LU92613I2 - Saxagliptin et ses dérivés pharmaceutiquement acceptables (ONGLYZA) - Google Patents

Saxagliptin et ses dérivés pharmaceutiquement acceptables (ONGLYZA) Download PDF

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Publication number
LU92613I2
LU92613I2 LU92613C LU92613C LU92613I2 LU 92613 I2 LU92613 I2 LU 92613I2 LU 92613 C LU92613 C LU 92613C LU 92613 C LU92613 C LU 92613C LU 92613 I2 LU92613 I2 LU 92613I2
Authority
LU
Luxembourg
Prior art keywords
onglyza
saxagliptin
pharmaceutically acceptable
acceptable derivatives
hyperglycaemia
Prior art date
Application number
LU92613C
Other languages
English (en)
Original Assignee
Royalty Pharma Collection Trust
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7792391&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92613(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Royalty Pharma Collection Trust filed Critical Royalty Pharma Collection Trust
Publication of LU92613I2 publication Critical patent/LU92613I2/fr

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/401—Proline; Derivatives thereof, e.g. captopril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
LU92613C 1996-04-25 2014-12-15 Saxagliptin et ses dérivés pharmaceutiquement acceptables (ONGLYZA) LU92613I2 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19616486.9A DE19616486C5 (de) 1996-04-25 1996-04-25 Verfahren zur Senkung des Blutglukosespiegels in Säugern

Publications (1)

Publication Number Publication Date
LU92613I2 true LU92613I2 (fr) 2015-10-21

Family

ID=7792391

Family Applications (7)

Application Number Title Priority Date Filing Date
LU91334C LU91334I2 (fr) 1996-04-25 2007-04-18 Sitagliptin, ou un sel de celui-ci pharmaceutiquement acceptable, en particulier le sel phosphate (JANUVIA)
LU91382C LU91382I2 (fr) 1996-04-25 2007-12-05 Vildagliptine ou un de ses sels pharmaceutiquementacceptables - GALVUS
LU92613C LU92613I2 (fr) 1996-04-25 2014-12-15 Saxagliptin et ses dérivés pharmaceutiquement acceptables (ONGLYZA)
LU92615C LU92615I2 (fr) 1996-04-25 2014-12-15 Alogliptin et ses dérivés pharmaceutiquement acceptables (VIPIDIA)
LU92611C LU92611I2 (fr) 1996-04-25 2014-12-15 Sitagliptin et ses dérivés pharmaceutiquement acceptables (JANUVIA)
LU92612C LU92612I2 (fr) 1996-04-25 2014-12-15 Vildagliptin et ses dérivés pharmaceutiquement acceptables (GALVUS)
LU92614C LU92614I2 (fr) 1996-04-25 2014-12-15 Linagliptin et ses dérivés pharmaceutiquement acceptables (TRAJENTA)

Family Applications Before (2)

Application Number Title Priority Date Filing Date
LU91334C LU91334I2 (fr) 1996-04-25 2007-04-18 Sitagliptin, ou un sel de celui-ci pharmaceutiquement acceptable, en particulier le sel phosphate (JANUVIA)
LU91382C LU91382I2 (fr) 1996-04-25 2007-12-05 Vildagliptine ou un de ses sels pharmaceutiquementacceptables - GALVUS

Family Applications After (4)

Application Number Title Priority Date Filing Date
LU92615C LU92615I2 (fr) 1996-04-25 2014-12-15 Alogliptin et ses dérivés pharmaceutiquement acceptables (VIPIDIA)
LU92611C LU92611I2 (fr) 1996-04-25 2014-12-15 Sitagliptin et ses dérivés pharmaceutiquement acceptables (JANUVIA)
LU92612C LU92612I2 (fr) 1996-04-25 2014-12-15 Vildagliptin et ses dérivés pharmaceutiquement acceptables (GALVUS)
LU92614C LU92614I2 (fr) 1996-04-25 2014-12-15 Linagliptin et ses dérivés pharmaceutiquement acceptables (TRAJENTA)

Country Status (21)

Country Link
US (1) US6303661B1 (fr)
EP (3) EP1084705B1 (fr)
JP (3) JP2001510442A (fr)
KR (5) KR20100036363A (fr)
CN (2) CN1132578C (fr)
AT (1) ATE202705T1 (fr)
AU (1) AU721477C (fr)
CA (1) CA2252576C (fr)
DE (5) DE122010000020I1 (fr)
DK (2) DK0896538T3 (fr)
ES (2) ES2505665T3 (fr)
FR (1) FR14C0089I1 (fr)
GR (1) GR3036788T3 (fr)
LT (3) LTPA2014045I1 (fr)
LU (7) LU91334I2 (fr)
NL (2) NL300280I2 (fr)
NZ (1) NZ332707A (fr)
PT (2) PT896538E (fr)
RU (1) RU2189233C2 (fr)
SI (1) SI1084705T1 (fr)
WO (1) WO1997040832A1 (fr)

Families Citing this family (300)

* Cited by examiner, † Cited by third party
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