JPS6236361A - キノロン治療薬及びその製法 - Google Patents
キノロン治療薬及びその製法Info
- Publication number
- JPS6236361A JPS6236361A JP61139954A JP13995486A JPS6236361A JP S6236361 A JPS6236361 A JP S6236361A JP 61139954 A JP61139954 A JP 61139954A JP 13995486 A JP13995486 A JP 13995486A JP S6236361 A JPS6236361 A JP S6236361A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- hydrogen
- lower alkyl
- quinolone
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/36—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Cardiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB858515209A GB8515209D0 (en) | 1985-06-15 | 1985-06-15 | Therapeutic agents |
| GB8515209 | 1985-06-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS6236361A true JPS6236361A (ja) | 1987-02-17 |
Family
ID=10580805
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP61139954A Pending JPS6236361A (ja) | 1985-06-15 | 1986-06-16 | キノロン治療薬及びその製法 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US4772614A (de) |
| EP (1) | EP0206616A3 (de) |
| JP (1) | JPS6236361A (de) |
| KR (1) | KR870000302A (de) |
| CN (1) | CN86104611A (de) |
| AU (1) | AU5838286A (de) |
| DD (1) | DD249010A5 (de) |
| DK (1) | DK272386A (de) |
| ES (1) | ES8801211A1 (de) |
| FI (1) | FI862519A7 (de) |
| GB (1) | GB8515209D0 (de) |
| GR (1) | GR861528B (de) |
| HU (1) | HUT42073A (de) |
| IL (1) | IL79039A0 (de) |
| JO (1) | JO1483B1 (de) |
| NO (1) | NO862372L (de) |
| PH (1) | PH22992A (de) |
| PT (1) | PT82760B (de) |
| ZA (1) | ZA864288B (de) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0172004B1 (de) * | 1984-08-15 | 1990-03-21 | The Boots Company PLC | Chinolinone, Verfahren zu ihrer Herstellung und die sie enthaltenden pharmazeutischen Präparate |
| GB8627698D0 (en) * | 1986-11-20 | 1986-12-17 | Boots Co Plc | Therapeutic agents |
| GB8726950D0 (en) * | 1987-11-18 | 1987-12-23 | Boots Co Plc | Chemical process |
| GB8804016D0 (en) * | 1988-02-22 | 1988-03-23 | Boots Co Plc | Therapeutic agents |
| US5081121A (en) * | 1988-05-24 | 1992-01-14 | Tatsushi Osawa | 4(1h)-quinolone derivatives |
| GB8918952D0 (en) * | 1989-08-19 | 1989-10-04 | Boots Co Plc | Therapeutic agents |
| US5927566A (en) * | 1996-07-11 | 1999-07-27 | Aptargroup, Inc. | One-piece dispensing system and method for making same |
| EP1107759A1 (de) * | 1998-08-03 | 2001-06-20 | Basf Corporation | Pyridinonen zur behandlung von seksuellen störungen |
| US6562838B2 (en) * | 2001-01-26 | 2003-05-13 | R. T. Alamo Ventures I, L.L.C. | Treatment of cardiovascular disease with quinolinone enantiomers |
| US6451813B1 (en) | 2001-01-26 | 2002-09-17 | R. T. Alamo Ventures I, Llc | Treatment of gastroparesis in certain patient groups |
| US6458804B1 (en) * | 2001-01-26 | 2002-10-01 | R.T. Alamo Venturesi, Llc | Methods for the treatment of central nervous system disorders in certain patient groups |
| JP2006514102A (ja) * | 2002-11-07 | 2006-04-27 | アストラゼネカ アクチボラグ | ２−オキソ−エタンスルホンアミド誘導体 |
| CN105017145B (zh) * | 2012-12-12 | 2017-12-05 | 王子厚 | 具有抗肿瘤活性的氯氧喹衍生物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4913185A (de) * | 1972-06-02 | 1974-02-05 | ||
| NZ193167A (en) * | 1979-03-27 | 1984-08-24 | Boots Co Plc | Quinoline derivatives and pharmaceutical compositions |
| IE51542B1 (en) * | 1980-09-26 | 1987-01-07 | Boots Co Ltd | Therapeutic agents |
| PT79031B (en) * | 1983-08-20 | 1986-08-22 | Boots Co Plc | Therapeutic agents |
| DE3578374D1 (de) * | 1984-01-13 | 1990-08-02 | Boots Co Ltd | Verwendung von chinolonen fuer die herstellung eines arzneimittels zur behandlung von herzerkrankungen. |
| EP0172004B1 (de) * | 1984-08-15 | 1990-03-21 | The Boots Company PLC | Chinolinone, Verfahren zu ihrer Herstellung und die sie enthaltenden pharmazeutischen Präparate |
-
1985
- 1985-06-15 GB GB858515209A patent/GB8515209D0/en active Pending
-
1986
- 1986-06-05 AU AU58382/86A patent/AU5838286A/en not_active Abandoned
- 1986-06-05 IL IL79039A patent/IL79039A0/xx unknown
- 1986-06-09 EP EP86304390A patent/EP0206616A3/de not_active Withdrawn
- 1986-06-09 PH PH33870A patent/PH22992A/en unknown
- 1986-06-09 ZA ZA864288A patent/ZA864288B/xx unknown
- 1986-06-10 DK DK272386A patent/DK272386A/da not_active Application Discontinuation
- 1986-06-12 PT PT82760A patent/PT82760B/pt unknown
- 1986-06-12 GR GR861528A patent/GR861528B/el unknown
- 1986-06-12 FI FI862519A patent/FI862519A7/fi not_active IP Right Cessation
- 1986-06-13 ES ES556027A patent/ES8801211A1/es not_active Expired
- 1986-06-13 HU HU862522A patent/HUT42073A/hu unknown
- 1986-06-13 US US06/874,217 patent/US4772614A/en not_active Expired - Fee Related
- 1986-06-13 DD DD86291288A patent/DD249010A5/de unknown
- 1986-06-13 NO NO862372A patent/NO862372L/no unknown
- 1986-06-14 JO JO19861483A patent/JO1483B1/en active
- 1986-06-14 KR KR1019860004738A patent/KR870000302A/ko not_active Withdrawn
- 1986-06-16 JP JP61139954A patent/JPS6236361A/ja active Pending
- 1986-07-07 CN CN198686104611A patent/CN86104611A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| PT82760B (en) | 1988-05-19 |
| NO862372L (no) | 1986-12-16 |
| FI862519A7 (fi) | 1986-12-16 |
| KR870000302A (ko) | 1987-02-17 |
| EP0206616A3 (de) | 1988-06-01 |
| EP0206616A2 (de) | 1986-12-30 |
| US4772614A (en) | 1988-09-20 |
| PH22992A (en) | 1989-02-24 |
| IL79039A0 (en) | 1986-09-30 |
| CN86104611A (zh) | 1988-01-27 |
| JO1483B1 (en) | 1988-03-10 |
| FI862519A0 (fi) | 1986-06-12 |
| PT82760A (en) | 1986-07-01 |
| HUT42073A (en) | 1987-06-29 |
| DK272386A (da) | 1986-12-16 |
| NO862372D0 (no) | 1986-06-13 |
| GB8515209D0 (en) | 1985-07-17 |
| DK272386D0 (da) | 1986-06-10 |
| GR861528B (en) | 1986-10-10 |
| AU5838286A (en) | 1986-12-18 |
| ES8801211A1 (es) | 1987-12-16 |
| DD249010A5 (de) | 1987-08-26 |
| ZA864288B (en) | 1987-01-28 |
| ES556027A0 (es) | 1987-12-16 |
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