JO3250B1 - إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 - Google Patents

إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7

Info

Publication number
JO3250B1
JO3250B1 JOP/2010/0321A JOP20100321A JO3250B1 JO 3250 B1 JO3250 B1 JO 3250B1 JO P20100321 A JOP20100321 A JO P20100321A JO 3250 B1 JO3250 B1 JO 3250B1
Authority
JO
Jordan
Prior art keywords
activators
acetylcholine receptor
nicotinic acetylcholine
receptor alpha
dopamine
Prior art date
Application number
JOP/2010/0321A
Other languages
English (en)
Inventor
Gomez-Mancilla Baltazar
Di Paolo Therese
Feuerbach Dominik
Johns Donald
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42990156&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JO3250(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of JO3250B1 publication Critical patent/JO3250B1/ar

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

يتعلق الإختراع بإستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 لمعالجة أو منع أو تأخير تعاقب علاج صعوبة الحركة المرتبطة بناهضة الدوبامين في مرض باركنسون.
JOP/2010/0321A 2009-09-22 2010-09-21 إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 JO3250B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24465809P 2009-09-22 2009-09-22

Publications (1)

Publication Number Publication Date
JO3250B1 true JO3250B1 (ar) 2018-09-16

Family

ID=42990156

Family Applications (1)

Application Number Title Priority Date Filing Date
JOP/2010/0321A JO3250B1 (ar) 2009-09-22 2010-09-21 إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7

Country Status (22)

Country Link
US (3) US10537539B2 (ar)
EP (1) EP2480228B1 (ar)
JP (2) JP6178074B2 (ar)
KR (1) KR20120068878A (ar)
CN (1) CN102573830A (ar)
AU (1) AU2010299967B2 (ar)
BR (1) BR112012006346A2 (ar)
CA (1) CA2774801C (ar)
CL (1) CL2012000702A1 (ar)
EA (1) EA036742B1 (ar)
ES (1) ES2614930T3 (ar)
IL (1) IL218299A (ar)
JO (1) JO3250B1 (ar)
MA (1) MA33590B1 (ar)
MX (1) MX359011B (ar)
NZ (1) NZ598316A (ar)
PH (1) PH12012500554A1 (ar)
SG (1) SG178832A1 (ar)
TN (1) TN2012000082A1 (ar)
TW (1) TWI558398B (ar)
WO (1) WO2011036167A1 (ar)
ZA (1) ZA201201066B (ar)

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