IT8320024A0 - 1h-pirazolo [1,5-a] pirimidine sostituite e procedimento per la loro preparazione - Google Patents

1h-pirazolo [1,5-a] pirimidine sostituite e procedimento per la loro preparazione

Info

Publication number
IT8320024A0
IT8320024A0 IT8320024A IT2002483A IT8320024A0 IT 8320024 A0 IT8320024 A0 IT 8320024A0 IT 8320024 A IT8320024 A IT 8320024A IT 2002483 A IT2002483 A IT 2002483A IT 8320024 A0 IT8320024 A0 IT 8320024A0
Authority
IT
Italy
Prior art keywords
pyrazole
procedure
preparation
substituted pyrimidines
pyrimidines
Prior art date
Application number
IT8320024A
Other languages
English (en)
Other versions
IT1194555B (it
Inventor
Gianfederico Doria
Carlo Passarotti
Ada Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838303089A external-priority patent/GB8303089D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IT8320024A0 publication Critical patent/IT8320024A0/it
Application granted granted Critical
Publication of IT1194555B publication Critical patent/IT1194555B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT20024/83A 1982-03-16 1983-03-11 1h-pirazolo (1,5-a) pirimidine sostituite e procedimento per la loro preparazione IT1194555B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8207637 1982-03-16
GB838303089A GB8303089D0 (en) 1983-02-04 1983-02-04 Substituted 1h-pyrazolo 1,5-a pyrimidines

Publications (2)

Publication Number Publication Date
IT8320024A0 true IT8320024A0 (it) 1983-03-11
IT1194555B IT1194555B (it) 1988-09-22

Family

ID=26282260

Family Applications (1)

Application Number Title Priority Date Filing Date
IT20024/83A IT1194555B (it) 1982-03-16 1983-03-11 1h-pirazolo (1,5-a) pirimidine sostituite e procedimento per la loro preparazione

Country Status (13)

Country Link
US (1) US4482555A (it)
AU (1) AU557300B2 (it)
CA (1) CA1192546A (it)
CH (1) CH654306A5 (it)
DE (1) DE3309432A1 (it)
DK (1) DK120783A (it)
FI (1) FI74469C (it)
FR (1) FR2523582B1 (it)
IL (1) IL68133A (it)
IT (1) IT1194555B (it)
NL (1) NL8300934A (it)
SE (1) SE450573B (it)
SU (1) SU1366060A3 (it)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USD344263S (en) 1991-11-15 1994-02-15 Masami Seido Plug-receiving metal fitting
RU2147584C1 (ru) * 1995-10-27 2000-04-20 Американ Цианамид Компани Способ получения дигалоидазолопиримидинов и способ получения дигидроксиазолопиримидинов
US6245759B1 (en) 1999-03-11 2001-06-12 Merck & Co., Inc. Tyrosine kinase inhibitors
MY125533A (en) 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
EP1782859A3 (en) * 2003-04-11 2009-09-30 High Point Pharmaceuticals, LLC Pharmaceutical use of substituted pyrazolo [1,5- a]pyrimidines
WO2004089471A2 (en) * 2003-04-11 2004-10-21 Novo Nordisk A/S NEW PYRAZOLO[1,5-a] PYRIMIDINES DERIVATIVES AND PHARMACEUTICAL USE THEREOF
US7772232B2 (en) 2004-04-15 2010-08-10 Bristol-Myers Squibb Company Quinazolinyl compounds as inhibitors of potassium channel function
US8138342B2 (en) * 2004-10-12 2012-03-20 High Point Pharmacueticals, LLC 11β-hydroxysteroid dehydrogenase type 1 active spiro compounds
JP2009513611A (ja) * 2005-11-01 2009-04-02 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 置換アミドの医薬用途
KR20080076916A (ko) * 2005-11-01 2008-08-20 트랜스테크 파르마, 인크. 치환된 아미드의 약학적 사용
EP2007722A1 (en) * 2006-03-21 2008-12-31 High Point Pharmaceuticals, LLC Adamantane derivatives for the treatment of the metabolic syndrome
KR20090014347A (ko) 2006-04-07 2009-02-10 하이 포인트 파마슈티칼스, 엘엘씨 11β-히드록시스테로이드 탈수소효소 타입 1 활성 화합물
JP2009539937A (ja) * 2006-06-16 2009-11-19 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 置換型ピペリジンカルボキサミドの医薬的使用
US8048908B2 (en) * 2006-07-13 2011-11-01 High Point Pharmaceuticals, Llc 11β-hydroxysteroid dehydrogenase type 1 active compounds
EP1878721A1 (en) * 2006-07-13 2008-01-16 Novo Nordisk A/S 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
US8334305B2 (en) * 2007-02-23 2012-12-18 High Point Pharmaceuticals, Llc N-adamantyl benzamides as inhibitors of 11-β-hydroxysteroid dehydrogenase
CA2675669C (en) * 2007-02-23 2015-05-26 High Point Pharmaceuticals, Llc Novel compounds
EP2125704A1 (en) * 2007-02-23 2009-12-02 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
WO2008101885A1 (en) * 2007-02-23 2008-08-28 High Point Pharmaceuticals, Llc N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
CN101652359A (zh) * 2007-03-09 2010-02-17 高点制药有限责任公司 作为羟类固醇脱氢酶抑制剂的吲哚-和苯并咪唑酰胺类
CA2681934A1 (en) * 2007-03-28 2008-10-02 High Point Pharmaceuticals, Llc 11beta-hsd1 active compounds
WO2008127924A1 (en) * 2007-04-11 2008-10-23 High Point Pharmaceuticals, Llc. Novel compounds
US8383683B2 (en) * 2007-04-24 2013-02-26 High Point Pharmaceuticals, Llc Pharmaceutical use of substituted amides

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
BE786611A (fr) * 1971-08-16 1973-01-22 Int Chem & Nuclear Corp Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio
US3925385A (en) * 1972-04-20 1975-12-09 Icn Pharmaceuticals 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
BE792533A (fr) * 1971-12-09 1973-06-08 Int Chem & Nuclear Corp Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US4093617A (en) * 1974-11-12 1978-06-06 Icn Pharmaceuticals, Inc. 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4048184A (en) * 1976-11-15 1977-09-13 E. R. Squibb & Sons, Inc. 6-Phenyl-2H-pyrazolo[3,4-b]pyridines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

Also Published As

Publication number Publication date
IL68133A (en) 1985-12-31
US4482555A (en) 1984-11-13
AU1230483A (en) 1983-09-22
FI830864L (fi) 1983-09-17
FI74469C (fi) 1988-02-08
IT1194555B (it) 1988-09-22
SE450573B (sv) 1987-07-06
NL8300934A (nl) 1983-10-17
AU557300B2 (en) 1986-12-18
FR2523582B1 (fr) 1985-12-06
DK120783A (da) 1983-09-17
FI830864A0 (fi) 1983-03-15
FI74469B (fi) 1987-10-30
CH654306A5 (de) 1986-02-14
SE8301412L (sv) 1983-09-17
SE8301412D0 (sv) 1983-03-15
CA1192546A (en) 1985-08-27
DK120783D0 (da) 1983-03-15
DE3309432A1 (de) 1983-09-22
IL68133A0 (en) 1983-06-15
FR2523582A1 (fr) 1983-09-23
SU1366060A3 (ru) 1988-01-07

Similar Documents

Publication Publication Date Title
IT8324207A0 (it) Carbossamido-derivati di 1,2,4-tiadiazolo [3,2-a] pirimidine e procedimento per la loro preparazione
IT1194555B (it) 1h-pirazolo (1,5-a) pirimidine sostituite e procedimento per la loro preparazione
IT8322837A0 (it) Cefem-derivati e procedimenti per la loro preparazione.
FI981709L (fi) Menetelmä 5-substituoitujen 2-amino-4-okso-pyrrolo/2,3-d/-pyrimidiinien valmistamiseksi
AR240926A1 (es) "procedimiento para la preparacion de 8-isopropil-6-dimetilamino metil-7-hidroxi-4-metil-cumarina".
ZA835338B (en) New 5-oxo-2,3,6,7-tetrahydro-5h-thiazolo/3,2-a/pyrimidine derivatives,their preparation and their use as herbicides
IT8423392A0 (it) Cefem composti e procedimenti per la loro preparazione.
IT8222353A0 (it) Tiazolo [3,2-a]pirimidine sostituite e procedimento per la loro preparazione
MX161035A (es) Procedimiento para la preparacion de imidazo(1,2-a)quinolinas
IT1193604B (it) 1,3,4-tiadiazolo (3,2-a) pirimidine sostituite e procedimento per la loro preparazione
IT1230584B (it) Isopolipeptidi e procedimento per la loro preparazione
GB2138418B (en) Novel s-triazole(1,5-a)pyrimidine derivatives
ES529131A0 (es) Procedimiento de obtencion de derivados de piracino (2', 3'-3, 4)pirido(1, 2-a)indol
IT8522317A0 (it) Carbapenem antibiotici eprocedimento per la loro preparazione.
IT8423805A0 (it) Composti azabiciclici e procedimenti per la loro preparazione.
PH22448A (en) Substituted carboxy-thiazolo/3,2-a/pyrimidine derivatives
IT8719009A0 (it) Composti antagonisti di recettori -h2 e procedimento per la loro preparazione.
GB8409424D0 (en) 1h,7h-pyrazolo(1'5-a)pyrimidine-7-one derivatives
IT1176376B (it) Procedimento per la preparazione di 3, 11-dimepil-2-nonacosanone
IT1201442B (it) Alchilsolfonipropeni,procedimento per la loro preparazione e loro impiego
IT8322499A0 (it) Cianalchilpiperazine procedimenti per la loro preparazione e loro impiego.
IT1210971B (it) Composti biciclici eprocedimento per la loro preparazione.
IT1141028B (it) Procedimento per la preparazione di 2,5-dimetil 2,4-esadiene
IT1200399B (it) 1-nor-2-idrossi-metil-derivati di carboprostacicline e procedimento per la loro preparazione
IT1174498B (it) Isossazoli e procedimento per la loro preparazione