JP5039268B2 - ベンゾイミダゾールおよび類縁体および蛋白キナーゼ阻害剤としてのその使用 - Google Patents

ベンゾイミダゾールおよび類縁体および蛋白キナーゼ阻害剤としてのその使用 Download PDF

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JP5039268B2
JP5039268B2 JP2003537632A JP2003537632A JP5039268B2 JP 5039268 B2 JP5039268 B2 JP 5039268B2 JP 2003537632 A JP2003537632 A JP 2003537632A JP 2003537632 A JP2003537632 A JP 2003537632A JP 5039268 B2 JP5039268 B2 JP 5039268B2
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Japan
Prior art keywords
benzimidazol
indazol
carboxylic acid
benzimidazole
amide
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Expired - Fee Related
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JP2003537632A
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Japanese (ja)
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JP2005509633A5 (fr
JP2005509633A (ja
Inventor
マイクル・ルイス・エドワーズ
ポール・ジョゼフ・コックス
シェリー・アーメンドーラ
ステファニー・ダニエル・デプレ
ティモシー・アラン・ギレスピー
クリストファー・デイヴィッド・エドリン
アンドルー・デイヴィッド・モーリー
チャールズ・ジェイ・ガードナー
ブライアン・ペドグリフト
エルヴェ・ブーシャール
ディディエ・ババン
ローラン・ゴージ
アレン・ルブラン
ターヒール・ネデーム・マジド
ジョン・シー・リーダー
ロイド・ジェイ・ペイン
ナワズ・エム・カーン
マイクル・チェリー
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アベンティス・ファーマスーティカルズ・インコーポレイテツド
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Priority claimed from FR0113868A external-priority patent/FR2831537B1/fr
Priority claimed from GB0206895A external-priority patent/GB0206895D0/en
Priority claimed from GB0206893A external-priority patent/GB0206893D0/en
Application filed by アベンティス・ファーマスーティカルズ・インコーポレイテツド filed Critical アベンティス・ファーマスーティカルズ・インコーポレイテツド
Publication of JP2005509633A publication Critical patent/JP2005509633A/ja
Publication of JP2005509633A5 publication Critical patent/JP2005509633A5/ja
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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JP2003537632A 2001-10-26 2002-10-24 ベンゾイミダゾールおよび類縁体および蛋白キナーゼ阻害剤としてのその使用 Expired - Fee Related JP5039268B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
FR0113868A FR2831537B1 (fr) 2001-10-26 2001-10-26 Nouveaux derives de benzimidazoles, leur procede de preparation, leur application a titre de medicament, compositions pharmaceutiques et nouvelle utilisation
FR01/13868 2001-10-26
GB0206895A GB0206895D0 (en) 2002-03-22 2002-03-22 Chemical compounds
GB0206895.5 2002-03-22
GB0206893.0 2002-03-22
GB0206893A GB0206893D0 (en) 2002-03-22 2002-03-22 Chemical compounds
US39506002P 2002-07-11 2002-07-11
US39515102P 2002-07-11 2002-07-11
US60/395,060 2002-07-11
US60/395,151 2002-07-11
PCT/GB2002/004763 WO2003035065A1 (fr) 2001-10-26 2002-10-24 Benzimidazoles et analogues et leur utilisation comme inhibiteurs de proteines kinases

Publications (3)

Publication Number Publication Date
JP2005509633A JP2005509633A (ja) 2005-04-14
JP2005509633A5 JP2005509633A5 (fr) 2012-07-12
JP5039268B2 true JP5039268B2 (ja) 2012-10-03

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JP2003537632A Expired - Fee Related JP5039268B2 (ja) 2001-10-26 2002-10-24 ベンゾイミダゾールおよび類縁体および蛋白キナーゼ阻害剤としてのその使用

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EP (1) EP1441725A1 (fr)
JP (1) JP5039268B2 (fr)
AU (1) AU2002334217B2 (fr)
BR (1) BR0213562A (fr)
CA (1) CA2465247C (fr)
IL (1) IL161576A0 (fr)
MX (1) MXPA04003954A (fr)
UY (1) UY27516A1 (fr)
WO (1) WO2003035065A1 (fr)

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JP2023526548A (ja) * 2020-05-22 2023-06-21 シャンハイ ロングウッド バイオファルマシューティカルズ カンパニー リミテッド 新規三環芳香族複素環化合物、ならびにその調製方法、医薬組成物および適用

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IL161576A0 (en) 2004-09-27
CA2465247C (fr) 2010-05-18
BR0213562A (pt) 2004-08-31
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