IT1287588B1 - Forma cristallina del doxazosin mesilato e processo per la sua produzione - Google Patents

Forma cristallina del doxazosin mesilato e processo per la sua produzione

Info

Publication number
IT1287588B1
IT1287588B1 IT96BO000657A ITBO960657A IT1287588B1 IT 1287588 B1 IT1287588 B1 IT 1287588B1 IT 96BO000657 A IT96BO000657 A IT 96BO000657A IT BO960657 A ITBO960657 A IT BO960657A IT 1287588 B1 IT1287588 B1 IT 1287588B1
Authority
IT
Italy
Prior art keywords
mesilate
doxazosin
production
crystalline form
crystalline
Prior art date
Application number
IT96BO000657A
Other languages
English (en)
Inventor
Vincenzo Cannata
Silvano Piani
Cristina Carrara
Stefano Saguatti
Original Assignee
Alfa Chem Ital
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfa Chem Ital filed Critical Alfa Chem Ital
Priority to IT96BO000657A priority Critical patent/IT1287588B1/it
Publication of ITBO960657A0 publication Critical patent/ITBO960657A0/it
Priority to EP97118048A priority patent/EP0848001A1/en
Priority to CA002219613A priority patent/CA2219613A1/en
Priority to JP9343363A priority patent/JPH10175974A/ja
Publication of ITBO960657A1 publication Critical patent/ITBO960657A1/it
Application granted granted Critical
Publication of IT1287588B1 publication Critical patent/IT1287588B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT96BO000657A 1996-12-13 1996-12-13 Forma cristallina del doxazosin mesilato e processo per la sua produzione IT1287588B1 (it)

Priority Applications (4)

Application Number Priority Date Filing Date Title
IT96BO000657A IT1287588B1 (it) 1996-12-13 1996-12-13 Forma cristallina del doxazosin mesilato e processo per la sua produzione
EP97118048A EP0848001A1 (en) 1996-12-13 1997-10-17 Crystalline form of the doxazosin mesylate and process for its production
CA002219613A CA2219613A1 (en) 1996-12-13 1997-10-29 Crystalline form of the doxazosin mesylate and process for its production
JP9343363A JPH10175974A (ja) 1996-12-13 1997-12-12 ドキサゾシンメシラートの結晶粉末およびその製造法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT96BO000657A IT1287588B1 (it) 1996-12-13 1996-12-13 Forma cristallina del doxazosin mesilato e processo per la sua produzione

Publications (3)

Publication Number Publication Date
ITBO960657A0 ITBO960657A0 (it) 1996-12-13
ITBO960657A1 ITBO960657A1 (it) 1998-06-13
IT1287588B1 true IT1287588B1 (it) 1998-08-06

Family

ID=11341786

Family Applications (1)

Application Number Title Priority Date Filing Date
IT96BO000657A IT1287588B1 (it) 1996-12-13 1996-12-13 Forma cristallina del doxazosin mesilato e processo per la sua produzione

Country Status (4)

Country Link
EP (1) EP0848001A1 (it)
JP (1) JPH10175974A (it)
CA (1) CA2219613A1 (it)
IT (1) IT1287588B1 (it)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19800214A1 (de) * 1998-01-06 1999-07-15 Knoll Ag Verfahren zur Herstellung von Doxazosin-Mcsylat in einer als Form A bezeichneten Kristallmodifikation und ein Zwischenprodukt dafür
ES2164520B1 (es) * 1999-03-16 2003-04-01 Medichem Sa "procedimiento de obtencion del polimorfo a del mesilato de doxazosina"
DE19912063A1 (de) * 1999-03-18 2000-09-21 Knoll Ag Neues Verfahren zur Herstellung von Doxazosin-Mesylat in einer als Form A bezeichneten Kristallmodifikation
DE19912573A1 (de) * 1999-03-19 2000-09-21 Knoll Ag Arzneimittel, enthaltend Doxazosin-Mesylat der Kristallmodifikaton D
NZ585558A (en) * 2007-12-24 2011-08-26 Cipla Ltd Crystalline polymorph of doxazosin mesylate (form iv) and process for preparation thereof
CN109988158A (zh) * 2018-01-03 2019-07-09 合肥立方制药股份有限公司 X晶型、含有x晶型的多沙唑嗪甲磺酸盐及其制备方法和用途

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4188390A (en) * 1977-11-05 1980-02-12 Pfizer Inc. Antihypertensive 4-amino-2-[4-(1,4-benzodioxan-2-carbonyl) piperazin-1-yl or homopiperazin-1-yl]quinazolines

Also Published As

Publication number Publication date
EP0848001A1 (en) 1998-06-17
CA2219613A1 (en) 1998-06-13
ITBO960657A0 (it) 1996-12-13
JPH10175974A (ja) 1998-06-30
ITBO960657A1 (it) 1998-06-13

Similar Documents

Publication Publication Date Title
BR9500835A (pt) Processo para produção de poliisobutenos
NO992860D0 (no) FremgangsmÕte for fremstilling av hydrokarboner
ITMI932628A0 (it) Processo per la produzione di policarbonati alifatico-armatici
BR9306120A (pt) Fibra e processo para sua produção
ITMI932478A0 (it) Processo per la produzione di policarbonati
IT1292427B1 (it) Procedimento e apparecchiatura per la produzione di melammina
IT1289763B1 (it) Processo per la produziond di cefazolina
ITBO960657A0 (it) Forma cristallina del doxazosin mesilato e processo per la sua produzione
ITMI920350A0 (it) Processo per la produzione di pezzi smaltati
ITMI932479A0 (it) Processo per la produzione di policarbonati
ITMI911393A0 (it) Processo per la produzione di profilati in composito fibroso
ITMI951612A0 (it) Processo per la produzione di agenti contrastografici iodurati
IT1310687B1 (it) Procedimento per la produzione e struttura di utensili per iltrattamento di sagomatura di pietre
ITRM960874A0 (it) Procedimento migliorato per la produzione di 5-idrossimetiltiazolo
ITMI913254A0 (it) Antibiotico ab-041 e processo per la sua produzione
ITMI921156A0 (it) Processo per la produzione di idrossialchil-glucosidi
FI952142L (fi) Parannettu suurtuotantomenetelmä atsapironin synteesiä varten
IT1286595B1 (it) Procedimento per la produzione di monili comprendenti pietre infilzate
ITMI940327A0 (it) Processo per la produzione di policarbonati alifatico-aromatici
IT1290850B1 (it) Processo per la produzione di polialcoli
IT1290851B1 (it) Processo per la produzione di polialcoli
IT1286790B1 (it) Processo per la produzione della forma i del terazosin monocloridrato anidro
IT1286789B1 (it) Processo per la produzione della forma i del terazosin monocloridato anidro
ITMI921303A0 (it) Processo per la produzione di l-amminoantrachinone
IT1279694B1 (it) Forma polimorfa di terazosin monocloridrato e processo per la sua produzione.

Legal Events

Date Code Title Description
0001 Granted