268834B2 (en) 2008-03-19 2012-09-18 Novartis Ag Pyrazine derivatives that inhibit phosphatidylinositol 3-kinase enzyme
WO2009140483A1 (en) 2008-05-15 2009-11-19 University Of Toledo Muscarinic agonists as cognitive enhancers
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WO2009152392A2 (en) * 2008-06-11 2009-12-17 University Of Toledo Muscarinic agonists for neurological disorders and methods of making the same
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US8389526B2 (en) 2009-08-07 2013-03-05 Novartis Ag 3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
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EP2673277A1 (en) 2011-02-10 2013-12-18 Novartis AG [1, 2, 4]triazolo [4, 3 -b]pyridazine compounds as inhibitors of the c-met tyrosine kinase
WO2012116237A2 (en) 2011-02-23 2012-08-30 Intellikine, Llc Heterocyclic compounds and uses thereof
MA34969B1 (fr) 2011-02-25 2014-03-01 Irm Llc Composes et compositions en tant qu inibiteurs de trk
US9549928B2 (en) 2011-04-29 2017-01-24 The University Of Toledo Muscarinic agonists as enhancers of cognitive flexibility
US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
CA2848809A1 (en) 2011-09-15 2013-03-21 Novartis Ag 6-substituted 3-(quinolin-6-ylthio)-[1,2,4]triazolo[4,3-a]pyradines as c-met tyrosine kinase
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JP6130391B2 (ja) 2011-11-23 2017-05-17 インテリカイン， エルエルシー Ｍｔｏｒ阻害剤を使用する強化された治療レジメン
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Also Published As

Publication number Publication date
BR0212983A (pt) 2004-10-13
IL160896A0 (en) 2004-08-31
US20050020660A1 (en) 2005-01-27
RU2004110717A (ru) 2005-10-20
EP1438309A1 (en) 2004-07-21
IS7186A (is) 2004-03-18
US7361668B2 (en) 2008-04-22
BG108683A (en) 2005-04-30
MXPA04002983A (es) 2004-07-15
KR20050030169A (ko) 2005-03-29
ZA200402060B (en) 2005-03-15
HUP0401849A2 (hu) 2004-12-28
HUP0401849A3 (en) 2007-05-02
CA2462980A1 (en) 2003-04-24
NZ532283A (en) 2005-06-24
PL370087A1 (en) 2005-05-16
CN1571787A (zh) 2005-01-26
JP2005512974A (ja) 2005-05-12
CZ2004501A3 (cs) 2004-09-15
WO2003033495A1 (en) 2003-04-24

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