MA24729A1 - Macrolides nouveaux. - Google Patents

Macrolides nouveaux.

Info

Publication number
MA24729A1
MA24729A1 MA25407A MA25407A MA24729A1 MA 24729 A1 MA24729 A1 MA 24729A1 MA 25407 A MA25407 A MA 25407A MA 25407 A MA25407 A MA 25407A MA 24729 A1 MA24729 A1 MA 24729A1
Authority
MA
Morocco
Prior art keywords
compounds
new macrolides
macrolides
new
infections
Prior art date
Application number
MA25407A
Other languages
English (en)
Inventor
Philip Dirlam John
Alastair Irvine Hamish
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA24729A1 publication Critical patent/MA24729A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

L'INVENTION CONCERNE DES COMPOSÉS DE FORMULE DANS LAQUELLE R1, R2, R3, R4 ET Y REPRÉSENTENT DIVERS RADICAUX. ELLE CONCERNE ÉGALEMENT UN PROCÉDÉ POUR LEUR PRÉPARATION AINSI QUE DES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT. APPLICATION : UTILISATION DE CES COMPOSÉS ET COMPOSITIONS DANS LE TRAITEMENT DE DIVERSES INFECTIONS BACTÉRIENNES ET INFECTIONS PAR DES PROTOZOAIRES.
MA25407A 1998-01-02 1998-12-30 Macrolides nouveaux. MA24729A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7034398P 1998-01-02 1998-01-02

Publications (1)

Publication Number Publication Date
MA24729A1 true MA24729A1 (fr) 1999-07-01

Family

ID=22094723

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25407A MA24729A1 (fr) 1998-01-02 1998-12-30 Macrolides nouveaux.

Country Status (34)

Country Link
US (2) US6472371B1 (fr)
EP (1) EP1044207A1 (fr)
JP (1) JP2002500230A (fr)
KR (1) KR100352809B1 (fr)
CN (1) CN1284081A (fr)
AP (1) AP9801420A0 (fr)
AR (4) AR014948A1 (fr)
AU (1) AU756409B2 (fr)
BG (1) BG104644A (fr)
BR (1) BR9814601A (fr)
CA (1) CA2316919C (fr)
CO (1) CO4970821A1 (fr)
CZ (1) CZ20002458A3 (fr)
DZ (1) DZ2698A1 (fr)
EA (1) EA200000594A1 (fr)
GT (1) GT199800206A (fr)
HR (1) HRP20000442A2 (fr)
HU (1) HUP0100420A3 (fr)
IL (1) IL137024A0 (fr)
IS (1) IS5528A (fr)
MA (1) MA24729A1 (fr)
NO (1) NO20003347L (fr)
NZ (1) NZ504986A (fr)
OA (1) OA11438A (fr)
PA (1) PA8465301A1 (fr)
PE (1) PE20000049A1 (fr)
PL (1) PL341642A1 (fr)
SK (1) SK9782000A3 (fr)
TN (1) TNSN98238A1 (fr)
TW (1) TW520374B (fr)
UY (2) UY25330A1 (fr)
WO (1) WO1999035156A1 (fr)
YU (1) YU41500A (fr)
ZA (1) ZA9811939B (fr)

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AP9801420A0 (en) 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
EP1437360A3 (fr) * 1998-08-19 2005-04-06 Pfizer Products Inc. C11-carbamates des macrolides antibactériens
US6043227A (en) * 1998-08-19 2000-03-28 Pfizer Inc. C11 carbamates of macrolide antibacterials
EP1754700A3 (fr) 1999-01-27 2007-05-09 Kosan Biosciences, Inc. synthese de polycetides
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
CA2370743A1 (fr) 1999-04-16 2000-10-26 Dennis Hlasta Agents antibacteriens cetolides
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
HUP0201516A3 (en) 1999-05-24 2003-03-28 Pfizer Prod Inc 13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
US20050209446A1 (en) * 2002-02-26 2005-09-22 Meiji Seika Kaisha Ltd. Novel 15-membered cyclic azalide, novel 16-membered cyclic diazalide derivative, and process for producing these
AU2005286723A1 (en) 2004-09-23 2006-03-30 Schering-Plough Pty. Limited Control of parasites in animals by the use of novel trifluoromethanesulfonanilide oxime ether derivatives
DE602005017419D1 (de) * 2004-11-19 2009-12-10 Schering Plough Ltd Kontrolle von parasiten bei tieren mittels verwendung von parasitiziden 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitril-derivaten
UA85937C2 (uk) 2004-12-21 2009-03-10 Пфайзер Продактс Інк. Макроліди
CA2609574A1 (fr) * 2005-06-09 2006-12-21 Schering-Plough Ltd. Controle de parasites chez des animaux a l'aide de derives de n-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide et de n-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
CA2672795A1 (fr) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Promedicaments solubles dans l'eau de chloramphenicol, thiamphenicol et analogues de ceux-ci
CN101605756A (zh) * 2006-12-13 2009-12-16 先灵-普劳有限公司 氟苯尼考及其类似物的水溶性前药
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
ES2549731T3 (es) 2007-06-27 2015-11-02 E. I. Du Pont De Nemours And Company Método para el control de plagas en animales
US20090131343A1 (en) * 2007-11-15 2009-05-21 Ly Tam Phan Use of bridged macrolides or tylosin derivatives in treating inflammatory bowel diseases
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
CN102131772B (zh) * 2008-07-30 2015-03-11 英特威国际有限公司 用作氟苯尼考的中间体的*唑啉-保护的氨基二醇化合物的制备方法
UA107804C2 (xx) 2009-08-05 2015-02-25 Du Pont Суміші мезоіонних пестицидів
AU2010279574A1 (en) 2009-08-05 2012-02-09 E. I. Du Pont De Nemours And Company Mesoionic pesticides
MX2012001646A (es) 2009-08-05 2012-03-21 Du Pont Pesticidas mesoionicos.
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
RS54677B1 (sr) 2010-05-27 2016-08-31 E. I. Du Pont De Nemours And Company Kristalni oblici 4-[5-[3-hloro-5-(trifluorometil)fenil]-4,5 -dihidro-5-(trifluorometil)-3-izoksazolil]-n-[2-okso-2-[(2,2,2-trifluoroetil)amino]etil]-1-naftalenkarboksamida
WO2012087630A1 (fr) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Composés de pyridine et de pyrimidine utilisés pour lutter contre des nuisibles invertébrés
BR112013019283A2 (pt) * 2011-01-31 2016-09-13 Meiji Seika Pharma Co Ltd composto, fármaco, composição farmacêutica e uso
CN103619818A (zh) 2011-06-20 2014-03-05 纳幕尔杜邦公司 用于治疗蠕虫感染的杂环化合物
CN102260306B (zh) * 2011-07-22 2012-07-18 山东鲁抗舍里乐药业有限公司 一种制备泰拉霉素的方法
TW201326128A (zh) 2011-11-28 2013-07-01 Du Pont 磺醯胺驅蟲劑
WO2013158422A1 (fr) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Composés hétérocycliques pour la lutte contre des animaux nuisibles invertébrés
WO2014099837A1 (fr) 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anti-helminthique
CN103965273B (zh) * 2013-08-23 2016-05-25 普莱柯生物工程股份有限公司 一种大环内酯类化合物
CN105669798B (zh) * 2013-08-23 2019-07-26 普莱柯生物工程股份有限公司 一种大环内酯类化合物

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HUP0201516A3 (en) 1999-05-24 2003-03-28 Pfizer Prod Inc 13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
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Also Published As

Publication number Publication date
UY25330A1 (es) 2000-12-29
CO4970821A1 (es) 2000-11-07
NO20003347L (no) 2000-08-28
US7015203B2 (en) 2006-03-21
DZ2698A1 (fr) 2003-03-29
WO1999035156A1 (fr) 1999-07-15
IL137024A0 (en) 2001-06-14
HUP0100420A2 (hu) 2001-07-30
BR9814601A (pt) 2000-10-17
AR020551A2 (es) 2002-05-15
EA200000594A1 (ru) 2001-04-23
UY25574A1 (es) 1999-09-27
GT199800206A (es) 2000-06-21
HUP0100420A3 (en) 2003-07-28
HRP20000442A2 (en) 2001-04-30
AR020851A2 (es) 2002-05-29
IS5528A (is) 2000-06-09
US20040092459A1 (en) 2004-05-13
PA8465301A1 (es) 2000-09-29
NO20003347D0 (no) 2000-06-27
TW520374B (en) 2003-02-11
SK9782000A3 (en) 2001-12-03
BG104644A (en) 2001-01-31
OA11438A (en) 2004-04-30
EP1044207A1 (fr) 2000-10-18
PE20000049A1 (es) 2000-02-07
KR20010024818A (ko) 2001-03-26
CA2316919A1 (fr) 1999-07-15
NZ504986A (en) 2003-03-28
YU41500A (sh) 2003-02-28
AP9801420A0 (en) 1998-12-31
AR014948A1 (es) 2001-04-11
AU1444799A (en) 1999-07-26
CZ20002458A3 (cs) 2001-10-17
PL341642A1 (en) 2001-04-23
WO1999035156B1 (fr) 1999-10-21
JP2002500230A (ja) 2002-01-08
TNSN98238A1 (fr) 2005-03-15
AU756409B2 (en) 2003-01-09
CA2316919C (fr) 2004-10-26
KR100352809B1 (ko) 2002-11-01
AR019787A2 (es) 2002-03-13
CN1284081A (zh) 2001-02-14
US6472371B1 (en) 2002-10-29
ZA9811939B (en) 2000-06-30

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