LU79028A1 - Nouveaux imidazoles et leurs derives sulfoxydes et sulfones correspondants,leur preparation et compositions pharmaceutiques les contenant - Google Patents
Nouveaux imidazoles et leurs derives sulfoxydes et sulfones correspondants,leur preparation et compositions pharmaceutiques les contenantInfo
- Publication number
- LU79028A1 LU79028A1 LU79028A LU79028A LU79028A1 LU 79028 A1 LU79028 A1 LU 79028A1 LU 79028 A LU79028 A LU 79028A LU 79028 A LU79028 A LU 79028A LU 79028 A1 LU79028 A1 LU 79028A1
- Authority
- LU
- Luxembourg
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- corresponding sulfoxide
- sulphone derivatives
- Prior art date
Links
- 150000002460 imidazoles Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003462 sulfoxides Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Rheumatology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US76721977A | 1977-02-09 | 1977-02-09 | |
| US05/865,831 US4182769A (en) | 1977-02-09 | 1978-01-05 | Anti-inflammatory 1-substituted-4,5-diaryl-2-(substituted-thio) imidazoles and their corresponding sulfoxides and sulfones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LU79028A1 true LU79028A1 (fr) | 1979-05-25 |
Family
ID=27117878
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU79028A LU79028A1 (fr) | 1977-02-09 | 1978-02-08 | Nouveaux imidazoles et leurs derives sulfoxydes et sulfones correspondants,leur preparation et compositions pharmaceutiques les contenant |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4182769A (fr) |
| JP (1) | JPS53130665A (fr) |
| AR (1) | AR221590A1 (fr) |
| AT (1) | AT363076B (fr) |
| AU (1) | AU524360B2 (fr) |
| CA (1) | CA1107286A (fr) |
| CH (1) | CH643834A5 (fr) |
| DE (1) | DE2805166A1 (fr) |
| DK (1) | DK16878A (fr) |
| ES (1) | ES466793A1 (fr) |
| FI (1) | FI68619C (fr) |
| FR (1) | FR2380264A1 (fr) |
| GB (1) | GB1587373A (fr) |
| GR (1) | GR64157B (fr) |
| HU (1) | HU181868B (fr) |
| IE (1) | IE46454B1 (fr) |
| IL (1) | IL53996A (fr) |
| IT (1) | IT1092439B (fr) |
| LU (1) | LU79028A1 (fr) |
| MX (1) | MX5934E (fr) |
| NL (1) | NL7801454A (fr) |
| NO (1) | NO149813C (fr) |
| NZ (1) | NZ186411A (fr) |
| PT (1) | PT67625B (fr) |
| SE (1) | SE7801466L (fr) |
| SU (1) | SU867301A3 (fr) |
| YU (1) | YU28978A (fr) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2823197A1 (de) * | 1978-05-24 | 1979-11-29 | Schering Ag | Neue imidazolderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
| EP0008072B1 (fr) * | 1978-08-10 | 1984-02-22 | Ciba-Geigy Ag | Amides substituées de l'acide anthranilique, procédé pour leur préparation et compositions pharmaceutiques les contenant et leur préparation |
| US4308277A (en) * | 1978-08-10 | 1981-12-29 | Ciba-Geigy Corporation | 2,4,5-Trisubstituted imidazolines and pharmaceutical compositions containing same |
| US4199592A (en) * | 1978-08-29 | 1980-04-22 | E. I. Du Pont De Nemours And Company | Antiinflammatory 4,5-diaryl-2-nitroimidazoles |
| DK337779A (da) * | 1978-10-02 | 1980-04-03 | Du Pont | Fremgangsmaade til fremstilling af antiinflammatoriske 2-substituerede 1h-phenantro (9,10)-imidazoler |
| DE2856909A1 (de) * | 1978-12-28 | 1980-07-17 | Schering Ag | Neue imidazolderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
| IT1110282B (it) * | 1979-02-19 | 1985-12-23 | Acraf | Tio-indazoli basici |
| DE3025484A1 (de) * | 1980-07-03 | 1982-02-04 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Neue imidazol-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
| US4438117A (en) | 1980-09-03 | 1984-03-20 | E. I. Du Pont De Nemours And Company | 2-Substituted thio-4,5-diarylpyrimidines |
| US4355041A (en) * | 1982-01-04 | 1982-10-19 | E. I. Du Pont De Nemours And Company | 4,5-Bis-(4-fluorophenyl)-1-(4-nitrobenzyl)-2-[((1,1,2,2-tetrafluoroethyl)sulfonyl]-1H-imidazole, composition and use |
| US4503065A (en) * | 1982-08-03 | 1985-03-05 | E. I. Du Pont De Nemours And Company | Antiinflammatory 4,5-diaryl 1-2-halo imidazoles |
| ZA826501B (en) * | 1982-09-06 | 1984-04-25 | Du Pont | Anti-hypertensive imidazole derivative |
| DE3504678A1 (de) * | 1985-02-12 | 1986-08-14 | A. Nattermann & Cie GmbH, 5000 Köln | Neue imidazolyl-oxyalkansaeuren und -thioalkansaeuren, ihre derivate und verfahren zu ihrer herstellung |
| DE3508665A1 (de) * | 1985-03-12 | 1986-09-18 | Hoechst Ag, 6230 Frankfurt | Heterocyclische sulfide und ihre anwendung als immunmodulatoren |
| US4686231A (en) * | 1985-12-12 | 1987-08-11 | Smithkline Beckman Corporation | Inhibition of 5-lipoxygenase products |
| US4780470A (en) * | 1986-08-19 | 1988-10-25 | Smithkline Beckman Corporation | Inhibition of interleukin-1 by monocytes and/or macrophages |
| US5300519A (en) * | 1988-07-06 | 1994-04-05 | The University Of Sheffield | Immunosuppressive agents |
| US5030644A (en) * | 1989-07-31 | 1991-07-09 | Merck & Co., Inc. | Imidazole compounds and their use as transglutaminase inhibitors |
| US5098707A (en) * | 1989-07-31 | 1992-03-24 | Merck & Co., Inc. | Imidazole compounds and their use as transglutaminase inhibitors |
| JPH03145473A (ja) * | 1989-10-27 | 1991-06-20 | Hisamitsu Pharmaceut Co Inc | 新規なイミダゾール酢酸誘導体 |
| GB9005966D0 (en) * | 1990-03-16 | 1990-05-09 | May & Baker Ltd | New compositions of matter |
| DE4010797A1 (de) * | 1990-04-04 | 1991-10-10 | Hoechst Ag | Substituierte azole, verfahren zu deren herstellung, diese enthaltende mittel und deren verwendung |
| AU8757098A (en) * | 1997-06-30 | 1999-02-10 | Ortho-Mcneil Pharmaceutical, Inc. | 2-substituted imidazoles useful in the treatment of inflammatory diseases |
| FR2823747B1 (fr) * | 2001-04-24 | 2003-05-23 | Oreal | Nouveaux composes de la famille des 3-alkyl-(4,5 diphenyl- imidazol-1-yl) et leur utilisation comme anti-inflammatoires |
| US10392381B2 (en) | 2014-07-18 | 2019-08-27 | Ohio University | Prevention and treatment of non-alcoholic fatty liver disease |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE688585A (fr) * | 1965-10-21 | 1967-04-20 | ||
| US3707475A (en) * | 1970-11-16 | 1972-12-26 | Pfizer | Antiinflammatory imidazoles |
| US3929807A (en) * | 1971-05-10 | 1975-12-30 | Ciba Geigy Corp | 2-Substituted-4(5)-(aryl)-5(4)-(2,3 or -4-pyridyl)-imidazoles |
| JPS5343958B2 (fr) * | 1972-07-29 | 1978-11-24 |
-
1978
- 1978-01-05 US US05/865,831 patent/US4182769A/en not_active Expired - Lifetime
- 1978-01-13 DK DK16878A patent/DK16878A/da not_active Application Discontinuation
- 1978-02-06 PT PT67625A patent/PT67625B/pt unknown
- 1978-02-07 CA CA296,605A patent/CA1107286A/fr not_active Expired
- 1978-02-07 IT IT20079/78A patent/IT1092439B/it active
- 1978-02-08 LU LU79028A patent/LU79028A1/fr unknown
- 1978-02-08 IL IL53996A patent/IL53996A/xx unknown
- 1978-02-08 IE IE280/78A patent/IE46454B1/en unknown
- 1978-02-08 SE SE7801466A patent/SE7801466L/xx unknown
- 1978-02-08 AT AT0087078A patent/AT363076B/de not_active IP Right Cessation
- 1978-02-08 SU SU782574555A patent/SU867301A3/ru active
- 1978-02-08 NO NO780432A patent/NO149813C/no unknown
- 1978-02-08 YU YU00289/78A patent/YU28978A/xx unknown
- 1978-02-08 ES ES466793A patent/ES466793A1/es not_active Expired
- 1978-02-08 DE DE19782805166 patent/DE2805166A1/de not_active Withdrawn
- 1978-02-08 FR FR7803517A patent/FR2380264A1/fr not_active Withdrawn
- 1978-02-08 MX MX786830U patent/MX5934E/es unknown
- 1978-02-08 NL NL7801454A patent/NL7801454A/xx not_active Application Discontinuation
- 1978-02-08 AU AU33097/78A patent/AU524360B2/en not_active Expired
- 1978-02-08 GB GB5097/78A patent/GB1587373A/en not_active Expired
- 1978-02-08 NZ NZ186411A patent/NZ186411A/xx unknown
- 1978-02-09 HU HU78DU280A patent/HU181868B/hu unknown
- 1978-02-09 AR AR271047A patent/AR221590A1/es active
- 1978-02-09 FI FI780429A patent/FI68619C/fi not_active IP Right Cessation
- 1978-02-09 CH CH147578A patent/CH643834A5/de not_active IP Right Cessation
- 1978-02-09 GR GR55397A patent/GR64157B/el unknown
- 1978-02-09 JP JP1304778A patent/JPS53130665A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU3309778A (en) | 1979-08-16 |
| AR221590A1 (es) | 1981-02-27 |
| NO149813B (no) | 1984-03-19 |
| GB1587373A (en) | 1981-04-01 |
| ES466793A1 (es) | 1979-08-01 |
| DK16878A (da) | 1978-08-10 |
| IL53996A (en) | 1982-04-30 |
| PT67625B (en) | 1979-07-17 |
| FI68619C (fi) | 1985-10-10 |
| AU524360B2 (en) | 1982-09-16 |
| JPS53130665A (en) | 1978-11-14 |
| ATA87078A (de) | 1980-12-15 |
| MX5934E (es) | 1984-08-30 |
| YU28978A (en) | 1983-01-21 |
| SE7801466L (sv) | 1978-08-10 |
| CH643834A5 (de) | 1984-06-29 |
| FI780429A7 (fi) | 1978-08-10 |
| SU867301A3 (ru) | 1981-09-23 |
| IE780280L (en) | 1978-08-09 |
| HU181868B (en) | 1983-11-28 |
| IT1092439B (it) | 1985-07-12 |
| FR2380264A1 (fr) | 1978-09-08 |
| AT363076B (de) | 1981-07-10 |
| PT67625A (en) | 1978-03-01 |
| IE46454B1 (en) | 1983-06-15 |
| IL53996A0 (en) | 1978-04-30 |
| NO149813C (no) | 1984-06-27 |
| US4182769A (en) | 1980-01-08 |
| DE2805166A1 (de) | 1978-08-10 |
| NL7801454A (nl) | 1978-08-11 |
| NZ186411A (en) | 1981-03-16 |
| NO780432L (no) | 1978-08-10 |
| GR64157B (en) | 1980-02-05 |
| CA1107286A (fr) | 1981-08-18 |
| IT7820079A0 (it) | 1978-02-07 |
| FI68619B (fi) | 1985-06-28 |
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