LU91225I2 - Plenaxis - Google Patents
PlenaxisInfo
- Publication number
- LU91225I2 LU91225I2 LU91225C LU91225C LU91225I2 LU 91225 I2 LU91225 I2 LU 91225I2 LU 91225 C LU91225 C LU 91225C LU 91225 C LU91225 C LU 91225C LU 91225 I2 LU91225 I2 LU 91225I2
- Authority
- LU
- Luxembourg
- Prior art keywords
- moiety
- peptide compound
- lhrh
- lhrh antagonist
- hydrophilic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/13—Luteinizing hormone-releasing hormone; related peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Gynecology & Obstetrics (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/480,494 US5843901A (en) | 1995-06-07 | 1995-06-07 | LHRH antagonist peptides |
| PCT/US1996/009852 WO1996040757A2 (fr) | 1995-06-07 | 1996-06-07 | Peptides antagonistes de la lh-rh |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LU91225I2 true LU91225I2 (fr) | 2006-05-03 |
Family
ID=23908180
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU91225C LU91225I2 (fr) | 1995-06-07 | 2006-03-03 | Plenaxis |
| LU91857C LU91857I2 (fr) | 1995-06-07 | 2011-08-22 | Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU91857C LU91857I2 (fr) | 1995-06-07 | 2011-08-22 | Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable |
Country Status (13)
| Country | Link |
|---|---|
| US (4) | US5843901A (fr) |
| EP (2) | EP1188768B1 (fr) |
| JP (3) | JP4164125B2 (fr) |
| AT (2) | ATE432941T1 (fr) |
| AU (1) | AU715399B2 (fr) |
| CA (1) | CA2219460C (fr) |
| DE (4) | DE122006000012I1 (fr) |
| DK (2) | DK1188768T3 (fr) |
| ES (2) | ES2177789T3 (fr) |
| HK (1) | HK1045161B (fr) |
| LU (2) | LU91225I2 (fr) |
| PT (2) | PT794961E (fr) |
| WO (1) | WO1996040757A2 (fr) |
Families Citing this family (110)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL117175A (en) * | 1995-02-20 | 2005-11-20 | Sankyo Co | Osteoclastogenesis inhibitory factor protein |
| US5843901A (en) | 1995-06-07 | 1998-12-01 | Advanced Research & Technology Institute | LHRH antagonist peptides |
| US5780435A (en) * | 1995-12-15 | 1998-07-14 | Praecis Pharmaceuticals Incorporated | Methods for treating prostate cancer with LHRH-R antagonists |
| US5968895A (en) | 1996-12-11 | 1999-10-19 | Praecis Pharmaceuticals, Inc. | Pharmaceutical formulations for sustained drug delivery |
| EP2003203A1 (fr) | 1996-12-23 | 2008-12-17 | Immunex Corporation | Ligand pour l'activateur des récepteurs du nf-kappa b, ligand est un membre de la superfamille de TNF |
| US5925730A (en) * | 1997-04-11 | 1999-07-20 | Ferring Bv | GnRH antagonists |
| EP2336168A1 (fr) * | 1997-04-15 | 2011-06-22 | Sankyo Company Limited | Nouvelle protéine et et procédé pour le produire |
| US6316408B1 (en) * | 1997-04-16 | 2001-11-13 | Amgen Inc. | Methods of use for osetoprotegerin binding protein receptors |
| ATE363533T1 (de) | 1997-04-16 | 2007-06-15 | Amgen Inc | Osteoprotegerin bindende proteine und rezeptoren |
| US6217844B1 (en) * | 1998-04-27 | 2001-04-17 | Praecis Pharmaceuticals, Inc. | Methods for detecting lesions in dense breast tissue using LHRH antagonists |
| WO1999055358A1 (fr) * | 1998-04-27 | 1999-11-04 | Praecis Pharmaceuticals Incorporated | Methodes de traitement des bouffees de chaleur et de la gynecomastie |
| US6191115B1 (en) * | 1998-08-12 | 2001-02-20 | Abbott Laboratories | C-terminus modified heptapeptide LHRH analogs |
| US6455499B1 (en) * | 1999-02-23 | 2002-09-24 | Indiana University Foundation | Methods for treating disorders associated with LHRH activity |
| US6703367B1 (en) * | 1999-04-27 | 2004-03-09 | Praecis Pharmaceuticals Inc. | Methods for treating hot flashes and gynaecomastia |
| JP2003506411A (ja) * | 1999-08-09 | 2003-02-18 | トリペップ アクチ ボラゲット | タンパク質重合阻害剤および使用方法 |
| CA2349406C (fr) * | 1999-09-03 | 2011-01-11 | Amgen Inc. | Compositions et procedes permettant la prevention ou le traitement du cancer et de la perte osseuse associee au cancer |
| US20030103978A1 (en) | 2000-02-23 | 2003-06-05 | Amgen Inc. | Selective binding agents of osteoprotegerin binding protein |
| US7109171B2 (en) * | 2000-02-28 | 2006-09-19 | Praecis Pharmaceuticals Inc. | Methods for treating FSH related conditions with GnRH antagonists |
| EP1298142A4 (fr) * | 2000-06-30 | 2005-12-21 | Suntory Ltd | Nouvelle hormone de liberation des gonatrophines, ses peptides precurseurs et genes codant pour eux |
| US6598784B2 (en) * | 2000-12-20 | 2003-07-29 | Meadwestvaco Packaging Syatens, Llc | Beverage carton with strap type carrying handle |
| WO2002056903A2 (fr) * | 2001-01-17 | 2002-07-25 | Praecis Pharmaceuticals Inc. | Methodes pour traiter des etats lies aux hormones au moyen d'une combinaison d'antagonistes de la lhrh et de modulateurs selectifs des recepteurs des oestrogenes |
| EP3342411B1 (fr) | 2001-02-19 | 2019-08-21 | Novartis Pharma AG | Dérivé de rapamycine pour le traitement du cancer du pancréas |
| KR20080091866A (ko) | 2001-05-16 | 2008-10-14 | 노파르티스 아게 | Ν-{5-[4-(4-메틸-피페라지노-메틸)-벤조일아미도]-2-메틸페닐}-4-(3-피리딜)-2-피리미딘-아민 및 화학치료제를 포함하는 배합물 |
| WO2003000156A1 (fr) | 2001-06-22 | 2003-01-03 | Southern Biosystems, Inc. | Implants coaxiaux a liberation prolongee d'ordre 0 |
| MY143582A (en) | 2001-06-26 | 2011-05-31 | Amgent Fremont Inc | Antibodies to opgl |
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| EP1624884A4 (fr) | 2003-04-22 | 2009-08-05 | Ipsen Pharma | Vecteurs de somatostatine |
| GB0320806D0 (en) | 2003-09-05 | 2003-10-08 | Astrazeneca Ab | Therapeutic treatment |
| JP4407322B2 (ja) * | 2004-03-09 | 2010-02-03 | 味の素株式会社 | ペプチドの製造方法 |
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| US20070106271A1 (en) * | 2005-11-09 | 2007-05-10 | Searete Llc, A Limited Liability Corporation | Remote control of substance delivery system |
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| AU2017444054B2 (en) | 2017-12-21 | 2021-10-07 | Hefei Institutes Of Physical Science, Chinese Academy Of Sciences | Class of pyrimidine derivative kinase inhibitors |
| CA3083040A1 (fr) | 2018-01-20 | 2019-07-25 | Sunshine Lake Pharma Co., Ltd. | Composes d'aminopyrimidine substitues et procedes d'utilisation |
| CN109926430A (zh) * | 2018-11-19 | 2019-06-25 | 云南省环境科学研究院(中国昆明高原湖泊国际研究中心) | 一种重金属废渣还原造锍熔炼处置的方法 |
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-
1995
- 1995-06-07 US US08/480,494 patent/US5843901A/en not_active Expired - Lifetime
-
1996
- 1996-06-07 AT AT01204149T patent/ATE432941T1/de active
- 1996-06-07 EP EP01204149A patent/EP1188768B1/fr not_active Expired - Lifetime
- 1996-06-07 DK DK01204149T patent/DK1188768T3/da active
- 1996-06-07 PT PT96919311T patent/PT794961E/pt unknown
- 1996-06-07 ES ES96919311T patent/ES2177789T3/es not_active Expired - Lifetime
- 1996-06-07 DE DE1996623254 patent/DE122006000012I1/de active Pending
- 1996-06-07 PT PT01204149T patent/PT1188768E/pt unknown
- 1996-06-07 DE DE69535963T patent/DE69535963D1/de not_active Expired - Lifetime
- 1996-06-07 DE DE122006000012C patent/DE122006000012I2/de active Active
- 1996-06-07 AT AT96919311T patent/ATE222924T1/de active
- 1996-06-07 EP EP96919311A patent/EP0794961B1/fr not_active Expired - Lifetime
- 1996-06-07 JP JP50205097A patent/JP4164125B2/ja not_active Expired - Fee Related
- 1996-06-07 US US08/973,378 patent/US6423686B1/en not_active Expired - Lifetime
- 1996-06-07 CA CA002219460A patent/CA2219460C/fr not_active Expired - Fee Related
- 1996-06-07 ES ES01204149T patent/ES2326861T3/es not_active Expired - Lifetime
- 1996-06-07 AU AU61680/96A patent/AU715399B2/en not_active Ceased
- 1996-06-07 DE DE69623254T patent/DE69623254T2/de not_active Expired - Lifetime
- 1996-06-07 WO PCT/US1996/009852 patent/WO1996040757A2/fr not_active Ceased
- 1996-06-07 DK DK96919311T patent/DK0794961T3/da active
-
2002
- 2002-04-02 US US10/115,553 patent/US20030040482A1/en not_active Abandoned
- 2002-04-05 US US10/117,364 patent/US7071165B2/en not_active Expired - Fee Related
- 2002-09-11 HK HK02106667.7A patent/HK1045161B/en not_active IP Right Cessation
-
2006
- 2006-03-03 LU LU91225C patent/LU91225I2/fr unknown
-
2007
- 2007-08-13 JP JP2007211155A patent/JP2007302695A/ja not_active Withdrawn
-
2008
- 2008-10-09 JP JP2008263288A patent/JP2009040793A/ja not_active Withdrawn
-
2011
- 2011-08-22 LU LU91857C patent/LU91857I2/fr unknown
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