JPS6043356B2 - 耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法 - Google Patents

耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法

Info

Publication number
JPS6043356B2
JPS6043356B2 JP51121237A JP12123776A JPS6043356B2 JP S6043356 B2 JPS6043356 B2 JP S6043356B2 JP 51121237 A JP51121237 A JP 51121237A JP 12123776 A JP12123776 A JP 12123776A JP S6043356 B2 JPS6043356 B2 JP S6043356B2
Authority
JP
Japan
Prior art keywords
kanamycin
amino
hydroxybutyryl
derivative
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP51121237A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5346940A (en
Inventor
浜夫 梅沢
信一 近藤
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Microbial Chemistry Research Foundation
Original Assignee
Microbial Chemistry Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chemistry Research Foundation filed Critical Microbial Chemistry Research Foundation
Priority to JP51121237A priority Critical patent/JPS6043356B2/ja
Priority to GB32436/77A priority patent/GB1567560A/en
Priority to DE2741431A priority patent/DE2741431C3/de
Priority to CA287,796A priority patent/CA1081693A/fr
Priority to FR7731107A priority patent/FR2367775A1/fr
Publication of JPS5346940A publication Critical patent/JPS5346940A/ja
Publication of JPS6043356B2 publication Critical patent/JPS6043356B2/ja
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP51121237A 1976-10-12 1976-10-12 耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法 Expired JPS6043356B2 (ja)

Priority Applications (5)

Application Number Priority Date Filing Date Title
JP51121237A JPS6043356B2 (ja) 1976-10-12 1976-10-12 耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法
GB32436/77A GB1567560A (en) 1976-10-12 1977-08-02 Kanamycin c derivatives active against various drug-resistant bacteria
DE2741431A DE2741431C3 (de) 1976-10-12 1977-09-14 l-N-(L-4-Amino-2-hydroxybutyryl)-3'-desoxykanamycin-C, l-N-(L-4-Amino-2hydroxybutyryl)-3',4'-didesoxykanamycin-C und deren Säureadditionssalze, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende antibakterielle Zusammensetzungen
CA287,796A CA1081693A (fr) 1976-10-12 1977-09-29 Derives de la kanamycine c
FR7731107A FR2367775A1 (fr) 1976-10-12 1977-10-11 Derives nouveaux de la kanamycine c actifs contre diverses bacteries resistantes aux medicaments

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP51121237A JPS6043356B2 (ja) 1976-10-12 1976-10-12 耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法

Publications (2)

Publication Number Publication Date
JPS5346940A JPS5346940A (en) 1978-04-27
JPS6043356B2 true JPS6043356B2 (ja) 1985-09-27

Family

ID=14806295

Family Applications (1)

Application Number Title Priority Date Filing Date
JP51121237A Expired JPS6043356B2 (ja) 1976-10-12 1976-10-12 耐性菌に有効なカナマイシンｃ誘導体およびそれらの製造法

Country Status (5)

Country Link
JP (1) JPS6043356B2 (fr)
CA (1) CA1081693A (fr)
DE (1) DE2741431C3 (fr)
FR (1) FR2367775A1 (fr)
GB (1) GB1567560A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63133258U (fr) * 1987-02-25 1988-08-31

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK157833C (da) * 1988-03-01 1991-04-29 Dansk Transfertryk Fremgangsmaade til laminering af tekstiler

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63133258U (fr) * 1987-02-25 1988-08-31

Also Published As

Publication number Publication date
DE2741431C3 (de) 1979-10-25
FR2367775A1 (fr) 1978-05-12
CA1081693A (fr) 1980-07-15
DE2741431B2 (de) 1979-03-08
DE2741431A1 (de) 1978-04-13
GB1567560A (en) 1980-05-14
FR2367775B1 (fr) 1980-11-28
JPS5346940A (en) 1978-04-27

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