JPS557204A - Derivative of 1-phthalazone - Google Patents
Derivative of 1-phthalazoneInfo
- Publication number
- JPS557204A JPS557204A JP7801878A JP7801878A JPS557204A JP S557204 A JPS557204 A JP S557204A JP 7801878 A JP7801878 A JP 7801878A JP 7801878 A JP7801878 A JP 7801878A JP S557204 A JPS557204 A JP S557204A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- phthalazone
- dimethyl
- derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000001875 compounds Chemical class 0.000 abstract 5
- 206010003210 Arteriosclerosis Diseases 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 208000011775 arteriosclerosis disease Diseases 0.000 abstract 2
- DSNBHJFQCNUKMA-SCKDECHMSA-N thromboxane A2 Chemical compound OC(=O)CCC\C=C/C[C@@H]1[C@@H](/C=C/[C@@H](O)CCCCC)O[C@@H]2O[C@H]1C2 DSNBHJFQCNUKMA-SCKDECHMSA-N 0.000 abstract 2
- 208000007536 Thrombosis Diseases 0.000 abstract 1
- 230000003042 antagnostic effect Effects 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 230000002785 anti-thrombosis Effects 0.000 abstract 1
- 229960004676 antithrombotic agent Drugs 0.000 abstract 1
- 230000002490 cerebral effect Effects 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- BEPAFCGSDWSTEL-UHFFFAOYSA-N dimethyl malonate Chemical compound COC(=O)CC(=O)OC BEPAFCGSDWSTEL-UHFFFAOYSA-N 0.000 abstract 1
- 230000000302 ischemic effect Effects 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- GXHFUVWIGNLZSC-UHFFFAOYSA-N meldrum's acid Chemical compound CC1(C)OC(=O)CC(=O)O1 GXHFUVWIGNLZSC-UHFFFAOYSA-N 0.000 abstract 1
- 125000001570 methylene group Chemical group [H]C([H])([*:1])[*:2] 0.000 abstract 1
- 208000031225 myocardial ischemia Diseases 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 208000019553 vascular disease Diseases 0.000 abstract 1
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A derivative of 1-phthalazone of formula I [R1-R5 are alkyl; R4 and R5 may together form a di-subsituted methylene group of formula II (R6, R7 are alkyl)].
EXAMPLE: A compound of formula I (R3=R4=R5=C2H5).
USE: Agents for arteriosclerosis, antithrombotics, or antagonists of thromboxane A2. The compound has an excellent antagonistic property for thromboxane A2 and is useful for prevention and remedy of arteriosclerosis, thrombosis, ischemic cerebral vascular disease and ischemic heart disease.
PROCESS: A compound of formula I is obtained by the treatment of a compound of formula III, e.g. 7-ethoxycarbonyl-6, 8-dimethyl-4-formyl-1-phthalazone, with a compound of formula IV, e.g. malonic acid dimethyl ester, 2, 2-dimethyl-1, 3- dioxane-4, 6-dione, etc.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP7801878A JPS557204A (en) | 1978-06-29 | 1978-06-29 | Derivative of 1-phthalazone |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP7801878A JPS557204A (en) | 1978-06-29 | 1978-06-29 | Derivative of 1-phthalazone |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS557204A true JPS557204A (en) | 1980-01-19 |
Family
ID=13650046
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP7801878A Pending JPS557204A (en) | 1978-06-29 | 1978-06-29 | Derivative of 1-phthalazone |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS557204A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56113220A (en) * | 1980-02-15 | 1981-09-07 | Iseki Agricult Mach | Up and down motion device for wheel of walking type rice transplanter |
-
1978
- 1978-06-29 JP JP7801878A patent/JPS557204A/en active Pending
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56113220A (en) * | 1980-02-15 | 1981-09-07 | Iseki Agricult Mach | Up and down motion device for wheel of walking type rice transplanter |
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