JOP20170099B1 - شكل متعدد الأشكال من n-{6-(2-هيدروكسي بروبان-2-يل)-2-[2-(مثيل سلفونيل) إثيل]-2h-إندازول-5-يل}-6-(ثلاثي فلورومثيل) بيريدين-2-كربوكساميد - Google Patents

شكل متعدد الأشكال من n-{6-(2-هيدروكسي بروبان-2-يل)-2-[2-(مثيل سلفونيل) إثيل]-2h-إندازول-5-يل}-6-(ثلاثي فلورومثيل) بيريدين-2-كربوكساميد

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Publication number
JOP20170099B1
JOP20170099B1 JOP/2017/0099A JOP20170099A JOP20170099B1 JO P20170099 B1 JOP20170099 B1 JO P20170099B1 JO P20170099 A JOP20170099 A JO P20170099A JO P20170099 B1 JOP20170099 B1 JO P20170099B1
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Jordan
Prior art keywords
carboxamide
trifluoromethyl
pyridine
ethyl
hydroxypropane
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JOP/2017/0099A
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English (en)
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Thaler Tobias
Platzek Johannes
GUIMOND Nicolas
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Bayer Pharma AG
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Abstract

يتعلق الاختراع الحالي بأشكال بلورية من N-{6-(2-Hydroxypropan-2-yl)-2-[2-(methylsulphonyl)ethyl]-2H-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide، وبعمليات لتحضيرها، وبتركيبات صيدلية تشملها وباستخدامها في مكافحة الاضطرابات.
JOP/2017/0099A 2016-04-29 2017-04-27 شكل متعدد الأشكال من n-{6-(2-هيدروكسي بروبان-2-يل)-2-[2-(مثيل سلفونيل) إثيل]-2h-إندازول-5-يل}-6-(ثلاثي فلورومثيل) بيريدين-2-كربوكساميد JOP20170099B1 (ar)

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JOP/2017/0100A JOP20170100B1 (ar) 2016-04-29 2017-04-27 توليف مركبات إندازول
JOP/2017/0099A JOP20170099B1 (ar) 2016-04-29 2017-04-27 شكل متعدد الأشكال من n-{6-(2-هيدروكسي بروبان-2-يل)-2-[2-(مثيل سلفونيل) إثيل]-2h-إندازول-5-يل}-6-(ثلاثي فلورومثيل) بيريدين-2-كربوكساميد

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