MA24529A1 - Pyrazolopyrimidinones nouvelles, procede pour leur preparation et compositions les contenant . - Google Patents

Pyrazolopyrimidinones nouvelles, procede pour leur preparation et compositions les contenant .

Info

Publication number: MA24529A1
Authority: MA; Morocco
Prior art keywords: preparation; compositions containing; pyrazolopyrimidinones; novel; novel pyrazolopyrimidinones
Prior art date: 1997-04-25

Application number

MA25040A

Other languages

English (en)

Inventor

Wood Anthony

Drek Albert Street Stephen

Edward Bunnage Mark

Paul Mathias John

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-04-25

Filing date

1998-04-22

Publication date

1998-12-31

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27268823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA24529(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1997-04-25 Priority claimed from GBGB9708406.5A external-priority patent/GB9708406D0/en

1997-07-22 Priority claimed from GB9715380A external-priority patent/GB9715380D0/en

1997-10-30 Priority claimed from GBGB9722954.6A external-priority patent/GB9722954D0/en

1998-04-22 Application filed by Pfizer filed Critical Pfizer

1998-12-31 Publication of MA24529A1 publication Critical patent/MA24529A1/fr

Links

239000000203 mixture Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/12—Ophthalmic agents for cataracts
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pulmonology (AREA)
Ophthalmology & Optometry (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Immunology (AREA)
Reproductive Health (AREA)
Hospice & Palliative Care (AREA)
Vascular Medicine (AREA)
Otolaryngology (AREA)
Gynecology & Obstetrics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

MA25040A 1997-04-25 1998-04-22 Pyrazolopyrimidinones nouvelles, procede pour leur preparation et compositions les contenant . MA24529A1 (fr)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB9708406.5A GB9708406D0 (en)	1997-04-25	1997-04-25	Therapeutic agents
GB9715380A GB9715380D0 (en)	1997-07-22	1997-07-22	Therapeutic agents
GBGB9722954.6A GB9722954D0 (en)	1997-10-30	1997-10-30	Therapeutic agents

Publications (1)

Publication Number	Publication Date
MA24529A1 true MA24529A1 (fr)	1998-12-31

Family

ID=27268823

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MA25040A MA24529A1 (fr)	1997-04-25	1998-04-22	Pyrazolopyrimidinones nouvelles, procede pour leur preparation et compositions les contenant .

Country Status (31)

Country	Link
US (2)	US6723719B1 (fr)
EP (1)	EP0977756A1 (fr)
JP (2)	JP3563078B2 (fr)
KR (2)	KR100441229B1 (fr)
CN (2)	CN1188415C (fr)
AP (1)	AP1002A (fr)
AR (1)	AR015595A1 (fr)
AU (1)	AU730670B2 (fr)
BG (1)	BG103828A (fr)
BR (1)	BR9810233A (fr)
CA (1)	CA2288910C (fr)
CO (1)	CO4940472A1 (fr)
CZ (1)	CZ299633B6 (fr)
DZ (1)	DZ2465A1 (fr)
EA (2)	EA002057B1 (fr)
HR (1)	HRP980222B1 (fr)
ID (1)	ID22834A (fr)
IL (5)	IL132276A0 (fr)
IS (1)	IS5200A (fr)
MA (1)	MA24529A1 (fr)
NO (1)	NO314585B1 (fr)
NZ (1)	NZ338075A (fr)
OA (1)	OA11168A (fr)
PA (1)	PA8450401A1 (fr)
PE (1)	PE68699A1 (fr)
PL (1)	PL336586A1 (fr)
RS (1)	RS50118B (fr)
SK (1)	SK285991B6 (fr)
TN (1)	TNSN98053A1 (fr)
TR (1)	TR199902646T2 (fr)
WO (1)	WO1998049166A1 (fr)

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GB9822238D0 (en) *	1998-10-12	1998-12-09	Pfizer Ltd	Process for preparation of pyrazolo[4,3-D]pyrimidin-7-ones and intermediates thereof
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GB9823103D0 (en)	1998-10-23	1998-12-16	Pfizer Ltd	Pharmaceutically active compounds
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EP1222190A1 (fr)	1999-10-11	2002-07-17	Pfizer Limited	Pyrimidine-7-ones 5-(2-substitutees-5-heterocyclylsulphonylpyride-3-yl)-dihydropyrazolo 4,3-d] servant d'inhibiteurs de la phosphodiesterase
GB9923968D0 (en) *	1999-10-11	1999-12-15	Pfizer Ltd	Therapeutic agents
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WO2001047928A2 (fr) *	1999-12-24	2001-07-05	Bayer Aktiengesellschaft	Nouveaux imidazo[1,3,5]triazinones et leur utilisation
CA2395410A1 (fr) *	1999-12-24	2001-07-05	Bayer Aktiengesellschaft	Triazolotriazinones et leur utilisation
KR100358083B1 (ko) *	2000-02-17	2002-10-25	에스케이케미칼주식회사	피롤로피리미디논 유도체와 이의 제조방법, 그리고 이의용도
WO2001087888A1 (fr) *	2000-05-17	2001-11-22	Sk Chemicals Co., Ltd.	Derives de pyrazolopyrimidinone, leur procede de preparation et leur utilisation
KR100377782B1 (ko) *	2000-06-23	2003-03-29	동아제약 주식회사	발기부전 치료에 효과를 갖는 피라졸로피리미디논화합물의 제조방법
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WO2005012256A1 (fr)	2003-07-22	2005-02-10	Astex Therapeutics Limited	Composes 1h-pyrazole 3,4-disubstitues et leur utilisation en tant que kinases dependant des cyclines (cdk) et modulateurs de la glycogene synthase kinase-3 (gsk-3)
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Publication number	Publication date
US20040180944A1 (en)	2004-09-16
CA2288910A1 (fr)	1998-11-05
CN1281588C (zh)	2006-10-25
HRP980222B1 (en)	2003-12-31
JP4036836B2 (ja)	2008-01-23
IL132276A (en)	2006-06-11
EA004315B1 (ru)	2004-02-26
RS50118B (sr)	2009-03-25
US6723719B1 (en)	2004-04-20
WO1998049166A1 (fr)	1998-11-05
TNSN98053A1 (fr)	2005-03-15
PL336586A1 (en)	2000-07-03
AP9801228A0 (en)	1998-06-30
DZ2465A1 (fr)	2003-01-18
CA2288910C (fr)	2003-06-24
AR015595A1 (es)	2001-05-16
JP3563078B2 (ja)	2004-09-08
SK144699A3 (en)	2001-03-12
KR20010020285A (ko)	2001-03-15
JP2000510485A (ja)	2000-08-15
BG103828A (en)	2000-06-30
CZ376799A3 (cs)	2000-04-12
EP0977756A1 (fr)	2000-02-09
BR9810233A (pt)	2000-10-17
IL157647A (en)	2007-05-15
ID22834A (id)	1999-12-09
AU730670B2 (en)	2001-03-08
EA200100504A1 (ru)	2002-02-28
NZ338075A (en)	2000-10-27
NO995211D0 (no)	1999-10-25
AP1002A (en)	2001-08-14
NO995211L (no)	1999-10-25
CN1188415C (zh)	2005-02-09
CO4940472A1 (es)	2000-07-24
HK1027808A1 (en)	2001-01-23
PA8450401A1 (es)	2000-05-24
SK285991B6 (sk)	2008-01-07
PE68699A1 (es)	1999-07-10
IL132276A0 (en)	2001-03-19
EA002057B1 (ru)	2001-12-24
IL157645A (en)	2007-03-08
KR100441229B1 (ko)	2004-07-22
US6916927B2 (en)	2005-07-12
JP2004196820A (ja)	2004-07-15
CZ299633B6 (cs)	2008-09-24
HRP980222A2 (en)	1999-02-28
CN1253561A (zh)	2000-05-17
TR199902646T2 (xx)	2000-05-22
EA199900866A1 (ru)	2000-04-24
YU52499A (fr)	2002-08-12
IS5200A (is)	1999-09-28
OA11168A (en)	2003-04-28
NO314585B1 (no)	2003-04-14
IL157646A (en)	2006-12-10
KR100390612B1 (ko)	2003-07-07
AU7644598A (en)	1998-11-24
CN1626516A (zh)	2005-06-15

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MA26551A1 (fr)	2004-12-20	Agonistes de prostaglandines nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA26558A1 (fr)	2004-12-20	Derives nouveaux de 6-0-methylerythromycine a, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA24832A1 (fr)	1999-12-31	Hydroxamides d'acides (4-arylsulfonylamino)-tetrahydropyranne-4-carboxyliques), procede pour leur preparation et compositions les contenant
MA26559A1 (fr)	2004-12-20	Derives de d-proline, procede pour leur preparation, compositions pharmaceutiques les contenant et leur utilisation
MA24484A1 (fr)	1998-10-01	Atropisomeres de 3-aryl-4(3h)-quinazolinones, procede pour leur preparation et compositions les contenant .
MA26508A1 (fr)	2004-12-20	Formulations pharmaceutiques contenant du variconazole, et procede pour leur preparation.
MA26499A1 (fr)	2004-12-20	Derives de tetrazole, procede pour leur preparation et compositions pharmaceutiques les contenant .
MA26490A1 (fr)	2004-12-20	Derives de tetrahydroisoquinoleine nouveaux, procedes pour leur preparation et compositions pharmaceutiques les contenant.
MA26514A1 (fr)	2004-12-20	Agonistes de prostaglandines, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA26707A1 (fr)	2004-12-20	Azalides nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA26519A1 (fr)	2004-12-20	Derives d'azetidinylpropylpiperidine, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA26487A1 (fr)	2004-12-20	Heterocyclecetohydrazides inhibiteurs de proteases, procede pour leur preparation et compositions pharmaceutiques les contenant .