LT3183247T - Aminopirimidinilo junginiai, kaip jak inhibitoriai - Google Patents

Aminopirimidinilo junginiai, kaip jak inhibitoriai

Info

Publication number
LT3183247T
LT3183247T LTEP15766627.2T LT15766627T LT3183247T LT 3183247 T LT3183247 T LT 3183247T LT 15766627 T LT15766627 T LT 15766627T LT 3183247 T LT3183247 T LT 3183247T
Authority
LT
Lithuania
Prior art keywords
jak inhibitors
aminopyrimidinyl
compounds
aminopyrimidinyl compounds
jak
Prior art date
Application number
LTEP15766627.2T
Other languages
English (en)
Inventor
Andrew Fensome
Ariamala Gopalsamy
Brian S. GERSTENBERGER
Ivan Viktorovich Efremov
Zhao-Kui Wan
Betsy PIERCE
Jean-Baptiste Telliez
John I Trujillo
Liying Zhang
Li Xing
Eddine Saiah
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54148580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT3183247(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of LT3183247T publication Critical patent/LT3183247T/lt

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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  • Health & Medical Sciences (AREA)
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LTEP15766627.2T 2014-08-21 2015-08-07 Aminopirimidinilo junginiai, kaip jak inhibitoriai LT3183247T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462039969P 2014-08-21 2014-08-21
PCT/IB2015/056021 WO2016027195A1 (en) 2014-08-21 2015-08-07 Aminopyrimidinyl compounds as jak inhibitors

Publications (1)

Publication Number Publication Date
LT3183247T true LT3183247T (lt) 2018-01-25

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LTEP15766627.2T LT3183247T (lt) 2014-08-21 2015-08-07 Aminopirimidinilo junginiai, kaip jak inhibitoriai

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US (5) US9663526B2 (lt)
EP (1) EP3183247B9 (lt)
JP (1) JP6218260B2 (lt)
KR (1) KR101877189B1 (lt)
CN (1) CN107074867B (lt)
AP (1) AP2017009748A0 (lt)
AR (1) AR101599A1 (lt)
AU (1) AU2015304883B2 (lt)
BR (1) BR112017003054B1 (lt)
CA (1) CA2900855C (lt)
CL (1) CL2017000406A1 (lt)
CO (1) CO2017001603A2 (lt)
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IL250709B (en) 2019-05-30
US10463675B2 (en) 2019-11-05
IL250709A0 (en) 2017-04-30
NZ729005A (en) 2020-06-26

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