MA23620A1 - Heteroaryl oxazolidinones contenant de l'azote a 6 membres. - Google Patents

Heteroaryl oxazolidinones contenant de l'azote a 6 membres.

Info

Publication number
MA23620A1
MA23620A1 MA23959A MA23959A MA23620A1 MA 23620 A1 MA23620 A1 MA 23620A1 MA 23959 A MA23959 A MA 23959A MA 23959 A MA23959 A MA 23959A MA 23620 A1 MA23620 A1 MA 23620A1
Authority
MA
Morocco
Prior art keywords
members
containing nitrogen
heteroaryl
oxazolidinones containing
heteroaryl oxazolidinones
Prior art date
Application number
MA23959A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MA23620A1 publication Critical patent/MA23620A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Quinoline Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA23959A 1994-07-20 1995-07-19 Heteroaryl oxazolidinones contenant de l'azote a 6 membres. MA23620A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4425612A DE4425612A1 (de) 1994-07-20 1994-07-20 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone

Publications (1)

Publication Number Publication Date
MA23620A1 true MA23620A1 (fr) 1996-04-01

Family

ID=6523632

Family Applications (1)

Application Number Title Priority Date Filing Date
MA23959A MA23620A1 (fr) 1994-07-20 1995-07-19 Heteroaryl oxazolidinones contenant de l'azote a 6 membres.

Country Status (28)

Country Link
US (2) US5627181A (fr)
EP (1) EP0694543A1 (fr)
JP (1) JPH0841056A (fr)
KR (1) KR960004344A (fr)
CN (1) CN1119647A (fr)
AU (1) AU699940B2 (fr)
BG (1) BG99790A (fr)
CA (1) CA2154025A1 (fr)
CO (1) CO4410194A1 (fr)
CZ (1) CZ187295A3 (fr)
DE (1) DE4425612A1 (fr)
DZ (1) DZ1912A1 (fr)
EE (1) EE9500045A (fr)
FI (1) FI953477A7 (fr)
HR (1) HRP950408A2 (fr)
HU (1) HUT75035A (fr)
IL (1) IL114626A (fr)
MA (1) MA23620A1 (fr)
NO (1) NO304468B1 (fr)
NZ (1) NZ272597A (fr)
PE (1) PE35496A1 (fr)
PL (1) PL309686A1 (fr)
RO (1) RO115262B1 (fr)
SK (1) SK91795A3 (fr)
SV (1) SV1995000041A (fr)
TN (1) TNSN95082A1 (fr)
YU (1) YU49295A (fr)
ZA (1) ZA956018B (fr)

Families Citing this family (78)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4425612A1 (de) * 1994-07-20 1996-04-04 Bayer Ag 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
DE19601265A1 (de) * 1996-01-16 1997-07-17 Bayer Ag 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone
DE19601627A1 (de) * 1996-01-18 1997-07-24 Bayer Ag Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
HRP970049A2 (en) 1996-02-06 1998-04-30 Bayer Ag New heteroaryl oxazolidinones
DE19604223A1 (de) 1996-02-06 1997-08-07 Bayer Ag Neue substituierte Oxazolidinone
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
EP0920306A2 (fr) 1996-07-12 1999-06-09 Leukosite, Inc. Antagonistes des recepteurs de la chemokine et procedes d'utilisation de ces derniers
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US6255304B1 (en) 1997-05-30 2001-07-03 Pharmacia & Upjohn Company Oxazolidinone antibacterial agents having a thiocarbonyl functionality
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GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
DE19802239A1 (de) * 1998-01-22 1999-07-29 Bayer Ag Neue mit Bicyclen substituierte Oxazolidinone
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US6239152B1 (en) 1998-01-23 2001-05-29 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
CN1311787A (zh) 1998-06-05 2001-09-05 阿斯特拉曾尼卡有限公司 噁唑烷酮衍生物、其制备方法以及含有它们的药物组合物
MY122454A (en) * 1998-06-05 2006-04-29 Upjohn Co Use of oxazolidinones for the preparation of a medicament for transdermal delivery
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US6420349B1 (en) 1998-08-24 2002-07-16 Bristol-Myers Squibb Company Isoxazolinone antibacterial agents
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US6465456B2 (en) 2000-06-29 2002-10-15 Bristol-Myers Squibb Company Isoxazolinone antibacterial agents
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WO2002018354A1 (fr) * 2000-08-31 2002-03-07 Abbott Laboratories Oxazolidinones et leur utilisation en tant qu'agents antibacteriens
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ATE319710T1 (de) 2000-12-21 2006-03-15 Pharmacia & Upjohn Co Llc Antimikrobielle chinolonderivate und ihre verwendung zur behandlung bakterieller infektionen
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ATE471937T1 (de) * 2003-07-02 2010-07-15 Merck Sharp & Dohme Cyclopropylgruppensubstituierte oxazolidinonantibiotika und derivate davon
CA2529294A1 (fr) * 2003-07-02 2005-01-20 Merck & Co., Inc. Antibiotiques de type oxazolidinones et derives de ceux-ci
AU2004256085B2 (en) * 2003-07-02 2007-12-06 Kyorin, Pharmaceutical Co., Ltd. Cyclopropyl Group Substituted Oxazolydinone Antibiotics and Derivatives Thereof
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JP2007503426A (ja) * 2003-08-25 2007-02-22 ワーナー−ランバート カンパニー リミティド ライアビリティー カンパニー 新規な抗微生物性アリールオキサゾリジノン化合物
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WO2005108370A1 (fr) * 2004-04-16 2005-11-17 Ajinomoto Co., Inc. Composés du benzène
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US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
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Also Published As

Publication number Publication date
IL114626A0 (en) 1995-11-27
NO304468B1 (no) 1998-12-21
BG99790A (en) 1996-04-30
FI953477L (fi) 1996-01-21
NO952865D0 (no) 1995-07-19
JPH0841056A (ja) 1996-02-13
CN1119647A (zh) 1996-04-03
TNSN95082A1 (fr) 1996-02-06
DZ1912A1 (fr) 2002-02-17
HU9502173D0 (en) 1995-09-28
IL114626A (en) 1999-08-17
ZA956018B (en) 1996-03-13
YU49295A (sh) 1998-12-23
KR960004344A (ko) 1996-02-23
HRP950408A2 (en) 1997-04-30
CA2154025A1 (fr) 1996-01-21
SK91795A3 (en) 1996-02-07
HUT75035A (en) 1997-03-28
FI953477A7 (fi) 1996-01-21
EE9500045A (et) 1996-02-15
CZ187295A3 (en) 1996-02-14
EP0694543A1 (fr) 1996-01-31
US5627181A (en) 1997-05-06
NZ272597A (en) 1997-01-29
FI953477A0 (fi) 1995-07-18
AU699940B2 (en) 1998-12-17
RO115262B1 (ro) 1999-12-30
PL309686A1 (en) 1996-01-22
NO952865L (no) 1996-01-22
DE4425612A1 (de) 1996-04-04
CO4410194A1 (es) 1997-01-09
SV1995000041A (es) 1996-03-28
AU2498595A (en) 1996-02-01
PE35496A1 (es) 1996-10-14
US5843967A (en) 1998-12-01

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