ATE232863T1 - Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate - Google Patents

Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate

Info

Publication number
ATE232863T1
ATE232863T1 AT97929472T AT97929472T ATE232863T1 AT E232863 T1 ATE232863 T1 AT E232863T1 AT 97929472 T AT97929472 T AT 97929472T AT 97929472 T AT97929472 T AT 97929472T AT E232863 T1 ATE232863 T1 AT E232863T1
Authority
AT
Austria
Prior art keywords
pyrimido
groups
derivatives containing
containing substituted
substituted pyrido
Prior art date
Application number
AT97929472T
Other languages
English (en)
Inventor
Yuhpyng Liang Chen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE232863T1 publication Critical patent/ATE232863T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
AT97929472T 1996-08-06 1997-07-23 Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate ATE232863T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2345396P 1996-08-06 1996-08-06
PCT/IB1997/000918 WO1998005661A1 (en) 1996-08-06 1997-07-23 Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives

Publications (1)

Publication Number Publication Date
ATE232863T1 true ATE232863T1 (de) 2003-03-15

Family

ID=21815208

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97929472T ATE232863T1 (de) 1996-08-06 1997-07-23 Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate

Country Status (40)

Country Link
US (1) US6492520B1 (de)
EP (1) EP0920429B1 (de)
JP (1) JP3345021B2 (de)
KR (1) KR20000029843A (de)
CN (1) CN1093130C (de)
AP (1) AP1096A (de)
AR (1) AR008829A1 (de)
AT (1) ATE232863T1 (de)
AU (1) AU709203B2 (de)
BG (1) BG103143A (de)
BR (1) BR9710808A (de)
CA (1) CA2262692C (de)
CO (1) CO4900060A1 (de)
CZ (1) CZ292806B6 (de)
DE (1) DE69719193T2 (de)
DK (1) DK0920429T3 (de)
DZ (1) DZ2289A1 (de)
EA (1) EA003188B1 (de)
ES (1) ES2191183T3 (de)
GT (1) GT199700089A (de)
HR (1) HRP970432B1 (de)
ID (1) ID17980A (de)
IL (1) IL128188A0 (de)
IS (1) IS4948A (de)
MA (1) MA24296A1 (de)
NO (1) NO313293B1 (de)
NZ (1) NZ333727A (de)
OA (1) OA10970A (de)
PA (1) PA8435201A1 (de)
PE (1) PE97098A1 (de)
PL (1) PL331602A1 (de)
SA (1) SA97180334A (de)
SK (1) SK14099A3 (de)
TN (1) TNSN97135A1 (de)
TR (1) TR199900228T2 (de)
TW (1) TW550265B (de)
UY (1) UY24655A1 (de)
WO (1) WO1998005661A1 (de)
YU (1) YU5399A (de)
ZA (1) ZA976954B (de)

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Also Published As

Publication number Publication date
IL128188A0 (en) 1999-11-30
CZ292806B6 (cs) 2003-12-17
TR199900228T2 (xx) 1999-03-22
PL331602A1 (en) 1999-08-02
PA8435201A1 (es) 1999-12-27
SK14099A3 (en) 2000-05-16
CA2262692A1 (en) 1998-02-12
NO313293B1 (no) 2002-09-09
OA10970A (en) 2001-11-05
CN1227552A (zh) 1999-09-01
WO1998005661A1 (en) 1998-02-12
JP2000501116A (ja) 2000-02-02
YU5399A (sh) 2002-03-18
HRP970432B1 (en) 2002-10-31
ES2191183T3 (es) 2003-09-01
AP9701052A0 (en) 1997-10-31
EP0920429A1 (de) 1999-06-09
DK0920429T3 (da) 2003-05-12
CO4900060A1 (es) 2000-03-27
UY24655A1 (es) 2000-09-29
AU709203B2 (en) 1999-08-26
EA003188B1 (ru) 2003-02-27
EP0920429B1 (de) 2003-02-19
US6492520B1 (en) 2002-12-10
SA97180334A (ar) 2005-12-03
GT199700089A (es) 1999-01-26
DE69719193T2 (de) 2003-09-25
HK1021734A1 (en) 2000-06-30
ID17980A (id) 1998-02-12
CZ41199A3 (cs) 2000-01-12
DE69719193D1 (de) 2003-03-27
BR9710808A (pt) 1999-08-17
NZ333727A (en) 2000-09-29
EA199900083A1 (ru) 1999-08-26
AP1096A (en) 2002-08-26
NO990544L (no) 1999-03-31
PE97098A1 (es) 1999-01-12
ZA976954B (en) 1999-02-05
KR20000029843A (ko) 2000-05-25
HRP970432A2 (en) 1998-08-31
AR008829A1 (es) 2000-02-23
TNSN97135A1 (fr) 2005-03-15
IS4948A (is) 1999-01-19
TW550265B (en) 2003-09-01
CA2262692C (en) 2002-06-11
CN1093130C (zh) 2002-10-23
MA24296A1 (fr) 1998-04-01
DZ2289A1 (fr) 2002-12-25
JP3345021B2 (ja) 2002-11-18
NO990544D0 (no) 1999-02-05
AU3356397A (en) 1998-02-25
BG103143A (en) 1999-09-30

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