LU85434A1 - Derives du spirosuccinimide utilisables comme medicaments - Google Patents

Derives du spirosuccinimide utilisables comme medicaments Download PDF

Info

Publication number
LU85434A1
LU85434A1 LU85434A LU85434A LU85434A1 LU 85434 A1 LU85434 A1 LU 85434A1 LU 85434 A LU85434 A LU 85434A LU 85434 A LU85434 A LU 85434A LU 85434 A1 LU85434 A1 LU 85434A1
Authority
LU
Luxembourg
Prior art keywords
group
alkyl
formula
benzyl
alkyl group
Prior art date
Application number
LU85434A
Other languages
English (en)
French (fr)
Original Assignee
Sandoz Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Sa filed Critical Sandoz Sa
Publication of LU85434A1 publication Critical patent/LU85434A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
LU85434A 1983-06-27 1984-06-27 Derives du spirosuccinimide utilisables comme medicaments LU85434A1 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
CH350483 1983-06-27
CH350583 1983-06-27
CH350383 1983-06-27
CH350483 1983-06-27
CH350583 1983-06-27
CH350383 1983-06-27

Publications (1)

Publication Number Publication Date
LU85434A1 true LU85434A1 (fr) 1985-03-26

Family

ID=27174377

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85434A LU85434A1 (fr) 1983-06-27 1984-06-27 Derives du spirosuccinimide utilisables comme medicaments

Country Status (16)

Country Link
AU (1) AU2983384A (de)
DE (1) DE3422411A1 (de)
DK (1) DK310184A (de)
ES (1) ES533735A0 (de)
FI (1) FI842547A7 (de)
FR (1) FR2549061A1 (de)
GB (1) GB2142332A (de)
GR (1) GR82274B (de)
HU (1) HUT36793A (de)
IL (1) IL72218A0 (de)
IT (1) IT1199148B (de)
LU (1) LU85434A1 (de)
NL (1) NL8401907A (de)
PT (1) PT78787B (de)
SE (1) SE8403376L (de)
WO (1) WO1985000171A1 (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3431195A1 (de) * 1984-08-24 1986-03-06 Troponwerke GmbH & Co KG, 5000 Köln Neue benzodiazepine, verfahren zu ihrer herstellung sowie ihre verwendung
EP0273659A1 (de) * 1986-12-27 1988-07-06 Takeda Chemical Industries, Ltd. Azaspiroverbindungen, ihre Herstellung und Verwendung
US5407938A (en) * 1990-04-10 1995-04-18 Israel Institute For Biological Research Certain 1-methyl-piperidine-4-spiro-4'-(1'-3'-oxazolines) and corresponding -(1',3' thiazolines)
JP2800953B2 (ja) * 1990-07-06 1998-09-21 住友製薬株式会社 新規なイミド誘導体
BE1007765A5 (fr) 1994-06-27 1995-10-17 Blagden Ind Plc Fut metallique a ouverture totale.
DE19715758C1 (de) * 1997-04-16 1998-11-05 Man B & W Diesel Gmbh Kolben für eine Hubkolbenbrennkraftmaschine
WO1999032489A1 (en) * 1997-12-23 1999-07-01 Alcon Laboratories, Inc. Muscarinic agents and use thereof to treat glaucoma, myopia and various other conditions
BR0312414A (pt) * 2002-07-05 2005-05-10 Targacept Inc Compostos de n-aril diazaespirociclico e métodos para a preparação e uso dos mesmos
EP1786815B1 (de) * 2003-09-10 2011-08-24 Virochem Pharma Inc. Spiroverbindungen und -verfahren zur modulation von chemokin-rezeptor-aktivität
US9017724B2 (en) 2004-02-24 2015-04-28 The General Hospital Corporation Catalytic radiofluorination
US8257680B1 (en) 2004-02-24 2012-09-04 The General Hospital Corporation Catalytic radiofluorination
JO2676B1 (en) 2004-04-06 2012-06-17 جانسين فارماسوتيكا ان. في Derivatives of second-aza-spiro- (5,4) -dikan and their use as antihistamines
WO2006094948A1 (en) 2005-03-08 2006-09-14 Janssen Pharmaceutica N.V. Diaza-spiro-[4.4]-nonane derivatives as neurokinin (nk1) antagonists
EP3231804B1 (de) * 2008-03-21 2021-03-03 The General Hospital Corporation Verbindungen und zusammensetzungen für den nachweis und die behandlung von morbus alzheimer und verwandten erkrankungen

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1211646B (de) * 1959-03-25 1966-03-03 Sandoz Ag Verfahren zur Herstellung von Spirosuccinimiden und deren Salzen
GB936477A (en) * 1959-03-25 1963-09-11 Sandoz Ltd Improvements in or relating to substituted succinimides
US3198800A (en) * 1964-05-07 1965-08-03 Sandoz Ltd 2, 8-(para-f-4-oxo-butyl)-diazaspiro[4, 5]-decane-1, 3-diones
BE897058A (fr) * 1982-06-25 1983-12-16 Sandoz Sa Utilisation d'un derive du spiro-succinimide dans le traitement de la demence du type alzheimer

Also Published As

Publication number Publication date
HUT36793A (en) 1985-10-28
GB2142332A (en) 1985-01-16
PT78787A (en) 1984-07-01
SE8403376D0 (sv) 1984-06-25
DK310184D0 (da) 1984-06-25
DK310184A (da) 1984-12-28
IT8448458A1 (it) 1985-12-26
SE8403376L (sv) 1984-12-28
AU2983384A (en) 1985-01-03
ES8601202A1 (es) 1985-10-16
FI842547A7 (fi) 1984-12-28
DE3422411A1 (de) 1985-01-03
FI842547A0 (fi) 1984-06-25
NL8401907A (nl) 1985-01-16
WO1985000171A1 (fr) 1985-01-17
GR82274B (de) 1984-12-13
FR2549061A1 (fr) 1985-01-18
IL72218A0 (en) 1984-10-31
ES533735A0 (es) 1985-10-16
IT1199148B (it) 1988-12-30
IT8448458A0 (it) 1984-06-26
GB8416172D0 (en) 1984-08-01
PT78787B (en) 1986-06-05

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