IT8324207A0 - Carbossamido-derivati di 1,2,4-tiadiazolo [3,2-a] pirimidine e procedimento per la loro preparazione - Google Patents

Carbossamido-derivati di 1,2,4-tiadiazolo [3,2-a] pirimidine e procedimento per la loro preparazione

Info

Publication number
IT8324207A0
IT8324207A0 IT8324207A IT2420783A IT8324207A0 IT 8324207 A0 IT8324207 A0 IT 8324207A0 IT 8324207 A IT8324207 A IT 8324207A IT 2420783 A IT2420783 A IT 2420783A IT 8324207 A0 IT8324207 A0 IT 8324207A0
Authority
IT
Italy
Prior art keywords
carboxamido
pyrimidines
thiadiazole
derivatives
procedure
Prior art date
Application number
IT8324207A
Other languages
English (en)
Other versions
IT1194521B (it
Inventor
Doria Gianfederico
Passarotti Carlo
Buttinoni Ada
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838329746A external-priority patent/GB8329746D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IT8324207A0 publication Critical patent/IT8324207A0/it
Application granted granted Critical
Publication of IT1194521B publication Critical patent/IT1194521B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT24207/83A 1982-12-23 1983-12-16 Carbossamido-derivati di 1,2,4-tiadiazolo (3,2-a) pirimidine e procedimento per la loro preparazione IT1194521B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8236642 1982-12-23
GB838329746A GB8329746D0 (en) 1983-11-08 1983-11-08 Carboxamido-derivatives

Publications (2)

Publication Number Publication Date
IT8324207A0 true IT8324207A0 (it) 1983-12-16
IT1194521B IT1194521B (it) 1988-09-22

Family

ID=26284768

Family Applications (1)

Application Number Title Priority Date Filing Date
IT24207/83A IT1194521B (it) 1982-12-23 1983-12-16 Carbossamido-derivati di 1,2,4-tiadiazolo (3,2-a) pirimidine e procedimento per la loro preparazione

Country Status (15)

Country Link
US (1) US4522944A (it)
AT (1) AT385036B (it)
AU (1) AU558600B2 (it)
CA (1) CA1211440A (it)
CH (1) CH657136A5 (it)
DE (1) DE3346223A1 (it)
DK (1) DK593983A (it)
FI (1) FI834698A7 (it)
FR (1) FR2538392B1 (it)
GR (1) GR79479B (it)
IL (1) IL70522A (it)
IT (1) IT1194521B (it)
NL (1) NL8304340A (it)
SE (1) SE454698B (it)
SU (1) SU1297731A3 (it)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3702758A1 (de) * 1987-01-30 1988-09-29 Hoechst Ag Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
KR102065319B1 (ko) 2007-03-12 2020-01-10 인트라-셀룰라 써래피스, 인코퍼레이티드. 치환된 헤테로환 융합 감마-카르볼린 합성
WO2013155504A1 (en) 2012-04-14 2013-10-17 Intra-Cellular Therapies, Inc. Novel methods
HUE053159T2 (hu) 2013-03-15 2021-06-28 Intra Cellular Therapies Inc Szerves vegyületek
IL305990B2 (en) 2013-12-03 2025-12-01 Intra Cellular Therapies Inc Long-acting injectable composition comprising polymeric microspheres of heterocycle fused gamma-carboline compounds or a pharmaceutical composition for sustained or delayed release comprising the compounds and their use in the treatment of bipolar disorder i and/or bipolar ii disorder
MX365969B (es) 2014-04-04 2019-06-21 Intra Cellular Therapies Inc Gamma-carbolinas fusionadas con heterociclos sustituidas con deuterio.
RU2016143091A (ru) 2014-04-04 2018-05-08 Интра-Селлулар Терапиз, Инк. Органические соединения
CN108883111B (zh) 2016-01-26 2021-10-08 细胞内治疗公司 有机化合物
US11014925B2 (en) 2016-03-28 2021-05-25 Intra-Cellular Therapies, Inc. Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide
JP2019513143A (ja) 2016-03-28 2019-05-23 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 新規塩類および結晶
EP3436083A4 (en) 2016-03-28 2019-11-27 Intra-Cellular Therapies, Inc. NOVEL COMPOSITIONS AND METHOD
US11331316B2 (en) 2016-10-12 2022-05-17 Intra-Cellular Therapies, Inc. Amorphous solid dispersions
US10906906B2 (en) 2016-12-29 2021-02-02 Intra-Cellular Therapies, Inc. Organic compounds
US10961245B2 (en) 2016-12-29 2021-03-30 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines for treatment of central nervous system disorders
IL268970B2 (en) 2017-03-24 2023-12-01 Intra Cellular Therapies Inc Oral transmucosal formulations of substituted heterocycle fused gamma carbolines
JP7224333B2 (ja) 2017-07-26 2023-02-17 イントラ－セルラー・セラピーズ・インコーポレイテッド 有機化合物
JP7223742B2 (ja) 2017-07-26 2023-02-16 イントラ－セルラー・セラピーズ・インコーポレイテッド 有機化合物
AU2019240226B2 (en) 2018-03-23 2024-11-28 Intra-Cellular Therapies, Inc. Organic compounds
IL321985A (en) 2018-06-06 2025-09-01 Intra Cellular Therapies Inc New salts and crystals
WO2019237037A1 (en) 2018-06-08 2019-12-12 Intra-Cellular Therapies, Inc. Novel methods
CA3106447A1 (en) 2018-06-11 2019-12-19 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines synthesis
EP3843729A4 (en) 2018-08-29 2022-06-01 Intra-Cellular Therapies, Inc. NOVEL COMPOSITIONS AND PROCESSES
CA3108558A1 (en) 2018-08-31 2020-03-05 Intra-Cellular Therapies, Inc. Novel methods
CN112584837A (zh) 2018-08-31 2021-03-30 细胞内治疗公司 新方法
JP7673040B2 (ja) 2019-07-07 2025-05-08 イントラ－セルラー・セラピーズ・インコーポレイテッド 新規方法
EP4072554A4 (en) 2019-12-11 2023-12-20 Intra-Cellular Therapies, Inc. ORGANIC CONNECTION
US12414948B2 (en) 2022-05-18 2025-09-16 Intra-Cellular Therapies, Inc. Methods

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5129981B2 (it) * 1973-07-17 1976-08-28
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) * 1979-02-28 1980-09-06 Teijin Ltd 6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) * 1981-02-27 1982-09-03 Dai Ichi Seiyaku Co Ltd Thiazolopyrimidine derivative

Also Published As

Publication number Publication date
SU1297731A3 (ru) 1987-03-15
AU558600B2 (en) 1987-02-05
IL70522A (en) 1986-02-28
CH657136A5 (de) 1986-08-15
SE8307133L (sv) 1984-06-24
SE8307133D0 (sv) 1983-12-22
FI834698A7 (fi) 1984-06-24
IT1194521B (it) 1988-09-22
DK593983D0 (da) 1983-12-22
NL8304340A (nl) 1984-07-16
FR2538392A1 (fr) 1984-06-29
US4522944A (en) 1985-06-11
FR2538392B1 (fr) 1987-01-16
GR79479B (it) 1984-10-30
IL70522A0 (en) 1984-03-30
SE454698B (sv) 1988-05-24
DE3346223A1 (de) 1984-06-28
ATA438383A (de) 1987-07-15
AT385036B (de) 1988-02-10
CA1211440A (en) 1986-09-16
FI834698A0 (fi) 1983-12-20
AU2252583A (en) 1984-06-28
DK593983A (da) 1984-06-24

Similar Documents

Publication Publication Date Title
IT8324207A0 (it) Carbossamido-derivati di 1,2,4-tiadiazolo [3,2-a] pirimidine e procedimento per la loro preparazione
ES546484A0 (es) Procedimiento para la preparacion de derivados de furazano
IT8320024A0 (it) 1h-pirazolo [1,5-a] pirimidine sostituite e procedimento per la loro preparazione
ES522886A0 (es) "procedimiento para la preparacion de derivados de 1-sulfo-2-oxoacetidina"
IT8548301A0 (it) Procedimento per la preparazione di xantoni e di tioxantoni
ES549119A0 (es) Procedimiento para la preparacion de silibinina exenta de isosilibina
IT8521570A0 (it) Procedimento di preparazione di microlattici invertiti ed i microlattici invertiti ottenuti.
IT8222353A0 (it) Tiazolo [3,2-a]pirimidine sostituite e procedimento per la loro preparazione
IT1200400B (it) Procedimento per la preparazione di 2-alchil ciclopent-2-enoni
IT8567535A0 (it) Procedimento per la preparazione di amminoidrossicefamcarbossilati
ES527201A0 (es) Procedimiento para la preparacion de derivados heterociclicos de fenilsulfonil-n'-pirimidinil- y -triacinil-ureas
IT1206115B (it) Iminoderivati di diidrobenzopirano e diidrobenzotiopirano sostituiti e procedimento per la loro preparazione.
MX161035A (es) Procedimiento para la preparacion de imidazo(1,2-a)quinolinas
IT8319192A0 (it) 1,3,4-tiadiazolo [3,2-a] pirimidine sostituite e procedimento per laloro preparazione
IT1200594B (it) Procedimento per la preparazione di alfa-omega-aloperfluorocarburi
ES546908A0 (es) Procedimiento para la preparacion de derivados de fenilace- tonitrilo
ES531159A0 (es) Procedimiento para la preparacion de aminociclotiadiazinas
IT1190358B (it) Procedimento per la preparazione di l-carnitina
IT1191806B (it) Procedimento per la preparazione di 2-bromo-alfa-ergocriptina
ES556590A0 (es) Procedimiento para la obtencion de derivados de piridazo(1,2-a)(1,2)diacepina
IT1222755B (it) Procedimento per la preparazione di idantoine 5-ariliden e alchiliden sostituite
MX7420E (es) Procedimiento para la preparacion de carbamoil-lactama-n-substituida
IT8822858A0 (it) Composizioni per la riduzione di flebectasie e procedimento per la loro preparazione
IT1200399B (it) 1-nor-2-idrossi-metil-derivati di carboprostacicline e procedimento per la loro preparazione
ES549829A0 (es) Procedimiento para la preparacion de carbazatos