IT1053787B - Macrolidi azotati e loro preparazione - Google Patents

Macrolidi azotati e loro preparazione

Info

Publication number
IT1053787B
IT1053787B IT28908/74A IT2890874A IT1053787B IT 1053787 B IT1053787 B IT 1053787B IT 28908/74 A IT28908/74 A IT 28908/74A IT 2890874 A IT2890874 A IT 2890874A IT 1053787 B IT1053787 B IT 1053787B
Authority
IT
Italy
Prior art keywords
macrolids
nitrogen
preparation
nitrogen macrolids
Prior art date
Application number
IT28908/74A
Other languages
English (en)
Original Assignee
Pastori A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pastori A filed Critical Pastori A
Priority to IT28908/74A priority Critical patent/IT1053787B/it
Priority to GB42393/75A priority patent/GB1480700A/en
Priority to US05/623,117 priority patent/US4007169A/en
Priority to DE19752548128 priority patent/DE2548128A1/de
Priority to JP50128976A priority patent/JPS5168597A/ja
Priority to DE19752548148 priority patent/DE2548148A1/de
Priority to JP50128975A priority patent/JPS5168596A/ja
Priority to FR7533002A priority patent/FR2289509A1/fr
Priority to FR7533001A priority patent/FR2289508A1/fr
Application granted granted Critical
Publication of IT1053787B publication Critical patent/IT1053787B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT28908/74A 1974-10-29 1974-10-29 Macrolidi azotati e loro preparazione IT1053787B (it)

Priority Applications (9)

Application Number Priority Date Filing Date Title
IT28908/74A IT1053787B (it) 1974-10-29 1974-10-29 Macrolidi azotati e loro preparazione
GB42393/75A GB1480700A (en) 1974-10-29 1975-10-16 Rifamycin s and sv derivatives
US05/623,117 US4007169A (en) 1974-10-29 1975-10-16 Method of preparing derivatives of rifamycin S
DE19752548128 DE2548128A1 (de) 1974-10-29 1975-10-28 Neue derivate des s-rifamycins und verfahren zu ihrer herstellung
JP50128976A JPS5168597A (en) 1974-10-29 1975-10-28 Rifuamaishin s judotainoseiho
DE19752548148 DE2548148A1 (de) 1974-10-29 1975-10-28 Verfahren zur herstellung von derivaten des s-rifamycins und neue s-rifamycinverbindungen
JP50128975A JPS5168596A (en) 1974-10-29 1975-10-28 Rifuamaishin s nojudotainoseiho
FR7533002A FR2289509A1 (fr) 1974-10-29 1975-10-29 Procede pour l'obtention de derives de la rifamycine s
FR7533001A FR2289508A1 (fr) 1974-10-29 1975-10-29 Derives de la rifamycine s

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT28908/74A IT1053787B (it) 1974-10-29 1974-10-29 Macrolidi azotati e loro preparazione

Publications (1)

Publication Number Publication Date
IT1053787B true IT1053787B (it) 1981-10-10

Family

ID=11224499

Family Applications (1)

Application Number Title Priority Date Filing Date
IT28908/74A IT1053787B (it) 1974-10-29 1974-10-29 Macrolidi azotati e loro preparazione

Country Status (6)

Country Link
US (1) US4007169A (it)
JP (2) JPS5168597A (it)
DE (2) DE2548128A1 (it)
FR (2) FR2289508A1 (it)
GB (1) GB1480700A (it)
IT (1) IT1053787B (it)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1068367B (it) * 1975-11-12 1985-03-21 Archifar Ind Chim Trentino 3 aldimino rifamicine ad alta attivita antibiotica loro derivati e procedimento per ottenerle
CH629212A5 (it) * 1976-10-18 1982-04-15 Erba Farmitalia Procedimento per la preparazione di composti di rifamicina.
GB1576886A (en) * 1977-04-20 1980-10-15 Lepetit Spa Rifamycin derivatives
IT7828731A0 (it) * 1977-11-05 1978-10-13 Archifar Lab Chim Farm Procedimento per la produzione di 3-aminoderivati della rifamicina s.
IT1090759B (it) * 1977-11-29 1985-06-26 Alfa Farmaceutici Spa Procedimento per la preparazione di 3 iodio e 3 bromo rifamicina s
GB1591697A (en) * 1978-03-09 1981-06-24 Archifar Lab Chim Farm Process for producing 3-amino-rifamycins s and sv
GB1591696A (en) * 1978-03-09 1981-06-24 Archifar Lab Chim Farm 3-nitro-rifamycins s and sv
US4217278A (en) * 1978-03-09 1980-08-12 Archifar Laboratori Chimico Farmacologici S.P.A. 3-Nitro-rifamycins S and SV
GR69740B (it) * 1979-07-20 1982-07-12 Ciba Geigy Ag
US4743619A (en) * 1985-08-29 1988-05-10 American Home Products Corporation Method of treating hepatitis
US4631290A (en) * 1985-08-29 1986-12-23 American Home Products Corporation Method of treating hepatitis
DE69227790T2 (de) * 1991-01-28 1999-06-10 Gruppo Lepetit S.P.A., Lainate Verfahren zur Herstellung von 2'-Diethylaminorifamycin P (P/DEA)
RU2245336C2 (ru) * 2002-09-27 2005-01-27 ЗАО "Вектон" Способ получения 3-аминопроизводных рифамицина s
RU2245337C2 (ru) * 2002-09-27 2005-01-27 ЗАО "Вектон" Способ получения 3-азидопроизводных рифамицина s
RU2256663C2 (ru) * 2003-07-22 2005-07-20 Гитлин Исаак Григорьевич Способ получения 3-аминорифампицина-s (варианты)
CN105001236B (zh) * 2015-06-26 2017-05-31 重庆华邦制药有限公司 3‑氨基‑利福霉素s的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH536851A (de) * 1966-10-25 1973-05-15 Ciba Geigy Ag Verfahren zur Herstellung neuer antibiotisch wirksamer Verbindungen der Rifamycinreihen
AR205434A1 (es) * 1972-03-27 1976-05-07 Lepetit Spa Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
US3900465A (en) * 1973-04-05 1975-08-19 Lepetit Spa 3-formylrifamycin azines

Also Published As

Publication number Publication date
FR2289508A1 (fr) 1976-05-28
GB1480700A (en) 1977-07-20
FR2289509A1 (fr) 1976-05-28
JPS5168597A (en) 1976-06-14
JPS5421360B2 (it) 1979-07-30
JPS5168596A (en) 1976-06-14
DE2548128A1 (de) 1976-05-13
DE2548148A1 (de) 1976-05-06
US4007169A (en) 1977-02-08

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