MA28267A1 - Formulations orales d'agonistes du recepteur 5-ht, utilisations et methodes de traitement faisant intervenir celles-ci - Google Patents
Formulations orales d'agonistes du recepteur 5-ht, utilisations et methodes de traitement faisant intervenir celles-ciInfo
- Publication number
- MA28267A1 MA28267A1 MA28986A MA28986A MA28267A1 MA 28267 A1 MA28267 A1 MA 28267A1 MA 28986 A MA28986 A MA 28986A MA 28986 A MA28986 A MA 28986A MA 28267 A1 MA28267 A1 MA 28267A1
- Authority
- MA
- Morocco
- Prior art keywords
- treatment
- methods
- same
- receptor agonists
- oral formulations
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 108091032151 5-hydroxytryptamine receptor family Proteins 0.000 title 1
- 102000014630 G protein-coupled serotonin receptor activity proteins Human genes 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
- 239000011162 core material Substances 0.000 abstract 2
- 239000011248 coating agent Substances 0.000 abstract 1
- 238000000576 coating method Methods 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000952 serotonin receptor agonist Substances 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
- 239000002982 water resistant material Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/288—Compounds of unknown constitution, e.g. material from plants or animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/282—Organic compounds, e.g. fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5015—Organic compounds, e.g. fats, sugars
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Zoology (AREA)
- Botany (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention concerne une formulation orale acceptable sur le plan pharmaceutique qui comprend un matériau central comportant une dose efficace sur le plan thérapeutique d'un agoniste du récepteur 5-HT, ou un sel, un solvate ou un dérivé associé acceptable sur le plan pharmaceutique ; ledit matériau central étant pourvu d'un revêtement sensiblement résistant à l'eau qui comprend un ou plusieurs matériaux sensiblement résistants à l'eau.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0325383A GB2407498B (en) | 2003-10-30 | 2003-10-30 | Oral formulations for 5-HT receptor agonists with reduced degradation of active ingredient |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA28267A1 true MA28267A1 (fr) | 2006-11-01 |
Family
ID=29725668
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA28986A MA28267A1 (fr) | 2003-10-30 | 2006-04-28 | Formulations orales d'agonistes du recepteur 5-ht, utilisations et methodes de traitement faisant intervenir celles-ci |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US20070077299A1 (fr) |
| EP (1) | EP1682100A2 (fr) |
| JP (1) | JP2007533652A (fr) |
| KR (1) | KR20060109919A (fr) |
| CN (1) | CN1901889A (fr) |
| AP (1) | AP2006003613A0 (fr) |
| AU (1) | AU2004287257B2 (fr) |
| BR (1) | BRPI0415803A (fr) |
| CA (1) | CA2544258A1 (fr) |
| GB (1) | GB2407498B (fr) |
| IL (1) | IL175303A0 (fr) |
| MA (1) | MA28267A1 (fr) |
| MX (1) | MXPA06004846A (fr) |
| WO (1) | WO2005044222A2 (fr) |
| ZA (1) | ZA200603438B (fr) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7901713B2 (en) * | 2001-06-20 | 2011-03-08 | Metaproteomics, Llc | Inhibition of COX-2 and/or 5-LOX activity by fractions isolated or derived from hops |
| GB2407498B (en) * | 2003-10-30 | 2008-06-11 | Cipla Ltd | Oral formulations for 5-HT receptor agonists with reduced degradation of active ingredient |
| US20070099931A1 (en) * | 2004-03-19 | 2007-05-03 | Wyeth | Pharmaceutical dosage forms and compositions |
| CA2620491A1 (fr) * | 2005-09-09 | 2007-03-15 | Wyeth | Formes dosifiees pharmaceutiques et compositions associees |
| CN101365450A (zh) * | 2006-02-09 | 2009-02-11 | 特瓦制药工业有限公司 | 孟鲁司特钠的稳定药物制剂 |
| ES2527448T3 (es) * | 2008-04-28 | 2015-01-23 | Zogenix, Inc. | Nuevas formulaciones para el tratamiento de la migraña |
| CN101757623B (zh) * | 2008-10-09 | 2013-12-04 | 北京德众万全药物技术开发有限公司 | 一种5-ht受体激动剂固体药物组合物 |
| JP6393274B2 (ja) | 2012-12-19 | 2018-09-19 | バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Animal Health Gmbh | 改良された許容性および良好な保存安定性を有する錠剤 |
| US9511561B2 (en) * | 2013-09-12 | 2016-12-06 | R.R. Donnelley & Sons Company | Multi-layer forms and methods of manufacturing the same |
| CN104739774A (zh) * | 2013-12-26 | 2015-07-01 | 康普药业股份有限公司 | 一种琥珀酸舒马曲坦颗粒及其制备工艺 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2614020C2 (de) * | 1976-04-01 | 1984-01-26 | Knoll Ag, 6700 Ludwigshafen | Verfahren zur Isolierung von Presslingen |
| GB8419575D0 (en) * | 1984-08-01 | 1984-09-05 | Glaxo Group Ltd | Chemical compounds |
| GB9104890D0 (en) * | 1991-03-08 | 1991-04-24 | Glaxo Group Ltd | Compositions |
| US5807571A (en) * | 1993-05-06 | 1998-09-15 | Lts Lohmann Therapie-Systeme Gmbh | Transdermal therapeutic systems for administering indole serotonin agonists |
| JP2987813B2 (ja) * | 1993-07-12 | 1999-12-06 | 住友製薬株式会社 | ワックス被覆製剤およびその製法 |
| JPH09216817A (ja) * | 1996-02-08 | 1997-08-19 | Amano Pharmaceut Co Ltd | 防湿性且つ易水崩壊性コーティング製剤 |
| EP0999841B1 (fr) * | 1997-07-03 | 2001-10-17 | Pfizer Limited | Compositions pharmaceutiques contenant l'hemisulfate d'eletriptane et de la cafeine |
| GB9816556D0 (en) * | 1998-07-30 | 1998-09-30 | Pfizer Ltd | Therapy |
| EP1064938A1 (fr) * | 1999-06-28 | 2001-01-03 | Sanofi-Synthelabo | Formes pharmaceutiques à libération contrôlée avec au moins une impulsion temporelle |
| US20030180352A1 (en) * | 1999-11-23 | 2003-09-25 | Patel Mahesh V. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| AT500063A1 (de) * | 1999-11-23 | 2005-10-15 | Sandoz Ag | Beschichtete tablettenkerne |
| GB0018968D0 (en) * | 2000-08-02 | 2000-09-20 | Pfizer Ltd | Particulate composition |
| CA2446904A1 (fr) * | 2001-05-24 | 2003-04-03 | Alexza Pharmaceuticals, Inc. | Administration d'esters medicamenteux par inhalation |
| MXPA04006163A (es) * | 2001-12-20 | 2004-11-01 | Pharmacia Corp | Formas de dosis de liberacion sostenida del orden-cero y metodo de fabricacion de las mismas. |
| BR0312795A (pt) * | 2002-07-19 | 2005-05-10 | Ranbaxy Lab Ltd | Apresentação farmacêutica de sumatriptan, processo para sua preparação e método para tratar a enxaqueca |
| GB2407498B (en) * | 2003-10-30 | 2008-06-11 | Cipla Ltd | Oral formulations for 5-HT receptor agonists with reduced degradation of active ingredient |
-
2003
- 2003-10-30 GB GB0325383A patent/GB2407498B/en not_active Expired - Fee Related
-
2004
- 2004-11-01 CN CNA2004800396624A patent/CN1901889A/zh active Pending
- 2004-11-01 CA CA002544258A patent/CA2544258A1/fr not_active Abandoned
- 2004-11-01 ZA ZA200603438A patent/ZA200603438B/en unknown
- 2004-11-01 AP AP2006003613A patent/AP2006003613A0/xx unknown
- 2004-11-01 JP JP2006537436A patent/JP2007533652A/ja active Pending
- 2004-11-01 KR KR1020067010245A patent/KR20060109919A/ko not_active Ceased
- 2004-11-01 AU AU2004287257A patent/AU2004287257B2/en not_active Ceased
- 2004-11-01 BR BRPI0415803-2A patent/BRPI0415803A/pt not_active Application Discontinuation
- 2004-11-01 MX MXPA06004846A patent/MXPA06004846A/es unknown
- 2004-11-01 WO PCT/GB2004/004605 patent/WO2005044222A2/fr not_active Ceased
- 2004-11-01 US US10/577,760 patent/US20070077299A1/en not_active Abandoned
- 2004-11-01 EP EP04798341A patent/EP1682100A2/fr not_active Withdrawn
-
2006
- 2006-04-27 IL IL175303A patent/IL175303A0/en unknown
- 2006-04-28 MA MA28986A patent/MA28267A1/fr unknown
-
2010
- 2010-09-22 US US12/887,599 patent/US20110008412A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| IL175303A0 (en) | 2006-09-05 |
| AU2004287257A2 (en) | 2005-05-19 |
| AP2006003613A0 (en) | 2006-06-30 |
| MXPA06004846A (es) | 2006-07-06 |
| KR20060109919A (ko) | 2006-10-23 |
| JP2007533652A (ja) | 2007-11-22 |
| GB0325383D0 (en) | 2003-12-03 |
| CN1901889A (zh) | 2007-01-24 |
| BRPI0415803A (pt) | 2006-12-26 |
| GB2407498A (en) | 2005-05-04 |
| EP1682100A2 (fr) | 2006-07-26 |
| WO2005044222A3 (fr) | 2006-01-12 |
| AU2004287257A1 (en) | 2005-05-19 |
| AU2004287257B2 (en) | 2011-04-14 |
| GB2407498B (en) | 2008-06-11 |
| US20110008412A1 (en) | 2011-01-13 |
| US20070077299A1 (en) | 2007-04-05 |
| WO2005044222A2 (fr) | 2005-05-19 |
| ZA200603438B (en) | 2008-01-30 |
| CA2544258A1 (fr) | 2005-05-19 |
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