JPS6163652A - （ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法 - Google Patents

（ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法

Info

Publication number
JPS6163652A
JPS6163652A JP18558384A JP18558384A JPS6163652A JP S6163652 A JPS6163652 A JP S6163652A JP 18558384 A JP18558384 A JP 18558384A JP 18558384 A JP18558384 A JP 18558384A JP S6163652 A JPS6163652 A JP S6163652A
Authority
JP
Japan
Prior art keywords
benzyl
hydroxypyrrolidine
acid
optically active
mandelic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP18558384A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0421662B2 (th
Inventor
Kazuharu Tamazawa
玉沢　一晴
Hideki Arima
有馬　英樹
Yasuo Isomura
磯村　八州男
Minoru Okada
稔 岡田
Hideetsu Kaniwa
鹿庭　秀悦
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astellas Pharma Inc
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Priority to JP18558384A priority Critical patent/JPS6163652A/ja
Publication of JPS6163652A publication Critical patent/JPS6163652A/ja
Publication of JPH0421662B2 publication Critical patent/JPH0421662B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
JP18558384A 1984-09-04 1984-09-04 （ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法 Granted JPS6163652A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP18558384A JPS6163652A (ja) 1984-09-04 1984-09-04 （ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP18558384A JPS6163652A (ja) 1984-09-04 1984-09-04 （ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法

Publications (2)

Publication Number Publication Date
JPS6163652A true JPS6163652A (ja) 1986-04-01
JPH0421662B2 JPH0421662B2 (th) 1992-04-13

Family

ID=16173342

Family Applications (1)

Application Number Title Priority Date Filing Date
JP18558384A Granted JPS6163652A (ja) 1984-09-04 1984-09-04 （ｓ）−（−）−１−ベンジル−３−ヒドロキシピロリジンの製造法

Country Status (1)

Country Link
JP (1) JPS6163652A (th)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5187094A (en) * 1989-09-06 1993-02-16 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Method for the preparation of optically active 3-hydroxypyrrolidine derivatives
EP0692471A1 (de) 1994-07-15 1996-01-17 Degussa Aktiengesellschaft Verfahren zur Herstellung optisch aktiver 3-Hydroxy-Pyrrolidine mit hoher Enantiomerenreinheit
WO1999065918A1 (en) * 1998-06-17 1999-12-23 Daiichi Pharmaceutical Co., Ltd. Enantiomerically pure substituted oxaaza compounds, salts of the same, and processes for the preparation of both
US6613550B2 (en) 2000-02-29 2003-09-02 Pfizer Inc. Microbial process for preparation of optically active 3-hydroxypyrrolidine derivatives
WO2007024113A1 (en) 2005-08-25 2007-03-01 Rstech Corporation Process for the preparation of chiral 3-hydroxy pyrrolidine compound and derivatives thereof having high optical purity
US7652152B2 (en) 2005-07-20 2010-01-26 Chiroad Incorporate Synthetic method of optically pure (S)-3-hydroxypyrrolidine
EP4382529A1 (en) 2022-12-07 2024-06-12 Bayer Consumer Care AG A process for preparing pure (3s)-pyrrolidin-3-ol and pure (3s)-pyrrolidin-3-ol hydrochloride

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5187094A (en) * 1989-09-06 1993-02-16 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Method for the preparation of optically active 3-hydroxypyrrolidine derivatives
EP0692471A1 (de) 1994-07-15 1996-01-17 Degussa Aktiengesellschaft Verfahren zur Herstellung optisch aktiver 3-Hydroxy-Pyrrolidine mit hoher Enantiomerenreinheit
WO1999065918A1 (en) * 1998-06-17 1999-12-23 Daiichi Pharmaceutical Co., Ltd. Enantiomerically pure substituted oxaaza compounds, salts of the same, and processes for the preparation of both
US6423843B1 (en) 1998-06-17 2002-07-23 Daiichi Pharmaceutical Co., Ltd. Enantiomerically pure substituted oxaaza compounds, salts of the same, and processes for the preparation of both
US6613550B2 (en) 2000-02-29 2003-09-02 Pfizer Inc. Microbial process for preparation of optically active 3-hydroxypyrrolidine derivatives
US7652152B2 (en) 2005-07-20 2010-01-26 Chiroad Incorporate Synthetic method of optically pure (S)-3-hydroxypyrrolidine
WO2007024113A1 (en) 2005-08-25 2007-03-01 Rstech Corporation Process for the preparation of chiral 3-hydroxy pyrrolidine compound and derivatives thereof having high optical purity
EP4382529A1 (en) 2022-12-07 2024-06-12 Bayer Consumer Care AG A process for preparing pure (3s)-pyrrolidin-3-ol and pure (3s)-pyrrolidin-3-ol hydrochloride
WO2024121219A1 (en) 2022-12-07 2024-06-13 Bayer Consumer Care Ag A process for preparing pure (3s)-pyrrolidin-3-ol and pure (3s)-pyrrolidin-3-ol hydrochloride

Also Published As

Publication number Publication date
JPH0421662B2 (th) 1992-04-13

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