MA27193A1 - Complexes et formulations pharmaceutiques sans gouts, directement compressibles, se dissolvant rapidement - Google Patents
Complexes et formulations pharmaceutiques sans gouts, directement compressibles, se dissolvant rapidementInfo
- Publication number
- MA27193A1 MA27193A1 MA27896A MA27896A MA27193A1 MA 27193 A1 MA27193 A1 MA 27193A1 MA 27896 A MA27896 A MA 27896A MA 27896 A MA27896 A MA 27896A MA 27193 A1 MA27193 A1 MA 27193A1
- Authority
- MA
- Morocco
- Prior art keywords
- pharmaceutical formulations
- complex
- preparation
- taste
- complexes
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 238000002360 preparation method Methods 0.000 abstract 6
- 230000009967 tasteless effect Effects 0.000 abstract 3
- 235000019658 bitter taste Nutrition 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 229920002125 Sokalan® Polymers 0.000 abstract 1
- 238000012512 characterization method Methods 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- RWTNPBWLLIMQHL-UHFFFAOYSA-N fexofenadine Chemical compound C1=CC(C(C)(C(O)=O)C)=CC=C1C(O)CCCN1CCC(C(O)(C=2C=CC=CC=2)C=2C=CC=CC=2)CC1 RWTNPBWLLIMQHL-UHFFFAOYSA-N 0.000 abstract 1
- 229960003592 fexofenadine Drugs 0.000 abstract 1
- 238000002955 isolation Methods 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
EXTRAIT DE L„INVENTION Un complexe effervescent qui est insipide, granuleux, directement compressible et stable composé d'une préparation de base ayant un goût amer, des formulations pharmaceutiques composées du complexe insipide de la préparation de base et des formes de dosage ainsi obtenues sont révélés. La préparation de base peut être le fexofenadine, et le complexe de la préparation de base peut être un complexe de fexofenadine-carbopol. Les procédures pour la préparation, l'isolation et la caractérisation du complexe insipide de la préparation de base ayant un goût amer et les procédures de la production des formulations pharmaceutiques sont révélées également.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN207DE2002 | 2002-03-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA27193A1 true MA27193A1 (fr) | 2005-01-03 |
Family
ID=27773181
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA27896A MA27193A1 (fr) | 2002-03-08 | 2004-10-08 | Complexes et formulations pharmaceutiques sans gouts, directement compressibles, se dissolvant rapidement |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20030170310A1 (fr) |
| AU (1) | AU2003209673B2 (fr) |
| BR (1) | BRPI0308445A2 (fr) |
| MA (1) | MA27193A1 (fr) |
| MX (1) | MXPA04008737A (fr) |
| TN (1) | TNSN04173A1 (fr) |
| WO (1) | WO2003075829A2 (fr) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9703673D0 (en) * | 1997-02-21 | 1997-04-09 | Bradford Particle Design Ltd | Method and apparatus for the formation of particles |
| GB0027357D0 (en) * | 2000-11-09 | 2000-12-27 | Bradford Particle Design Plc | Particle formation methods and their products |
| GB0208742D0 (en) | 2002-04-17 | 2002-05-29 | Bradford Particle Design Ltd | Particulate materials |
| US7582284B2 (en) | 2002-04-17 | 2009-09-01 | Nektar Therapeutics | Particulate materials |
| GB0216562D0 (en) | 2002-04-25 | 2002-08-28 | Bradford Particle Design Ltd | Particulate materials |
| US9339459B2 (en) | 2003-04-24 | 2016-05-17 | Nektar Therapeutics | Particulate materials |
| BRPI0409962A (pt) | 2003-05-08 | 2006-04-25 | Nektar Therapeutics Uk Ltd | co-formulação particulada de uma substáncia ativa e um excipiente, composição farmacêutica ou nutricêutrica, produto farmacêutico ou nutricêutico, método para preparar uma co-formulação particulada de uma substáncia ativa e um excipiente, e, uso de uma substáncia ativa e um excipiente |
| US7282217B1 (en) * | 2003-08-29 | 2007-10-16 | Kv Pharmaceutical Company | Rapidly disintegrable tablets |
| DE10351448A1 (de) * | 2003-11-04 | 2005-06-09 | Bayer Healthcare Ag | Geschmackstoffhaltige Arzneimittelformulierungen mit verbesserten pharmazeutischen Eigenschaften |
| DE602004023764D1 (de) * | 2004-03-19 | 2009-12-03 | Zentiva Kimyasal Ueruenler San | Herstellung von lipid-beschichtetem cefuroxime axetil |
| US20070092553A1 (en) * | 2005-10-21 | 2007-04-26 | Pfab Lp | Compositions and methods of making rapidly dissolving lonically masked formulations |
| EP2043613A1 (fr) * | 2006-07-14 | 2009-04-08 | Fmc Corporation | Forme solide |
| ES2538082T3 (es) | 2007-02-11 | 2015-06-17 | Map Pharmaceuticals Inc | Método de administración terapéutica de DHE para permitir el rápido alivio de migraña mientras que se minimiza el perfil de efectos secundarios |
| WO2008114280A1 (fr) * | 2007-03-21 | 2008-09-25 | Lupin Limited | Nouvelles compositions pharmaceutiques à dose réduite de fexofénadine et de pseudoéphédrine |
| US20080311162A1 (en) * | 2007-05-16 | 2008-12-18 | Olivia Darmuzey | Solid form |
| RU2563623C2 (ru) | 2009-12-02 | 2015-09-20 | Апталис Фарма Лимитед | Микрокапсулы фексофенадина и содержащие их композиции |
| EP2640736B1 (fr) | 2010-11-19 | 2016-08-31 | Cargill, Incorporated | Procédé d'enrichissement de rebaudioside b et/ou de rebaudioside d dans des compositions de glycosides dérivés de stévia par chromatographie d'adsorption-désorption avec une résine adsorbante neutre macroporeuse |
| US9808030B2 (en) | 2011-02-11 | 2017-11-07 | Grain Processing Corporation | Salt composition |
| US20150010622A1 (en) * | 2013-07-03 | 2015-01-08 | R.P. Scherer Technologies, Llc | Capsule formulation comprising fexofenadine |
| US11727516B2 (en) | 2019-06-26 | 2023-08-15 | PharmaCCX, Inc. | System and methods for securing a drug therapy |
| GB2629127A (en) * | 2022-08-31 | 2024-10-23 | Novumgen Ltd | An orodispersible tablet of fexofenadine and its process of preparation |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5840529B2 (ja) * | 1975-09-29 | 1983-09-06 | 明治製菓株式会社 | ケイコウヨウセイザイノセイホウ |
| KR960011236B1 (ko) * | 1987-05-08 | 1996-08-21 | 스미스 클라인 앤드 프렌취 라보라토리스 리미티드 | 제약학적 조성물 및 고체 제형 |
| NL193682C (nl) * | 1987-05-14 | 2000-07-04 | Glaxo Group Ltd | Beklede cefuroximaxetilsamenstelling. |
| US4808411A (en) * | 1987-06-05 | 1989-02-28 | Abbott Laboratories | Antibiotic-polymer compositions |
| US4916161A (en) * | 1988-10-25 | 1990-04-10 | Bristol-Myers Squibb | Taste-masking pharmaceutical agents |
| WO1994008576A1 (fr) * | 1992-10-16 | 1994-04-28 | Glaxo Group Limited | Compositions a base de ranitidine masquant le gout de celle-ci |
| US6027746A (en) * | 1997-04-23 | 2000-02-22 | Warner-Lambert Company | Chewable soft gelatin-encapsulated pharmaceutical adsorbates |
| FR2776302B1 (fr) * | 1998-03-19 | 2002-04-12 | Hoechst Marion Roussel Inc | Nouveau procede de preparation de la fexofenadine |
| US6051585A (en) * | 1998-12-07 | 2000-04-18 | Weinstein; Robert E. | Single-dose antihistamine/decongestant formulations for treating rhinitis |
| US6723348B2 (en) * | 2001-11-16 | 2004-04-20 | Ethypharm | Orodispersible tablets containing fexofenadine |
| US6667026B1 (en) * | 2002-03-15 | 2003-12-23 | Pocono Falls, Inc. | Allergic contact dermatitis treatment and composition therefor |
-
2003
- 2003-03-07 AU AU2003209673A patent/AU2003209673B2/en not_active Ceased
- 2003-03-07 MX MXPA04008737A patent/MXPA04008737A/es active IP Right Grant
- 2003-03-07 WO PCT/IN2003/000048 patent/WO2003075829A2/fr not_active Ceased
- 2003-03-07 US US10/383,433 patent/US20030170310A1/en not_active Abandoned
- 2003-03-07 BR BRPI0308445A patent/BRPI0308445A2/pt not_active IP Right Cessation
-
2004
- 2004-09-08 TN TNP2004000173A patent/TNSN04173A1/en unknown
- 2004-10-08 MA MA27896A patent/MA27193A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA04008737A (es) | 2005-07-13 |
| AU2003209673B2 (en) | 2007-10-18 |
| WO2003075829A3 (fr) | 2004-11-18 |
| AU2003209673A1 (en) | 2003-09-22 |
| TNSN04173A1 (en) | 2007-03-12 |
| US20030170310A1 (en) | 2003-09-11 |
| WO2003075829A2 (fr) | 2003-09-18 |
| BRPI0308445A2 (pt) | 2016-08-02 |
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