MA29376B1 - Formes pharmaceutiques a proprietes pharmacocinetique ameliorees. - Google Patents

Formes pharmaceutiques a proprietes pharmacocinetique ameliorees.

Info

Publication number
MA29376B1
MA29376B1 MA30265A MA30265A MA29376B1 MA 29376 B1 MA29376 B1 MA 29376B1 MA 30265 A MA30265 A MA 30265A MA 30265 A MA30265 A MA 30265A MA 29376 B1 MA29376 B1 MA 29376B1
Authority
MA
Morocco
Prior art keywords
pharmacokinetic properties
pharmaceutical forms
improved pharmacokinetic
formulations
vardenafil
Prior art date
Application number
MA30265A
Other languages
English (en)
Inventor
Peter Serno
Roland Heinig
Kerstin Pauli
Yutaka Hayauchi
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36264023&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA29376(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of MA29376B1 publication Critical patent/MA29376B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

LA PRÉSENTE INVENTION CONCERNE DE NOUVELLES FORMULATIONS PHARMACEUTIQUES DE VARDÉNAFIL À DISSOLUTION RAPIDE EN BOUCHE, LESQUELLES FORMULATIONS INDUISENT UNE AUGMENTATION DE LA BIODISPONIBILITÉ ET UNE COURBE DE CONCENTRATION PLASMATIQUE EN PLATEAU. CETTE INVENTION CONCERNE ÉGALEMENT UN PROCÉDÉ DE PRODUCTION DESDITES FORMULATIONS.
MA30265A 2005-03-01 2007-10-01 Formes pharmaceutiques a proprietes pharmacocinetique ameliorees. MA29376B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005009240A DE102005009240A1 (de) 2005-03-01 2005-03-01 Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften

Publications (1)

Publication Number Publication Date
MA29376B1 true MA29376B1 (fr) 2008-04-01

Family

ID=36264023

Family Applications (1)

Application Number Title Priority Date Filing Date
MA30265A MA29376B1 (fr) 2005-03-01 2007-10-01 Formes pharmaceutiques a proprietes pharmacocinetique ameliorees.

Country Status (38)

Country Link
US (2) US8613950B2 (fr)
EP (2) EP2377523A1 (fr)
JP (1) JP5122984B2 (fr)
KR (1) KR101360526B1 (fr)
CN (2) CN102198140B (fr)
AR (2) AR053552A1 (fr)
AT (1) ATE552828T1 (fr)
AU (1) AU2006220100B2 (fr)
BR (1) BRPI0609375A2 (fr)
CA (1) CA2599617C (fr)
CR (2) CR9339A (fr)
CY (1) CY1112874T1 (fr)
DE (1) DE102005009240A1 (fr)
DK (1) DK1858490T3 (fr)
DO (1) DOP2006000049A (fr)
ES (1) ES2384109T3 (fr)
GT (1) GT200600097A (fr)
HN (1) HN2006009000A (fr)
HR (1) HRP20120545T1 (fr)
IL (2) IL185552A (fr)
MA (1) MA29376B1 (fr)
MX (1) MX2007010527A (fr)
MY (2) MY177386A (fr)
NO (2) NO332368B1 (fr)
NZ (1) NZ561004A (fr)
PE (2) PE20100740A1 (fr)
PL (1) PL1858490T3 (fr)
PT (1) PT1858490E (fr)
RS (1) RS52374B (fr)
RU (2) RU2423970C2 (fr)
SG (1) SG160330A1 (fr)
SI (1) SI1858490T1 (fr)
TN (1) TNSN07336A1 (fr)
TW (1) TWI387465B (fr)
UA (1) UA93200C2 (fr)
UY (1) UY29395A1 (fr)
WO (1) WO2006092207A1 (fr)
ZA (1) ZA200707320B (fr)

Families Citing this family (21)

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FR2906140B1 (fr) * 2006-09-22 2008-12-05 Philippe Perovitch Forme galenique pour l'administration par voie trans-muqueuse de principes actifs
DE102007027067A1 (de) 2007-06-12 2008-12-18 Ratiopharm Gmbh Verfahren zur Herstellung eines Arzneimittels enthaltend Vardenafil Hydrochlorid Trihydrat
DE102009020888A1 (de) * 2009-05-12 2010-11-18 Ratiopharm Gmbh Schmelztablette, enthaltend ein Vardenafil-Salz
US8920839B2 (en) 2009-05-20 2014-12-30 Sumitomo Dainippon Pharma Co., Ltd. Dry-coated orally-disintegrating tablet
GB2497728A (en) 2011-12-14 2013-06-26 Londonpharma Ltd Statin formulations for transmucosal delivery
GB2497933B (en) * 2011-12-21 2014-12-24 Londonpharma Ltd Drug delivery technology
CN103372014B (zh) * 2012-04-26 2015-10-21 齐鲁制药有限公司 一种能快速溶出、稳定的盐酸伐地那非口服固体制剂及其制备方法
CN102727455B (zh) * 2012-07-03 2016-06-29 北京科信必成医药科技发展有限公司 一种他达那非口腔崩解片及其制备方法
WO2015089105A1 (fr) 2013-12-09 2015-06-18 Respira Therapeutics, Inc. Formulations en poudre d'inhibiteur pde5 et procédés y associés
CN110193015A (zh) * 2018-02-27 2019-09-03 广州朗圣药业有限公司 一种盐酸伐地那非口腔崩解片及其制备方法
CN108272765B (zh) * 2018-04-26 2021-02-02 江西杏林白马药业股份有限公司 含盐酸伐地那非的药物组合物、口崩片及其制备、应用
SG11202010792TA (en) 2018-05-02 2020-11-27 Ferring Bv Improved pharmaceutical formulations
CN110840851A (zh) * 2019-08-16 2020-02-28 天津仁卫生物医药科技有限公司 一种盐酸伐地那非口腔崩解片及其制备方法
IT201900020350A1 (it) 2019-11-05 2021-05-05 Alpex Pharma Sa Formulazione orodispersibile di vardenafil
EP4096791A1 (fr) 2020-01-31 2022-12-07 Nanocopoeia LLC Microparticules de nilotinib amorphe et leurs utilisations
IL297776A (en) 2020-04-30 2022-12-01 Nanocopoeia Llc Orally disintegrating tablets containing an amorphous solid dispersion of nalotinib
AU2021280285A1 (en) * 2020-05-26 2023-02-02 Strategic Drug Solutions, Inc. Formulations and methods for treating erectile dysfunction
CN114848603B (zh) * 2022-04-25 2023-12-12 湖北菲瑞生物药业有限公司 一种伐地那非冻干闪释片及其制备工艺

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Also Published As

Publication number Publication date
EP1858490A1 (fr) 2007-11-28
SI1858490T1 (sl) 2012-07-31
JP2008531614A (ja) 2008-08-14
TWI387465B (zh) 2013-03-01
TNSN07336A1 (en) 2008-12-31
IL246548A0 (en) 2016-08-31
IL185552A (en) 2017-06-29
CR20130381A (es) 2013-09-12
EP2377523A1 (fr) 2011-10-19
HK1118457A1 (en) 2009-02-13
MY148698A (en) 2013-05-31
AR053552A1 (es) 2007-05-09
NO344546B1 (no) 2020-01-27
PE20061015A1 (es) 2006-10-20
NO20120203L (no) 2007-09-27
RU2481110C2 (ru) 2013-05-10
NO20074848L (no) 2007-09-27
US20080249096A1 (en) 2008-10-09
CA2599617A1 (fr) 2006-09-08
HN2006009000A (es) 2010-08-05
WO2006092207A1 (fr) 2006-09-08
RU2011111106A (ru) 2012-09-27
JP5122984B2 (ja) 2013-01-16
PL1858490T3 (pl) 2012-09-28
ATE552828T1 (de) 2012-04-15
RU2423970C2 (ru) 2011-07-20
DK1858490T3 (da) 2012-07-23
CN102198140B (zh) 2016-06-08
EP1858490B1 (fr) 2012-04-11
CY1112874T1 (el) 2016-04-13
RU2007135982A (ru) 2009-04-10
RS52374B (sr) 2012-12-31
CA2599617C (fr) 2012-01-10
CR9339A (es) 2007-12-17
US20140186444A1 (en) 2014-07-03
GT200600097A (es) 2006-11-13
HRP20120545T1 (hr) 2012-07-31
AR111572A2 (es) 2019-07-31
PE20100740A1 (es) 2010-10-28
CN101141950B (zh) 2011-06-08
AU2006220100B2 (en) 2011-08-18
TW200640503A (en) 2006-12-01
ES2384109T3 (es) 2012-06-29
PT1858490E (pt) 2012-06-19
NZ561004A (en) 2010-12-24
DE102005009240A1 (de) 2006-09-07
DOP2006000049A (es) 2006-10-31
CN101141950A (zh) 2008-03-12
UY29395A1 (es) 2006-10-02
SG160330A1 (en) 2010-04-29
CN102198140A (zh) 2011-09-28
US8613950B2 (en) 2013-12-24
NO332368B1 (no) 2012-09-03
KR101360526B1 (ko) 2014-02-21
IL185552A0 (en) 2008-01-06
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BRPI0609375A2 (pt) 2010-03-30
ZA200707320B (en) 2009-08-26
MY177386A (en) 2020-09-14
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