ITMI20032044A1 - Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica - Google Patents

Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica

Info

Publication number
ITMI20032044A1
ITMI20032044A1 IT002044A ITMI20032044A ITMI20032044A1 IT MI20032044 A1 ITMI20032044 A1 IT MI20032044A1 IT 002044 A IT002044 A IT 002044A IT MI20032044 A ITMI20032044 A IT MI20032044A IT MI20032044 A1 ITMI20032044 A1 IT MI20032044A1
Authority
IT
Italy
Prior art keywords
chinolizidinilalchil
chinolizidinil
antimalaric
chinoline
derivatives
Prior art date
Application number
IT002044A
Other languages
English (en)
Inventor
Vito Boido
Boido Caterina Canu
Anna Sparatone
Anna Sparatore
Fabio Sparatore
Donatella Taramelli
Original Assignee
Univ Degli Studi Milano
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Degli Studi Milano filed Critical Univ Degli Studi Milano
Priority to IT002044A priority Critical patent/ITMI20032044A1/it
Priority to AT04791711T priority patent/ATE417044T1/de
Priority to AP2006003616A priority patent/AP2006003616A0/xx
Priority to ES04791711T priority patent/ES2319201T3/es
Priority to DE602004018355T priority patent/DE602004018355D1/de
Priority to CNA2004800381525A priority patent/CN1902199A/zh
Priority to EP04791711A priority patent/EP1675855B1/en
Priority to PCT/IB2004/003393 priority patent/WO2005037833A1/en
Publication of ITMI20032044A1 publication Critical patent/ITMI20032044A1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0046Ruthenium compounds
    • C07F15/0053Ruthenium compounds without a metal-carbon linkage
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0073Rhodium compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/60Quinoline or hydrogenated quinoline ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT002044A 2003-10-21 2003-10-21 Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica ITMI20032044A1 (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT002044A ITMI20032044A1 (it) 2003-10-21 2003-10-21 Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica
AT04791711T ATE417044T1 (de) 2003-10-21 2004-10-18 4-amino-chinolin-, -chinolizidinyl- und - chinolizidinylalkylderivate mit antimalariawirkung
AP2006003616A AP2006003616A0 (en) 2003-10-21 2004-10-18 4-amino-quinoline quinolizidinyl and quinolizidinylalkyl derivatives with antimalarial activity
ES04791711T ES2319201T3 (es) 2003-10-21 2004-10-18 Quinolizidinil-y quinolizidinilalquil-derivados de 4-amino-quinolina con actividad antipaludica.
DE602004018355T DE602004018355D1 (de) 2003-10-21 2004-10-18 4-amino-chinolin-, -chinolizidinyl- und -chinolizidinylalkylderivate mit antimalariawirkung
CNA2004800381525A CN1902199A (zh) 2003-10-21 2004-10-18 有抗疟活性的4-氨基-喹啉喹嗪啶基-和喹嗪啶烷基-衍生物
EP04791711A EP1675855B1 (en) 2003-10-21 2004-10-18 4-amino-quinoline ouinolizidinyl-and quinolizidinylalkyl-derivatives with antimalarial activity
PCT/IB2004/003393 WO2005037833A1 (en) 2003-10-21 2004-10-18 4-amino-quinoline ouinolizidinyl-and quinolizidinylalkyl-derivatives with antimalarial activity

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002044A ITMI20032044A1 (it) 2003-10-21 2003-10-21 Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica

Publications (1)

Publication Number Publication Date
ITMI20032044A1 true ITMI20032044A1 (it) 2005-04-22

Family

ID=34452253

Family Applications (1)

Application Number Title Priority Date Filing Date
IT002044A ITMI20032044A1 (it) 2003-10-21 2003-10-21 Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica

Country Status (8)

Country Link
EP (1) EP1675855B1 (it)
CN (1) CN1902199A (it)
AP (1) AP2006003616A0 (it)
AT (1) ATE417044T1 (it)
DE (1) DE602004018355D1 (it)
ES (1) ES2319201T3 (it)
IT (1) ITMI20032044A1 (it)
WO (1) WO2005037833A1 (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006082030A1 (en) * 2005-02-04 2006-08-10 Ctg Pharma S.R.L. New 4-aminoquinoline derivatives as antimalarials
ITMI20052008A1 (it) * 2005-10-21 2007-04-22 Ctg Pharma S R L Nuovi antimalarici derivati della 4-aminochinolina

Also Published As

Publication number Publication date
DE602004018355D1 (de) 2009-01-22
ATE417044T1 (de) 2008-12-15
ES2319201T3 (es) 2009-05-05
WO2005037833A1 (en) 2005-04-28
CN1902199A (zh) 2007-01-24
AP2006003616A0 (en) 2006-06-30
EP1675855A1 (en) 2006-07-05
EP1675855B1 (en) 2008-12-10

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