ATA438383A - Verfahren zum herstellen von neuen carboxamidoderivaten von 5h-1,3,4-thiadiazolo(3,2-a)-pyrimidinen und ihren pharmazeutisch unbedenklichen salzen - Google Patents

Verfahren zum herstellen von neuen carboxamidoderivaten von 5h-1,3,4-thiadiazolo(3,2-a)-pyrimidinen und ihren pharmazeutisch unbedenklichen salzen

Info

Publication number: ATA438383A
Authority: AT; Austria
Prior art keywords: thiadiazolo; pyrimidines; producing new; pharmaceutically safe; safe salts
Prior art date: 1982-12-23

Application number

AT0438383A

Other languages

English (en)

Other versions

AT385036B (de

Inventor

Doria Gianfederico

Carlo Passarotti

Ada Buttinoni

Original Assignee

Erba Farmitalia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-12-23

Filing date

1983-12-15

Publication date

1987-07-15

1983-11-08 Priority claimed from GB838329746A external-priority patent/GB8329746D0/en

1983-12-15 Application filed by Erba Farmitalia filed Critical Erba Farmitalia

1987-07-15 Publication of ATA438383A publication Critical patent/ATA438383A/de

1988-02-10 Application granted granted Critical

1988-02-10 Publication of AT385036B publication Critical patent/AT385036B/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT0438383A 1982-12-23 1983-12-15 Verfahren zum herstellen von neuen carboxamidoderivaten von 5h-1,3,4-thiadiazolo(3,2-a)-pyrimidinen und ihren pharmazeutisch unbedenklichen salzen AT385036B (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8236642		1982-12-23
GB838329746A GB8329746D0 (en)	1983-11-08	1983-11-08	Carboxamido-derivatives

Publications (2)

Publication Number	Publication Date
ATA438383A true ATA438383A (de)	1987-07-15
AT385036B AT385036B (de)	1988-02-10

Family

ID=26284768

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT0438383A AT385036B (de)	1982-12-23	1983-12-15	Verfahren zum herstellen von neuen carboxamidoderivaten von 5h-1,3,4-thiadiazolo(3,2-a)-pyrimidinen und ihren pharmazeutisch unbedenklichen salzen

Country Status (15)

Country	Link
US (1)	US4522944A (de)
AT (1)	AT385036B (de)
AU (1)	AU558600B2 (de)
CA (1)	CA1211440A (de)
CH (1)	CH657136A5 (de)
DE (1)	DE3346223A1 (de)
DK (1)	DK593983A (de)
FI (1)	FI834698A7 (de)
FR (1)	FR2538392B1 (de)
GR (1)	GR79479B (de)
IL (1)	IL70522A (de)
IT (1)	IT1194521B (de)
NL (1)	NL8304340A (de)
SE (1)	SE454698B (de)
SU (1)	SU1297731A3 (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3702758A1 (de) *	1987-01-30	1988-09-29	Hoechst Ag	Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
CA2679754C (en)	2007-03-12	2018-08-07	Intra-Cellular Therapies, Inc.	Substituted heterocycle fused gamma-carbolines synthesis
JP2015514135A (ja)	2012-04-14	2015-05-18	イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−ＣｅｌｌｕｌａｒＴｈｅｒａｐｉｅｓ，Ｉｎｃ．	新規組成物および方法
DK2968320T3 (da)	2013-03-15	2021-02-01	Intra Cellular Therapies Inc	Organiske forbindelser
CA3148303C (en)	2013-12-03	2024-02-27	Intra-Cellular Therapies, Inc.	Heterocycle fused gamma-carboline compounds for use in treatment of bipolar disorders
CA2944512C (en)	2014-04-04	2018-04-24	Intra-Cellular Therapies, Inc.	Heterocycle fused gamma-carbolines for treatment of central nervous system disorders
CA2944755A1 (en)	2014-04-04	2015-10-08	Intra-Cellular Therapies, Inc.	Organic compounds
PT3407888T (pt)	2016-01-26	2021-03-19	Intra Cellular Therapies Inc	Compostos de piridopirroloquinoxalina, suas composições e utilizações
US10682354B2 (en)	2016-03-28	2020-06-16	Intra-Cellular Therapies, Inc.	Compositions and methods
EP3436016B1 (de)	2016-03-28	2022-04-27	Intra-Cellular Therapies, Inc.	Neuartige co-kristalle
EP3436455A4 (de)	2016-03-28	2019-09-04	Intra-Cellular Therapies, Inc.	Neuartige salze und kristalle
JP7013454B2 (ja)	2016-10-12	2022-02-15	イントラ－セルラー・セラピーズ・インコーポレイテッド	アモルファス固体分散体
WO2018126140A1 (en)	2016-12-29	2018-07-05	Intra-Cellular Therapies, Inc.	Organic compounds
WO2018126143A1 (en)	2016-12-29	2018-07-05	Intra-Cellular Therapies, Inc.	Organic compounds
IL304026B2 (en)	2017-03-24	2024-11-01	Intra Cellular Therapies Inc	A pharmaceutical preparation containing 1-(4-fluoro-phenyl)-4-((Sa10,Rb6)-3-D2-2,2-methyl-2, 3, a10, 10, 9, b6- hexahydro-H7, H1- Pyrido[3',4',:4,5]pyrrolo[3,2,1-de]quioxalin-8-yl)-butan-1-one and its uses
JP7223742B2 (ja)	2017-07-26	2023-02-16	イントラ－セルラー・セラピーズ・インコーポレイテッド	有機化合物
US11427587B2 (en)	2017-07-26	2022-08-30	Intra-Cellular Therapies, Inc.	Organic compounds
IL277504B1 (en)	2018-03-23	2026-02-01	Intra Cellular Therapies Inc	Deuterium-converted ((sa10,rb6)-8-(3-(4-fluorophenoxy)propyl 6b, 7, 8, 9, 10, 10a-hexahydro-1h-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-82(h3)-one compounds, pharmaceutical composition containing them and their uses
JP7476115B2 (ja)	2018-06-06	2024-04-30	イントラ－セルラー・セラピーズ・インコーポレイテッド	新規の塩および結晶
WO2019237037A1 (en)	2018-06-08	2019-12-12	Intra-Cellular Therapies, Inc.	Novel methods
DK3609891T3 (da)	2018-06-11	2026-02-23	Intra Cellular Therapies Inc	Syntese af substituerede heterocykliske fusionerede gamma-carboliner
US12144808B2 (en)	2018-08-29	2024-11-19	Intra-Cellular Therapies, Inc.	Compositions and methods
MX2021002321A (es)	2018-08-31	2021-04-28	Intra Cellular Therapies Inc	Nuevos metodos.
AU2019328528B2 (en)	2018-08-31	2025-01-23	Intra-Cellular Therapies, Inc.	Novel methods
CN114072150A (zh)	2019-07-07	2022-02-18	细胞内治疗公司	新方法
EP4072554A4 (de)	2019-12-11	2023-12-20	Intra-Cellular Therapies, Inc.	Organische verbindung
US12414948B2 (en)	2022-05-18	2025-09-16	Intra-Cellular Therapies, Inc.	Methods

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5129981B2 (de) *	1973-07-17	1976-08-28
GB1568962A (en) *	1975-10-31	1980-06-11	Beecham Group Ltd	Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) *	1979-02-28	1980-09-06	Teijin Ltd	6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) *	1981-02-27	1982-09-03	Dai Ichi Seiyaku Co Ltd	Thiazolopyrimidine derivative

1983
- 1983-12-08 US US06/559,322 patent/US4522944A/en not_active Expired - Fee Related
- 1983-12-15 AT AT0438383A patent/AT385036B/de not_active IP Right Cessation
- 1983-12-15 GR GR73259A patent/GR79479B/el unknown
- 1983-12-16 IT IT24207/83A patent/IT1194521B/it active
- 1983-12-16 NL NL8304340A patent/NL8304340A/nl not_active Application Discontinuation
- 1983-12-19 AU AU22525/83A patent/AU558600B2/en not_active Ceased
- 1983-12-20 CH CH6783/83A patent/CH657136A5/de not_active IP Right Cessation
- 1983-12-20 FI FI834698A patent/FI834698A7/fi not_active Application Discontinuation
- 1983-12-21 DE DE19833346223 patent/DE3346223A1/de not_active Withdrawn
- 1983-12-22 DK DK593983A patent/DK593983A/da not_active Application Discontinuation
- 1983-12-22 SU SU833682101A patent/SU1297731A3/ru active
- 1983-12-22 SE SE8307133A patent/SE454698B/sv not_active IP Right Cessation
- 1983-12-22 CA CA000444151A patent/CA1211440A/en not_active Expired
- 1983-12-22 IL IL70522A patent/IL70522A/xx not_active IP Right Cessation
- 1983-12-23 FR FR8320704A patent/FR2538392B1/fr not_active Expired

Also Published As

Publication number	Publication date
SU1297731A3 (ru)	1987-03-15
AU558600B2 (en)	1987-02-05
US4522944A (en)	1985-06-11
FR2538392B1 (fr)	1987-01-16
IL70522A (en)	1986-02-28
AU2252583A (en)	1984-06-28
NL8304340A (nl)	1984-07-16
DK593983D0 (da)	1983-12-22
CA1211440A (en)	1986-09-16
CH657136A5 (de)	1986-08-15
DE3346223A1 (de)	1984-06-28
IT8324207A0 (it)	1983-12-16
GR79479B (de)	1984-10-30
IL70522A0 (en)	1984-03-30
FI834698A0 (fi)	1983-12-20
SE454698B (sv)	1988-05-24
FR2538392A1 (fr)	1984-06-29
FI834698A7 (fi)	1984-06-24
AT385036B (de)	1988-02-10
IT1194521B (it)	1988-09-22
SE8307133D0 (sv)	1983-12-22
SE8307133L (sv)	1984-06-24
DK593983A (da)	1984-06-24

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Legal Events

Date	Code	Title	Description
1991-04-15	ELJ	Ceased due to non-payment of the annual fee