LU90991I2 - Tamiflu ses sels et dérivés pharmaceutiquement acceptables - Google Patents
Tamiflu ses sels et dérivés pharmaceutiquement acceptablesInfo
- Publication number
- LU90991I2 LU90991I2 LU90991C LU90991C LU90991I2 LU 90991 I2 LU90991 I2 LU 90991I2 LU 90991 C LU90991 C LU 90991C LU 90991 C LU90991 C LU 90991C LU 90991 I2 LU90991 I2 LU 90991I2
- Authority
- LU
- Luxembourg
- Prior art keywords
- tamiflu
- derivatives
- pharmaceutically acceptable
- acceptable salts
- neuraminidase
- Prior art date
Links
- PGZUMBJQJWIWGJ-ONAKXNSWSA-N oseltamivir phosphate Chemical compound OP(O)(O)=O.CCOC(=O)C1=C[C@@H](OC(CC)CC)[C@H](NC(C)=O)[C@@H](N)C1 PGZUMBJQJWIWGJ-ONAKXNSWSA-N 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 229940061367 tamiflu Drugs 0.000 title 1
- 102000005348 Neuraminidase Human genes 0.000 abstract 3
- 108010006232 Neuraminidase Proteins 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000002378 acidificating effect Effects 0.000 abstract 1
- 150000001335 aliphatic alkanes Chemical class 0.000 abstract 1
- -1 antibodies Substances 0.000 abstract 1
- 230000000890 antigenic effect Effects 0.000 abstract 1
- 238000003556 assay Methods 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 229920000642 polymer Polymers 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Virology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Pyrane Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Polyesters Or Polycarbonates (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39524595A | 1995-02-27 | 1995-02-27 | |
| US08/476,946 US5866601A (en) | 1995-02-27 | 1995-06-06 | Carbocyclic compounds |
| US58056795A | 1995-12-29 | 1995-12-29 | |
| PCT/US1996/002882 WO1996026933A1 (fr) | 1995-02-27 | 1996-02-26 | Nouveaux inhibiteurs selectifs de neuraminidases virales ou bacteriennes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LU90991I2 true LU90991I2 (fr) | 2003-02-11 |
Family
ID=27410155
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU90991C LU90991I2 (fr) | 1995-02-27 | 2002-12-11 | Tamiflu ses sels et dérivés pharmaceutiquement acceptables |
Country Status (26)
| Country | Link |
|---|---|
| US (3) | US5952375A (fr) |
| EP (1) | EP0759917B1 (fr) |
| JP (3) | JP3300365B2 (fr) |
| KR (1) | KR100447096B1 (fr) |
| CN (2) | CN100409844C (fr) |
| AT (2) | ATE191711T1 (fr) |
| AU (1) | AU720933B2 (fr) |
| BR (2) | BR9607098A (fr) |
| CZ (1) | CZ297945B6 (fr) |
| DE (4) | DE69635231T2 (fr) |
| DK (1) | DK0759917T3 (fr) |
| ES (2) | ES2118674T3 (fr) |
| GR (1) | GR3033914T3 (fr) |
| HU (1) | HU228450B1 (fr) |
| LU (1) | LU90991I2 (fr) |
| MX (1) | MX9706496A (fr) |
| NL (1) | NL300105I2 (fr) |
| NO (1) | NO318455B1 (fr) |
| NZ (1) | NZ306625A (fr) |
| PL (1) | PL194173B1 (fr) |
| PT (1) | PT759917E (fr) |
| RU (1) | RU2181357C2 (fr) |
| SG (1) | SG45864A1 (fr) |
| SI (1) | SI9620042A (fr) |
| UA (1) | UA56128C2 (fr) |
| WO (1) | WO1996026933A1 (fr) |
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|---|---|---|---|---|
| CN100409844C (zh) * | 1995-02-27 | 2008-08-13 | 吉里德科学公司 | 神经氨酸苷酶抑制剂 |
| US5714509A (en) * | 1995-05-03 | 1998-02-03 | The University Of Alabama | Inhibitors of bacterial sialidase and methods of making and using the same |
| US5763483A (en) * | 1995-12-29 | 1998-06-09 | Gilead Sciences, Inc. | Carbocyclic compounds |
| US6093816A (en) | 1996-06-27 | 2000-07-25 | Isis Pharmaceuticals, Inc. | Cationic lipids |
| US6518438B2 (en) | 1996-08-23 | 2003-02-11 | Gilead Sciences, Inc. | Preparation of cyclohexene carboxylate derivatives |
| US5859284A (en) * | 1996-08-23 | 1999-01-12 | Gilead Sciences, Inc. | Preparation of carbocyclic compounds |
| EP0920410B1 (fr) * | 1996-08-23 | 2002-03-27 | Gilead Sciences, Inc. | Preparation de derives de cyclohexene carboxylate |
| CN1238762A (zh) * | 1996-10-21 | 1999-12-15 | 吉里德科学公司 | 哌啶化合物 |
| US5994377A (en) * | 1996-10-21 | 1999-11-30 | Gilead Sciences, Inc. | Piperidine compounds |
| KR20000068986A (ko) * | 1996-11-14 | 2000-11-25 | 리차드웨드레이 | 신규 용도 화합물 및 그 제조방법 |
| WO1999006369A1 (fr) * | 1997-08-01 | 1999-02-11 | University Of Florida | Inhibiteurs de neuraminidase |
| US5886213A (en) * | 1997-08-22 | 1999-03-23 | Gilead Sciences, Inc. | Preparation of carbocyclic compounds |
| US20040053999A1 (en) * | 1997-09-17 | 2004-03-18 | Bischofberger Norbert W. | Novel compounds and methods for synthesis and therapy |
| KR20010024123A (ko) * | 1997-09-17 | 2001-03-26 | 헨슬레이 맥스 디. | 6-원 고리를 갖는 화합물, 그의 제조 방법 및의약물로서의 용도 |
| TW477783B (en) * | 1997-12-12 | 2002-03-01 | Gilead Sciences Inc | Novel compounds useful as neuraminidase inhibitors and pharmaceutical compositions containing same |
| PT1040094E (pt) * | 1997-12-17 | 2009-06-03 | Biocryst Pharm Inc | Compostos de ciclopentano e de ciclopenteno substituídos úteis como inibidores da neuraminidase |
| US6455571B1 (en) | 1998-04-23 | 2002-09-24 | Abbott Laboratories | Inhibitors of neuraminidases |
| WO1999054299A1 (fr) * | 1998-04-23 | 1999-10-28 | Abbott Laboratories | Pyrrolidines utilises comme inhibiteurs de neuraminidases |
| US6518305B1 (en) | 1998-04-23 | 2003-02-11 | Abbott Laboratories | Five-membered carbocyclic and heterocyclic inhibitors of neuraminidases |
| DK0957078T3 (da) * | 1998-05-13 | 2002-04-02 | Hoffmann La Roche | Fremgangsmåde til fremstilling af shikimisyre og derivater deraf |
| WO2000029385A1 (fr) * | 1998-11-13 | 2000-05-25 | Gilead Sciences, Inc. | Composes 1,4,5,6-tetrahydro-pyridaziniques, leur elaboration et leur utilisation comme inhibiteurs des neuraminidases |
| AUPP913999A0 (en) | 1999-03-12 | 1999-04-01 | Biota Scientific Management Pty Ltd | Novel chemical compounds and their use |
| EP1059283B1 (fr) | 1999-06-11 | 2003-05-28 | F. Hoffmann-La Roche Ag | Procédé pour préparer un inhibiteur de la neuraminidase ro-64-0796 |
| DE19930177B4 (de) | 1999-06-30 | 2007-02-08 | Nikolai Vladimirovich Bovin | Intermolekular assoziierende Verbindungen und deren Verwendung |
| WO2001028981A1 (fr) * | 1999-10-19 | 2001-04-26 | Abbott Laboratories | Acide 1-cyclohexene-1-carboxylique et 1-cyclohexene1-1carboxylates comme inhibiteurs de la neuraminidase |
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| EP1486499A1 (fr) | 1999-12-27 | 2004-12-15 | Sagami Chemical Research Center | Dérive d'endo-2,3-epoxy-7-oxabicyclo[2.2.1]heptane-endo-5 acide carboxylique |
| US8642051B2 (en) * | 2000-03-21 | 2014-02-04 | Suzanne Jaffe Stillman | Method of hydration; infusion packet system(s), support member(s), delivery system(s), and method(s); with business model(s) and Method(s) |
| AU2001252578A1 (en) * | 2000-04-25 | 2001-11-07 | Sankyo Company Limited | Preventives for influenza |
| GB0015324D0 (en) * | 2000-06-22 | 2000-08-16 | Biota Scient Management | Medicaments |
| ES2269441T3 (es) | 2000-06-27 | 2007-04-01 | F. Hoffmann-La Roche Ag | Metodo para la preparacion de una composicion. |
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| WO2002092555A1 (fr) * | 2001-05-11 | 2002-11-21 | Sankyo Company, Limited | Derives d'acides sialiques |
| US6964784B2 (en) * | 2002-03-07 | 2005-11-15 | Optigenex, Inc. | Method of preparation and composition of a water soluble extract of the bioactive component of the plant species uncaria for enhancing immune, anti-inflammatory, anti-tumor and dna repair processes of warm blooded animals |
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| JP6453050B2 (ja) * | 2013-11-15 | 2019-01-16 | 国立大学法人富山大学 | 2−デオキシ−2,3−ジデヒドロシアル酸誘導体およびその製造法 |
| CN103819357B (zh) * | 2014-01-28 | 2016-03-16 | 浙江大学 | (-)-有效霉醇叠氮四乙酸酯的制备方法 |
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| KR102339817B1 (ko) | 2016-06-30 | 2021-12-16 | 한미약품 주식회사 | 오셀타미비어 함유 경구용 고형제제 및 그 제조방법 |
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-
1996
- 1996-02-26 CN CNB011247142A patent/CN100409844C/zh not_active Expired - Lifetime
- 1996-02-26 PL PL96322000A patent/PL194173B1/pl unknown
- 1996-02-26 JP JP52644296A patent/JP3300365B2/ja not_active Expired - Lifetime
- 1996-02-26 UA UA97094796A patent/UA56128C2/uk unknown
- 1996-02-26 AT AT96912404T patent/ATE191711T1/de active
- 1996-02-26 DE DE69635231T patent/DE69635231T2/de not_active Expired - Lifetime
- 1996-02-26 CN CNB961901330A patent/CN1185223C/zh not_active Expired - Lifetime
- 1996-02-26 MX MX9706496A patent/MX9706496A/es unknown
- 1996-02-26 DE DE2002199052 patent/DE10299052I1/de active Pending
- 1996-02-26 WO PCT/US1996/002882 patent/WO1996026933A1/fr not_active Ceased
- 1996-02-26 EP EP96912404A patent/EP0759917B1/fr not_active Expired - Lifetime
- 1996-02-26 DE DE69607704T patent/DE69607704T2/de not_active Expired - Lifetime
- 1996-02-26 AT AT99117934T patent/ATE305453T1/de active
- 1996-02-26 BR BR9607098A patent/BR9607098A/pt not_active IP Right Cessation
- 1996-02-26 ES ES96912404T patent/ES2118674T3/es not_active Expired - Lifetime
- 1996-02-26 CZ CZ0269097A patent/CZ297945B6/cs not_active IP Right Cessation
- 1996-02-26 RU RU97116714/04A patent/RU2181357C2/ru active
- 1996-02-26 BR BRPI9607098-6B8D patent/BR9607098B8/pt unknown
- 1996-02-26 KR KR1019970705932A patent/KR100447096B1/ko not_active Expired - Lifetime
- 1996-02-26 US US08/606,624 patent/US5952375A/en not_active Expired - Lifetime
- 1996-02-26 HU HU9800026A patent/HU228450B1/hu unknown
- 1996-02-26 NZ NZ306625A patent/NZ306625A/xx not_active IP Right Cessation
- 1996-02-26 DK DK96912404T patent/DK0759917T3/da active
- 1996-02-26 SG SG1997004840A patent/SG45864A1/en unknown
- 1996-02-26 DE DE0759917T patent/DE759917T1/de active Pending
- 1996-02-26 AU AU53571/96A patent/AU720933B2/en not_active Expired
- 1996-02-26 PT PT96912404T patent/PT759917E/pt unknown
- 1996-02-26 SI SI9620042A patent/SI9620042A/sl not_active IP Right Cessation
- 1996-02-26 ES ES99117934T patent/ES2249863T3/es not_active Expired - Lifetime
- 1996-05-24 US US08/653,034 patent/US20050176758A1/en not_active Abandoned
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1997
- 1997-08-26 NO NO19973908A patent/NO318455B1/no not_active IP Right Cessation
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1999
- 1999-04-08 US US09/288,091 patent/US6225341B1/en not_active Expired - Lifetime
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2000
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2001
- 2001-08-24 JP JP2001255372A patent/JP4234917B2/ja not_active Expired - Lifetime
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2002
- 2002-10-29 NL NL300105C patent/NL300105I2/nl unknown
- 2002-12-11 LU LU90991C patent/LU90991I2/fr unknown
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2005
- 2005-07-15 JP JP2005207906A patent/JP2006036770A/ja not_active Withdrawn
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