IT8047529A0 - Derivati di acido epossisuccinico dotati di proprieta' farmacologiche - Google Patents

Derivati di acido epossisuccinico dotati di proprieta' farmacologiche

Info

Publication number
IT8047529A0
IT8047529A0 IT8047529A IT4752980A IT8047529A0 IT 8047529 A0 IT8047529 A0 IT 8047529A0 IT 8047529 A IT8047529 A IT 8047529A IT 4752980 A IT4752980 A IT 4752980A IT 8047529 A0 IT8047529 A0 IT 8047529A0
Authority
IT
Italy
Prior art keywords
acid derivatives
pharmacological properties
epoxysuccinic acid
derivatives equipped
epoxysuccinic
Prior art date
Application number
IT8047529A
Other languages
English (en)
Other versions
IT1188891B (it
IT8047529A1 (it
Inventor
Masaharu Tamai
Adachi Takashi
Morimoto Shigeo
Oguma Kiyoshi
Hanada Kazunori
Omura Sadafumi
Original Assignee
Taisho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taisho Pharmaceutical Co Ltd filed Critical Taisho Pharmaceutical Co Ltd
Publication of IT8047529A0 publication Critical patent/IT8047529A0/it
Publication of IT8047529A1 publication Critical patent/IT8047529A1/it
Application granted granted Critical
Publication of IT1188891B publication Critical patent/IT1188891B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06043—Leu-amino acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
IT47529/80A 1979-02-27 1980-01-07 Derivait di acido epossisuccinico dotati di propireta' farmacologiche IT1188891B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2236579A JPS55115878A (en) 1979-02-27 1979-02-27 Epoxysuccinic acid derivative

Publications (3)

Publication Number Publication Date
IT8047529A0 true IT8047529A0 (it) 1980-01-07
IT8047529A1 IT8047529A1 (it) 1981-07-07
IT1188891B IT1188891B (it) 1988-01-28

Family

ID=12080591

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47529/80A IT1188891B (it) 1979-02-27 1980-01-07 Derivait di acido epossisuccinico dotati di propireta' farmacologiche

Country Status (6)

Country Link
US (2) US4333879A (it)
JP (1) JPS55115878A (it)
DE (1) DE3000628A1 (it)
FR (1) FR2450256A1 (it)
GB (1) GB2046730B (it)
IT (1) IT1188891B (it)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57169478A (en) * 1981-04-10 1982-10-19 Nippon Chemiphar Co Ltd Piperazine derivative
JPS6276A (ja) * 1985-03-26 1987-01-06 Toyo Jozo Co Ltd 酵素阻害性新規物質
US5068354A (en) * 1989-05-18 1991-11-26 Taisho Pharmaceutical Co., Ltd. Epoxysuccinic acid derivatives
CA2047226A1 (en) * 1989-12-27 1991-06-28 Jun-Ichi Haruta 1,3,2-dioxathiolane oxide derivative
JP2808877B2 (ja) * 1990-09-29 1998-10-08 大正製薬株式会社 エポキシスクシナム酸誘導体およびその中間体
JPH04120450U (ja) * 1991-04-16 1992-10-28 エヌオーケー株式会社 水耕栽培装置
EP0641563A4 (en) * 1992-05-20 1995-04-19 Taisho Pharmaceutical Co Ltd MEDICINAL AGAINST CATARACT AND ITS PRODUCTION.
US5556853A (en) * 1993-10-29 1996-09-17 Takeda Chemical Industries, Ltd. Epoxysuccinic acid derivatives
CA2190151A1 (en) * 1994-05-31 1995-12-07 Shigetoshi Tsubotani Epoxysuccinic acid derivatives, their production and use
US5733911A (en) * 1996-01-26 1998-03-31 Hitachi Chemical Co., Ltd. Method for inducing death of neoplastic cells using piperazne derivatives
EP1022276B1 (en) * 1997-09-04 2003-05-28 Nippon Chemiphar Co., Ltd. Epoxysuccinamide derivatives
DE10023430A1 (de) * 2000-05-12 2001-11-15 Bayer Ag Substituierte N-Benzoyl-N'-(tetrazolylphenyl)-harnstoffe
CN100478030C (zh) * 2003-05-08 2009-04-15 北京摩力克科技有限公司 抗传染性非典型性肺炎药物作用靶标及其预防和治疗药物
DE602006020052D1 (de) * 2005-09-28 2011-03-24 Robert Ternansky Neue arzneimittel gegen demenz
AU2007305138A1 (en) * 2006-06-13 2008-04-10 The Board Of Trustees Of The Leland Stanford Junior University Epoxide inhibitors of cysteine proteases
US20100216875A1 (en) * 2006-12-20 2010-08-26 Gregory Hook Methods of treating alzheimer's disease
US9403843B2 (en) 2012-02-01 2016-08-02 The Trustees Of Columbia University In The City Of New York Cysteine protease inhibitors and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS548759B2 (it) * 1973-03-06 1979-04-18
GB1469797A (en) * 1974-11-07 1977-04-06 Pfizer Ltd Antibacterial cephalosporin derivatives
GB1595168A (en) 1977-03-03 1981-08-12 Taisho Pharmaceutical Co Ltd Expoxysuccinic acid derivatives
US4091221A (en) * 1977-03-17 1978-05-23 Shell Oil Company 3-(Benzoyl)oxiranecarboxamides

Also Published As

Publication number Publication date
JPS55115878A (en) 1980-09-06
US4382889A (en) 1983-05-10
US4333879A (en) 1982-06-08
IT1188891B (it) 1988-01-28
FR2450256A1 (fr) 1980-09-26
GB2046730A (en) 1980-11-19
IT8047529A1 (it) 1981-07-07
JPH0154348B2 (it) 1989-11-17
DE3000628C2 (it) 1988-09-08
DE3000628A1 (de) 1980-09-04
GB2046730B (en) 1983-05-05
FR2450256B1 (it) 1983-05-13

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