IT1053787B - Macrolidi azotati e loro preparazione - Google Patents
Macrolidi azotati e loro preparazioneInfo
- Publication number
- IT1053787B IT1053787B IT28908/74A IT2890874A IT1053787B IT 1053787 B IT1053787 B IT 1053787B IT 28908/74 A IT28908/74 A IT 28908/74A IT 2890874 A IT2890874 A IT 2890874A IT 1053787 B IT1053787 B IT 1053787B
- Authority
- IT
- Italy
- Prior art keywords
- macrolids
- nitrogen
- preparation
- nitrogen macrolids
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT28908/74A IT1053787B (it) | 1974-10-29 | 1974-10-29 | Macrolidi azotati e loro preparazione |
| GB42393/75A GB1480700A (en) | 1974-10-29 | 1975-10-16 | Rifamycin s and sv derivatives |
| US05/623,117 US4007169A (en) | 1974-10-29 | 1975-10-16 | Method of preparing derivatives of rifamycin S |
| DE19752548128 DE2548128A1 (de) | 1974-10-29 | 1975-10-28 | Neue derivate des s-rifamycins und verfahren zu ihrer herstellung |
| JP50128976A JPS5168597A (en) | 1974-10-29 | 1975-10-28 | Rifuamaishin s judotainoseiho |
| DE19752548148 DE2548148A1 (de) | 1974-10-29 | 1975-10-28 | Verfahren zur herstellung von derivaten des s-rifamycins und neue s-rifamycinverbindungen |
| JP50128975A JPS5168596A (en) | 1974-10-29 | 1975-10-28 | Rifuamaishin s nojudotainoseiho |
| FR7533002A FR2289509A1 (fr) | 1974-10-29 | 1975-10-29 | Procede pour l'obtention de derives de la rifamycine s |
| FR7533001A FR2289508A1 (fr) | 1974-10-29 | 1975-10-29 | Derives de la rifamycine s |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT28908/74A IT1053787B (it) | 1974-10-29 | 1974-10-29 | Macrolidi azotati e loro preparazione |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IT1053787B true IT1053787B (it) | 1981-10-10 |
Family
ID=11224499
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT28908/74A IT1053787B (it) | 1974-10-29 | 1974-10-29 | Macrolidi azotati e loro preparazione |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US4007169A (it) |
| JP (2) | JPS5168597A (it) |
| DE (2) | DE2548128A1 (it) |
| FR (2) | FR2289508A1 (it) |
| GB (1) | GB1480700A (it) |
| IT (1) | IT1053787B (it) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1068367B (it) * | 1975-11-12 | 1985-03-21 | Archifar Ind Chim Trentino | 3 aldimino rifamicine ad alta attivita antibiotica loro derivati e procedimento per ottenerle |
| CH629212A5 (it) * | 1976-10-18 | 1982-04-15 | Erba Farmitalia | Procedimento per la preparazione di composti di rifamicina. |
| GB1576886A (en) * | 1977-04-20 | 1980-10-15 | Lepetit Spa | Rifamycin derivatives |
| IT7828731A0 (it) * | 1977-11-05 | 1978-10-13 | Archifar Lab Chim Farm | Procedimento per la produzione di 3-aminoderivati della rifamicina s. |
| IT1090759B (it) * | 1977-11-29 | 1985-06-26 | Alfa Farmaceutici Spa | Procedimento per la preparazione di 3 iodio e 3 bromo rifamicina s |
| GB1591697A (en) * | 1978-03-09 | 1981-06-24 | Archifar Lab Chim Farm | Process for producing 3-amino-rifamycins s and sv |
| GB1591696A (en) * | 1978-03-09 | 1981-06-24 | Archifar Lab Chim Farm | 3-nitro-rifamycins s and sv |
| US4217278A (en) * | 1978-03-09 | 1980-08-12 | Archifar Laboratori Chimico Farmacologici S.P.A. | 3-Nitro-rifamycins S and SV |
| GR69740B (it) * | 1979-07-20 | 1982-07-12 | Ciba Geigy Ag | |
| US4743619A (en) * | 1985-08-29 | 1988-05-10 | American Home Products Corporation | Method of treating hepatitis |
| US4631290A (en) * | 1985-08-29 | 1986-12-23 | American Home Products Corporation | Method of treating hepatitis |
| DE69227790T2 (de) * | 1991-01-28 | 1999-06-10 | Gruppo Lepetit S.P.A., Lainate | Verfahren zur Herstellung von 2'-Diethylaminorifamycin P (P/DEA) |
| RU2245336C2 (ru) * | 2002-09-27 | 2005-01-27 | ЗАО "Вектон" | Способ получения 3-аминопроизводных рифамицина s |
| RU2245337C2 (ru) * | 2002-09-27 | 2005-01-27 | ЗАО "Вектон" | Способ получения 3-азидопроизводных рифамицина s |
| RU2256663C2 (ru) * | 2003-07-22 | 2005-07-20 | Гитлин Исаак Григорьевич | Способ получения 3-аминорифампицина-s (варианты) |
| CN105001236B (zh) * | 2015-06-26 | 2017-05-31 | 重庆华邦制药有限公司 | 3‑氨基‑利福霉素s的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH536851A (de) * | 1966-10-25 | 1973-05-15 | Ciba Geigy Ag | Verfahren zur Herstellung neuer antibiotisch wirksamer Verbindungen der Rifamycinreihen |
| AR205434A1 (es) * | 1972-03-27 | 1976-05-07 | Lepetit Spa | Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv |
| US3900465A (en) * | 1973-04-05 | 1975-08-19 | Lepetit Spa | 3-formylrifamycin azines |
-
1974
- 1974-10-29 IT IT28908/74A patent/IT1053787B/it active
-
1975
- 1975-10-16 US US05/623,117 patent/US4007169A/en not_active Expired - Lifetime
- 1975-10-16 GB GB42393/75A patent/GB1480700A/en not_active Expired
- 1975-10-28 JP JP50128976A patent/JPS5168597A/ja active Pending
- 1975-10-28 JP JP50128975A patent/JPS5168596A/ja active Granted
- 1975-10-28 DE DE19752548128 patent/DE2548128A1/de active Pending
- 1975-10-28 DE DE19752548148 patent/DE2548148A1/de active Pending
- 1975-10-29 FR FR7533001A patent/FR2289508A1/fr not_active Withdrawn
- 1975-10-29 FR FR7533002A patent/FR2289509A1/fr not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| FR2289508A1 (fr) | 1976-05-28 |
| GB1480700A (en) | 1977-07-20 |
| FR2289509A1 (fr) | 1976-05-28 |
| JPS5168597A (en) | 1976-06-14 |
| JPS5421360B2 (it) | 1979-07-30 |
| JPS5168596A (en) | 1976-06-14 |
| DE2548128A1 (de) | 1976-05-13 |
| DE2548148A1 (de) | 1976-05-06 |
| US4007169A (en) | 1977-02-08 |
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