MA24296A1 - Derives 6,6- ou 6,7 bicycliques a noyau pyrimido substitues. - Google Patents

Derives 6,6- ou 6,7 bicycliques a noyau pyrimido substitues.

Info

Publication number
MA24296A1
MA24296A1 MA24755A MA24755A MA24296A1 MA 24296 A1 MA24296 A1 MA 24296A1 MA 24755 A MA24755 A MA 24755A MA 24755 A MA24755 A MA 24755A MA 24296 A1 MA24296 A1 MA 24296A1
Authority
MA
Morocco
Prior art keywords
pyrimido
bicyclic derivatives
substituted core
substituted
core
Prior art date
Application number
MA24755A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA24296A1 publication Critical patent/MA24296A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
MA24755A 1996-08-06 1997-08-06 Derives 6,6- ou 6,7 bicycliques a noyau pyrimido substitues. MA24296A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2345396P 1996-08-06 1996-08-06

Publications (1)

Publication Number Publication Date
MA24296A1 true MA24296A1 (fr) 1998-04-01

Family

ID=21815208

Family Applications (1)

Application Number Title Priority Date Filing Date
MA24755A MA24296A1 (fr) 1996-08-06 1997-08-06 Derives 6,6- ou 6,7 bicycliques a noyau pyrimido substitues.

Country Status (40)

Country Link
US (1) US6492520B1 (fr)
EP (1) EP0920429B1 (fr)
JP (1) JP3345021B2 (fr)
KR (1) KR20000029843A (fr)
CN (1) CN1093130C (fr)
AP (1) AP1096A (fr)
AR (1) AR008829A1 (fr)
AT (1) ATE232863T1 (fr)
AU (1) AU709203B2 (fr)
BG (1) BG103143A (fr)
BR (1) BR9710808A (fr)
CA (1) CA2262692C (fr)
CO (1) CO4900060A1 (fr)
CZ (1) CZ292806B6 (fr)
DE (1) DE69719193T2 (fr)
DK (1) DK0920429T3 (fr)
DZ (1) DZ2289A1 (fr)
EA (1) EA003188B1 (fr)
ES (1) ES2191183T3 (fr)
GT (1) GT199700089A (fr)
HR (1) HRP970432B1 (fr)
ID (1) ID17980A (fr)
IL (1) IL128188A0 (fr)
IS (1) IS4948A (fr)
MA (1) MA24296A1 (fr)
NO (1) NO313293B1 (fr)
NZ (1) NZ333727A (fr)
OA (1) OA10970A (fr)
PA (1) PA8435201A1 (fr)
PE (1) PE97098A1 (fr)
PL (1) PL331602A1 (fr)
SA (1) SA97180334A (fr)
SK (1) SK14099A3 (fr)
TN (1) TNSN97135A1 (fr)
TR (1) TR199900228T2 (fr)
TW (1) TW550265B (fr)
UY (1) UY24655A1 (fr)
WO (1) WO1998005661A1 (fr)
YU (1) YU5399A (fr)
ZA (1) ZA976954B (fr)

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Also Published As

Publication number Publication date
AR008829A1 (es) 2000-02-23
EP0920429A1 (fr) 1999-06-09
JP3345021B2 (ja) 2002-11-18
PE97098A1 (es) 1999-01-12
US6492520B1 (en) 2002-12-10
HRP970432B1 (en) 2002-10-31
HRP970432A2 (en) 1998-08-31
DE69719193T2 (de) 2003-09-25
AU709203B2 (en) 1999-08-26
ATE232863T1 (de) 2003-03-15
CN1227552A (zh) 1999-09-01
ES2191183T3 (es) 2003-09-01
NO313293B1 (no) 2002-09-09
EA199900083A1 (ru) 1999-08-26
IL128188A0 (en) 1999-11-30
CA2262692C (fr) 2002-06-11
UY24655A1 (es) 2000-09-29
NZ333727A (en) 2000-09-29
DE69719193D1 (de) 2003-03-27
IS4948A (is) 1999-01-19
AP9701052A0 (en) 1997-10-31
WO1998005661A1 (fr) 1998-02-12
TNSN97135A1 (fr) 2005-03-15
CA2262692A1 (fr) 1998-02-12
TR199900228T2 (xx) 1999-03-22
KR20000029843A (ko) 2000-05-25
PL331602A1 (en) 1999-08-02
EP0920429B1 (fr) 2003-02-19
PA8435201A1 (es) 1999-12-27
NO990544L (no) 1999-03-31
JP2000501116A (ja) 2000-02-02
CN1093130C (zh) 2002-10-23
TW550265B (en) 2003-09-01
DZ2289A1 (fr) 2002-12-25
BR9710808A (pt) 1999-08-17
GT199700089A (es) 1999-01-26
EA003188B1 (ru) 2003-02-27
SK14099A3 (en) 2000-05-16
ZA976954B (en) 1999-02-05
OA10970A (en) 2001-11-05
BG103143A (en) 1999-09-30
AU3356397A (en) 1998-02-25
CO4900060A1 (es) 2000-03-27
CZ292806B6 (cs) 2003-12-17
AP1096A (en) 2002-08-26
SA97180334A (ar) 2005-12-03
NO990544D0 (no) 1999-02-05
YU5399A (sh) 2002-03-18
CZ41199A3 (cs) 2000-01-12
HK1021734A1 (en) 2000-06-30
DK0920429T3 (da) 2003-05-12
ID17980A (id) 1998-02-12

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