JPH0215097A - ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法 - Google Patents
ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法Info
- Publication number
- JPH0215097A JPH0215097A JP1115265A JP11526589A JPH0215097A JP H0215097 A JPH0215097 A JP H0215097A JP 1115265 A JP1115265 A JP 1115265A JP 11526589 A JP11526589 A JP 11526589A JP H0215097 A JPH0215097 A JP H0215097A
- Authority
- JP
- Japan
- Prior art keywords
- group
- derivative
- general formula
- drug
- amino acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/10—Peptides having 12 to 20 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU2251-2347/88 | 1988-05-10 | ||
| HU882347A HU199694B (en) | 1988-05-10 | 1988-05-10 | Process for producing citostatic pharmaceutical compositions containing gonadoliberin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPH0215097A true JPH0215097A (ja) | 1990-01-18 |
Family
ID=10958948
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP1115265A Pending JPH0215097A (ja) | 1988-05-10 | 1989-05-10 | ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法 |
Country Status (16)
| Country | Link |
|---|---|
| JP (1) | JPH0215097A (fr) |
| KR (1) | KR900017610A (fr) |
| BE (1) | BE1004932A3 (fr) |
| CH (1) | CH678013A5 (fr) |
| DE (1) | DE3915317A1 (fr) |
| DK (1) | DK228289A (fr) |
| FI (1) | FI892275A7 (fr) |
| FR (1) | FR2631237A1 (fr) |
| GB (1) | GB2218335B (fr) |
| GR (1) | GR890100315A (fr) |
| HU (1) | HU199694B (fr) |
| IL (1) | IL89998A0 (fr) |
| IT (1) | IT1229251B (fr) |
| LU (1) | LU87516A1 (fr) |
| NL (1) | NL8901159A (fr) |
| SE (1) | SE8901660L (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5760000A (en) * | 1994-05-13 | 1998-06-02 | University Technologies International,Inc. | Inhibition of liver cancer by the use of GnRH and GnRH analogs |
| US6054432A (en) * | 1996-09-12 | 2000-04-25 | Asta Medica Aktiengesellschaft | Means for treating prostate hypertrophy and prostate cancer |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4410514A (en) * | 1982-12-06 | 1983-10-18 | The Salk Institute For Biological Studies | GnRH Agonists |
| IT1178775B (it) * | 1983-12-23 | 1987-09-16 | Konzponti Valto Es Hitelbank R | Derivati della gonadoliberina e procedimento per la loro preparazione |
| HU189394B (en) * | 1983-12-23 | 1986-06-30 | Koezponti Valto- Es Hitelbank Rt Innovacios Alap,Hu | Method for producing spermatozoa suitable for fertilization from mature fishes |
| US4760053A (en) * | 1984-08-02 | 1988-07-26 | Fernand Labrie | Combination therapy for selected sex steroid dependent cancers |
| WO1986001105A1 (fr) * | 1984-08-02 | 1986-02-27 | Fernand Labrie | Composition pharmaceutique pour le traitement de cancers dependant d'hormones |
| HU193607B (en) * | 1985-07-18 | 1987-11-30 | Innofinance Altalanos Innovaci | Process for production of sexual products applyable for natural or artificial insemination for mammates |
| US4721775A (en) * | 1985-08-26 | 1988-01-26 | Board Of Regents, The University Of Texas System | Effective peptides related to the luteinizing hormone releasing hormone from L-amino acids |
| HU194913B (en) * | 1986-01-03 | 1988-03-28 | Innofinance Altalanos Innovaci | Process for producing novel gonadoliberin derivatives containing in the sixth position aromatic amino carboxylic acid and medical preparations containing these compounds |
-
1988
- 1988-05-10 HU HU882347A patent/HU199694B/hu active IP Right Revival
-
1989
- 1989-04-18 IL IL89998A patent/IL89998A0/xx unknown
- 1989-05-08 CH CH1725/89A patent/CH678013A5/de not_active IP Right Cessation
- 1989-05-09 NL NL8901159A patent/NL8901159A/nl not_active Application Discontinuation
- 1989-05-10 LU LU87516A patent/LU87516A1/fr unknown
- 1989-05-10 GB GB8910724A patent/GB2218335B/en not_active Expired - Fee Related
- 1989-05-10 KR KR1019890006230A patent/KR900017610A/ko not_active Withdrawn
- 1989-05-10 BE BE8900499A patent/BE1004932A3/fr not_active IP Right Cessation
- 1989-05-10 GR GR890100315A patent/GR890100315A/el unknown
- 1989-05-10 JP JP1115265A patent/JPH0215097A/ja active Pending
- 1989-05-10 DE DE3915317A patent/DE3915317A1/de not_active Withdrawn
- 1989-05-10 SE SE8901660A patent/SE8901660L/ not_active Application Discontinuation
- 1989-05-10 DK DK228289A patent/DK228289A/da not_active Application Discontinuation
- 1989-05-10 FI FI892275A patent/FI892275A7/fi not_active Application Discontinuation
- 1989-05-10 FR FR8906094A patent/FR2631237A1/fr active Pending
- 1989-05-11 IT IT8920435A patent/IT1229251B/it active
Also Published As
| Publication number | Publication date |
|---|---|
| HU199694B (en) | 1990-03-28 |
| IT1229251B (it) | 1991-07-26 |
| GB2218335A (en) | 1989-11-15 |
| FI892275A0 (fi) | 1989-05-10 |
| SE8901660D0 (sv) | 1989-05-10 |
| GB8910724D0 (en) | 1989-06-28 |
| HUT49813A (en) | 1989-11-28 |
| NL8901159A (nl) | 1989-12-01 |
| BE1004932A3 (fr) | 1993-03-02 |
| KR900017610A (ko) | 1990-12-19 |
| IL89998A0 (en) | 1989-12-15 |
| CH678013A5 (fr) | 1991-07-31 |
| DK228289D0 (da) | 1989-05-10 |
| SE8901660L (sv) | 1989-11-11 |
| IT8920435A0 (it) | 1989-05-11 |
| GB2218335B (en) | 1991-09-25 |
| FR2631237A1 (fr) | 1989-11-17 |
| GR890100315A (el) | 1990-03-12 |
| FI892275A7 (fi) | 1989-11-11 |
| DE3915317A1 (de) | 1989-11-23 |
| LU87516A1 (fr) | 1990-12-11 |
| DK228289A (da) | 1989-11-11 |
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| JPH0215097A (ja) | ゴナドリベリン誘導体含有薬剤の製造方法及びその使用方法 | |
| Korkut et al. | Inhibition of growth of experimental prostate cancer with sustained delivery systems (microcapsules and microgranules) of the luteinizing hormone-releasing hormone antagonist SB-75. | |
| Schally et al. | Combination of a long-acting delivery system for luteinizing hormone-releasing hormone agonist with Novantrone chemotherapy: increased efficacy in the rat prostate cancer model. | |
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