JPH09504512A - 抗菌活性、抗マイコプラズマ活性、抗真菌類活性および除草活性を有するモン酸ａおよびｃの誘導体 - Google Patents

抗菌活性、抗マイコプラズマ活性、抗真菌類活性および除草活性を有するモン酸ａおよびｃの誘導体

Info

Publication number
JPH09504512A
JPH09504512A JP7506705A JP50670595A JPH09504512A JP H09504512 A JPH09504512 A JP H09504512A JP 7506705 A JP7506705 A JP 7506705A JP 50670595 A JP50670595 A JP 50670595A JP H09504512 A JPH09504512 A JP H09504512A
Authority
JP
Japan
Prior art keywords
formula
dithiolo
compound
methyl
mmol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP7506705A
Other languages
English (en)
Japanese (ja)
Inventor
ブルーム，ニジェール・ジョン・ペリーマン
オハンロン，ピーター・ジョン
オズボーン，ニール・フレデリック
ペンジェリー，ドンナ
Original Assignee
スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939316879A external-priority patent/GB9316879D0/en
Priority claimed from GB9400592A external-priority patent/GB9400592D0/en
Priority claimed from GB9401139A external-priority patent/GB9401139D0/en
Application filed by スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー filed Critical スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー
Publication of JPH09504512A publication Critical patent/JPH09504512A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP7506705A 1993-08-13 1994-08-02 抗菌活性、抗マイコプラズマ活性、抗真菌類活性および除草活性を有するモン酸ａおよびｃの誘導体 Pending JPH09504512A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB9316879.7 1993-08-13
GB939316879A GB9316879D0 (en) 1993-08-13 1993-08-13 Novel compounds
GB9400592A GB9400592D0 (en) 1994-01-14 1994-01-14 Novel compounds
GB9400592.3 1994-01-14
GB9401139A GB9401139D0 (en) 1994-01-21 1994-01-21 Novel compounds
GB9401139.2 1994-01-21
PCT/EP1994/002552 WO1995005384A1 (fr) 1993-08-13 1994-08-02 Derives d'acides moniques a et c a activite antibacterienne, antimycoplasmique, antifongique et herbicide

Publications (1)

Publication Number Publication Date
JPH09504512A true JPH09504512A (ja) 1997-05-06

Family

ID=27266812

Family Applications (1)

Application Number Title Priority Date Filing Date
JP7506705A Pending JPH09504512A (ja) 1993-08-13 1994-08-02 抗菌活性、抗マイコプラズマ活性、抗真菌類活性および除草活性を有するモン酸ａおよびｃの誘導体

Country Status (7)

Country Link
EP (1) EP0712405A1 (fr)
JP (1) JPH09504512A (fr)
AP (1) AP9400663A0 (fr)
AU (1) AU7497594A (fr)
IL (1) IL110620A0 (fr)
MA (1) MA23309A1 (fr)
WO (1) WO1995005384A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012201669A (ja) * 2011-03-28 2012-10-22 Tokyo Univ Of Pharmacy & Life Science ミキソピロニン誘導体含有抗菌剤

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996023795A1 (fr) * 1995-01-31 1996-08-08 Sankyo-Company, Limited Derives d'acide pseudomonique
US5726195A (en) * 1995-07-28 1998-03-10 Cubist Pharmaceuticals, Inc. Aminoacyl adenylate mimics as novel antimicrobial and antiparasitic agents
WO1997005126A1 (fr) * 1995-07-29 1997-02-13 Smithkline Beecham Plc Mupirocinsulfamates a activite antibacterienne
GB9822241D0 (en) * 1998-10-12 1998-12-09 Smithkline Beecham Plc Novel compounds
CA2372079A1 (fr) 1999-05-05 2000-11-09 Aaron H. Leeman Nouveaux catechols utilises comme agents antimicrobiens
EP1176959B1 (fr) 1999-05-05 2006-03-08 Merck & Co., Inc. Prolines en tant qu'agents antimicrobiens
CN1425025A (zh) 1999-12-15 2003-06-18 卡比斯特制药公司 作为抗菌剂的新颖的脂肽
US6696412B1 (en) 2000-01-20 2004-02-24 Cubist Pharmaceuticals, Inc. High purity lipopeptides, Lipopeptide micelles and processes for preparing same
IL156394A0 (en) 2000-12-18 2004-01-04 Cubist Pharm Inc Methods for preparing purified lipopeptides
EP1932853A1 (fr) 2001-08-06 2008-06-18 Cubist Pharmaceutical Inc. Nouveaux depsipeptides et leur procédé de préparation
JP4530667B2 (ja) 2002-03-26 2010-08-25 ウェリケム バイオテック インコーポレーテッド 治療活性を有する新規ジチオロピロロン（ｄｉｔｈｉｏｌｏｐｙｒｒｏｌｏｎｅｓ）
US20060004185A1 (en) 2004-07-01 2006-01-05 Leese Richard A Peptide antibiotics and peptide intermediates for their prepartion
US8071637B2 (en) 2006-09-29 2011-12-06 Welichem Biotech Inc. Dithiolopyrrolones compounds and their therapeutic applications
BRPI0923567A2 (pt) 2008-12-22 2016-09-27 Cubist Pharm Inc agentes antibactericidas novos para o tratamento de infecções gram positivas
TW201035111A (en) 2008-12-23 2010-10-01 Biosource Pharm Inc Antibiotic compositions for the treatment of gram negative infections
US8415307B1 (en) 2010-06-23 2013-04-09 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
TW201343645A (zh) 2012-03-30 2013-11-01 Cubist Pharm Inc １，３，４－□二唑及１，３，４－噻二唑β－內醯胺酶抑制劑

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2860726D1 (en) * 1977-11-05 1981-08-27 Beecham Group Plc Antibacterially active amides, process for their preparation and pharmaceutical compositions containing said amides
EP0087953B1 (fr) * 1982-02-27 1988-04-27 Beecham Group Plc Composés 1-normon-2-yl-hétérocycliques antibactériens
ZA923242B (en) * 1991-05-07 1993-01-27 Sankyo Co Novel anti-bacterial compound
WO1993015072A1 (fr) * 1992-01-24 1993-08-05 Smithkline Beecham Plc Cetones de thiazolyle 1-normon-2-yl

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012201669A (ja) * 2011-03-28 2012-10-22 Tokyo Univ Of Pharmacy & Life Science ミキソピロニン誘導体含有抗菌剤

Also Published As

Publication number Publication date
EP0712405A1 (fr) 1996-05-22
AP9400663A0 (en) 1996-02-10
AU7497594A (en) 1995-03-14
IL110620A0 (en) 1994-11-11
MA23309A1 (fr) 1995-04-01
WO1995005384A1 (fr) 1995-02-23

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