JPH0215097A - ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法 - Google Patents

ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法

Info

Publication number
JPH0215097A
JPH0215097A JP1115265A JP11526589A JPH0215097A JP H0215097 A JPH0215097 A JP H0215097A JP 1115265 A JP1115265 A JP 1115265A JP 11526589 A JP11526589 A JP 11526589A JP H0215097 A JPH0215097 A JP H0215097A
Authority
JP
Japan
Prior art keywords
group
derivative
general formula
drug
amino acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1115265A
Other languages
English (en)
Japanese (ja)
Inventor
Gyoergy Keri
ジェルジ ケーリ
Robert I Nicholson
ロバート アイ ニコルソン
Istvan Teplan
イシュトワーン テプラーン
Tamas Gulyas
タマーシュ グイヤーシュ
Aniko Horvath
アニコー ホルヴァート
Gyoergy Boekoenyi-Nee-Major
ジェルジ ベケーニュイ ネーエ マヨル
Balazs Szoeke
バラーズ セーケ
Agnes Balogh
アグネシュ バロフ
Orsolya Csuka
オルソイヤ チュカ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Innofinance Altalanos Innovacios Penzintezet
Original Assignee
Innofinance Altalanos Innovacios Penzintezet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Innofinance Altalanos Innovacios Penzintezet filed Critical Innofinance Altalanos Innovacios Penzintezet
Publication of JPH0215097A publication Critical patent/JPH0215097A/ja
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10Peptides having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • A61K38/09Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
JP1115265A 1988-05-10 1989-05-10 ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法 Pending JPH0215097A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU2251-2347/88 1988-05-10
HU882347A HU199694B (en) 1988-05-10 1988-05-10 Process for producing citostatic pharmaceutical compositions containing gonadoliberin derivatives

Publications (1)

Publication Number Publication Date
JPH0215097A true JPH0215097A (ja) 1990-01-18

Family

ID=10958948

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1115265A Pending JPH0215097A (ja) 1988-05-10 1989-05-10 ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法

Country Status (16)

Country Link
JP (1) JPH0215097A (fr)
KR (1) KR900017610A (fr)
BE (1) BE1004932A3 (fr)
CH (1) CH678013A5 (fr)
DE (1) DE3915317A1 (fr)
DK (1) DK228289A (fr)
FI (1) FI892275A7 (fr)
FR (1) FR2631237A1 (fr)
GB (1) GB2218335B (fr)
GR (1) GR890100315A (fr)
HU (1) HU199694B (fr)
IL (1) IL89998A0 (fr)
IT (1) IT1229251B (fr)
LU (1) LU87516A1 (fr)
NL (1) NL8901159A (fr)
SE (1) SE8901660L (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5760000A (en) * 1994-05-13 1998-06-02 University Technologies International,Inc. Inhibition of liver cancer by the use of GnRH and GnRH analogs
US6054432A (en) * 1996-09-12 2000-04-25 Asta Medica Aktiengesellschaft Means for treating prostate hypertrophy and prostate cancer

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4410514A (en) * 1982-12-06 1983-10-18 The Salk Institute For Biological Studies GnRH Agonists
IT1178775B (it) * 1983-12-23 1987-09-16 Konzponti Valto Es Hitelbank R Derivati della gonadoliberina e procedimento per la loro preparazione
HU189394B (en) * 1983-12-23 1986-06-30 Koezponti Valto- Es Hitelbank Rt Innovacios Alap,Hu Method for producing spermatozoa suitable for fertilization from mature fishes
US4760053A (en) * 1984-08-02 1988-07-26 Fernand Labrie Combination therapy for selected sex steroid dependent cancers
WO1986001105A1 (fr) * 1984-08-02 1986-02-27 Fernand Labrie Composition pharmaceutique pour le traitement de cancers dependant d'hormones
HU193607B (en) * 1985-07-18 1987-11-30 Innofinance Altalanos Innovaci Process for production of sexual products applyable for natural or artificial insemination for mammates
US4721775A (en) * 1985-08-26 1988-01-26 Board Of Regents, The University Of Texas System Effective peptides related to the luteinizing hormone releasing hormone from L-amino acids
HU194913B (en) * 1986-01-03 1988-03-28 Innofinance Altalanos Innovaci Process for producing novel gonadoliberin derivatives containing in the sixth position aromatic amino carboxylic acid and medical preparations containing these compounds

Also Published As

Publication number Publication date
HU199694B (en) 1990-03-28
IT1229251B (it) 1991-07-26
GB2218335A (en) 1989-11-15
FI892275A0 (fi) 1989-05-10
SE8901660D0 (sv) 1989-05-10
GB8910724D0 (en) 1989-06-28
HUT49813A (en) 1989-11-28
NL8901159A (nl) 1989-12-01
BE1004932A3 (fr) 1993-03-02
KR900017610A (ko) 1990-12-19
IL89998A0 (en) 1989-12-15
CH678013A5 (fr) 1991-07-31
DK228289D0 (da) 1989-05-10
SE8901660L (sv) 1989-11-11
IT8920435A0 (it) 1989-05-11
GB2218335B (en) 1991-09-25
FR2631237A1 (fr) 1989-11-17
GR890100315A (el) 1990-03-12
FI892275A7 (fi) 1989-11-11
DE3915317A1 (de) 1989-11-23
LU87516A1 (fr) 1990-12-11
DK228289A (da) 1989-11-11

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