MA31796B1 - Composes organiques - Google Patents
Composes organiquesInfo
- Publication number
- MA31796B1 MA31796B1 MA32802A MA32802A MA31796B1 MA 31796 B1 MA31796 B1 MA 31796B1 MA 32802 A MA32802 A MA 32802A MA 32802 A MA32802 A MA 32802A MA 31796 B1 MA31796 B1 MA 31796B1
- Authority
- MA
- Morocco
- Prior art keywords
- antagonist
- inhibitor
- component
- adrenoreceptor
- beta
- Prior art date
Links
- 150000002894 organic compounds Chemical class 0.000 title 1
- 239000005557 antagonist Substances 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003149 muscarinic antagonist Substances 0.000 abstract 2
- 229940122086 Adenosine A2a receptor agonist Drugs 0.000 abstract 1
- 208000000884 Airway Obstruction Diseases 0.000 abstract 1
- 229940121786 Beta 2 adrenoreceptor agonist Drugs 0.000 abstract 1
- 229940123415 Beta 2 adrenoreceptor antagonist Drugs 0.000 abstract 1
- 102100039705 Beta-2 adrenergic receptor Human genes 0.000 abstract 1
- 101710152983 Beta-2 adrenergic receptor Proteins 0.000 abstract 1
- 229940123169 Caspase inhibitor Drugs 0.000 abstract 1
- 229940126052 ENaC inhibitor Drugs 0.000 abstract 1
- 229940121948 Muscarinic receptor antagonist Drugs 0.000 abstract 1
- 229940123932 Phosphodiesterase 4 inhibitor Drugs 0.000 abstract 1
- 229940122055 Serine protease inhibitor Drugs 0.000 abstract 1
- 101710102218 Serine protease inhibitor Proteins 0.000 abstract 1
- GUGOEEXESWIERI-UHFFFAOYSA-N Terfenadine Chemical compound C1=CC(C(C)(C)C)=CC=C1C(O)CCCN1CCC(C(O)(C=2C=CC=CC=2)C=2C=CC=CC=2)CC1 GUGOEEXESWIERI-UHFFFAOYSA-N 0.000 abstract 1
- 239000002465 adenosine A2a receptor agonist Substances 0.000 abstract 1
- 230000001387 anti-histamine Effects 0.000 abstract 1
- 239000000739 antihistaminic agent Substances 0.000 abstract 1
- 239000003246 corticosteroid Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000002713 epithelial sodium channel blocking agent Substances 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 150000002615 leukotriene B4 derivatives Chemical class 0.000 abstract 1
- 239000002587 phosphodiesterase IV inhibitor Substances 0.000 abstract 1
- 239000003001 serine protease inhibitor Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
L'invention concerne un médicament comprenant, séparément ou ensemble :, un composant (a) qui est un agoniste de récepteur d'adénosine a2a tel que défini dans la description; et un composant (b) qui est constitué d'un ou plusieurs composés choisis parmi : (i) un corticostéroïde, (ii) un agoniste d'adrénorécepteur bêta-2, (iii) un agent antimuscarinique, (iv) un antagoniste de a 2b, (v) un antihistaminique, (vi) un inhibiteur de caspase, (vii) un inhibiteur de enac, (viii) un antagoniste de ltb4, (ix) un antagoniste de ltd4, (x) un inhibiteur de sérine protéase, (xi) un inhibiteur de pde4 et (xii) un composé à double action agoniste d'adrénorécepteur bêta-2/antagoniste muscarinique, pour une administration simultanée, séquentielle ou séparée dans le traitement d'une maladie inflammatoire ou d'obstruction des voies aériennes.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07118721 | 2007-10-17 | ||
| PCT/EP2008/063869 WO2009050198A2 (fr) | 2007-10-17 | 2008-10-15 | Composés organiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA31796B1 true MA31796B1 (fr) | 2010-10-01 |
Family
ID=39185790
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA32802A MA31796B1 (fr) | 2007-10-17 | 2010-04-30 | Composes organiques |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20090181934A1 (fr) |
| EP (1) | EP2211865A2 (fr) |
| JP (1) | JP2011500630A (fr) |
| KR (1) | KR20100075925A (fr) |
| CN (1) | CN101827596A (fr) |
| AR (1) | AR068879A1 (fr) |
| AU (1) | AU2008313788A1 (fr) |
| BR (1) | BRPI0818005A2 (fr) |
| CA (1) | CA2702942A1 (fr) |
| CL (1) | CL2008003057A1 (fr) |
| CR (1) | CR11341A (fr) |
| CU (1) | CU20100065A7 (fr) |
| EA (1) | EA201000617A1 (fr) |
| IL (1) | IL204723A0 (fr) |
| MA (1) | MA31796B1 (fr) |
| MX (1) | MX2010004252A (fr) |
| PE (1) | PE20091392A1 (fr) |
| TN (1) | TN2010000168A1 (fr) |
| TW (1) | TW200927129A (fr) |
| WO (1) | WO2009050198A2 (fr) |
| ZA (1) | ZA201002336B (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GT200500281A (es) * | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
| GB0500785D0 (en) | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
| GB0607945D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607953D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607948D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607944D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607950D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| PT2322525E (pt) * | 2006-04-21 | 2013-12-26 | Novartis Ag | Derivados de purina para utilização como agonistas do recetor de adenosina a2a |
| EP1889846A1 (fr) | 2006-07-13 | 2008-02-20 | Novartis AG | Dérivés de purine comme agonistes du recepteur A2a |
| EP1903044A1 (fr) * | 2006-09-14 | 2008-03-26 | Novartis AG | Derivés de l'adénosine en tant qu' agonistes du récepteur A2A |
| CN101553459A (zh) * | 2006-11-10 | 2009-10-07 | 诺瓦提斯公司 | 环戊烯二醇单乙酸酯衍生物 |
| BRPI0818578A2 (pt) * | 2007-10-17 | 2015-07-21 | Novartis Ag | Derivados de purina como ligantes receptores de adenosina a1 |
| KR20140146217A (ko) | 2012-04-20 | 2014-12-24 | 유씨비 파마, 에스.에이. | 파킨슨병을 치료하는 방법 |
| MX2021008094A (es) | 2019-01-11 | 2021-09-21 | Omeros Corp | Metodos y composiciones para el tratamiento del cancer. |
| WO2026006723A1 (fr) * | 2024-06-27 | 2026-01-02 | Anand Rene | Réactifs et méthodes pour traiter les céphalées, dont les migraines, ainsi que leurs comorbidités |
| WO2026064126A1 (fr) | 2024-09-19 | 2026-03-26 | University Of Rochester | Utilisation d'inhibiteurs de gadd34 tels que sephin1 pour le traitement d'une maladie fibrotique des voies respiratoires |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GT200500281A (es) * | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
| GB0607950D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607953D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607945D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| PT2322525E (pt) * | 2006-04-21 | 2013-12-26 | Novartis Ag | Derivados de purina para utilização como agonistas do recetor de adenosina a2a |
-
2008
- 2008-10-08 US US12/247,764 patent/US20090181934A1/en not_active Abandoned
- 2008-10-15 PE PE2008001774A patent/PE20091392A1/es not_active Application Discontinuation
- 2008-10-15 WO PCT/EP2008/063869 patent/WO2009050198A2/fr not_active Ceased
- 2008-10-15 AU AU2008313788A patent/AU2008313788A1/en not_active Abandoned
- 2008-10-15 EP EP08838649A patent/EP2211865A2/fr not_active Withdrawn
- 2008-10-15 MX MX2010004252A patent/MX2010004252A/es not_active Application Discontinuation
- 2008-10-15 JP JP2010529369A patent/JP2011500630A/ja active Pending
- 2008-10-15 KR KR1020107008300A patent/KR20100075925A/ko not_active Withdrawn
- 2008-10-15 EA EA201000617A patent/EA201000617A1/ru unknown
- 2008-10-15 CA CA2702942A patent/CA2702942A1/fr not_active Abandoned
- 2008-10-15 AR ARP080104494A patent/AR068879A1/es not_active Application Discontinuation
- 2008-10-15 CN CN200880112188A patent/CN101827596A/zh active Pending
- 2008-10-15 BR BRPI0818005 patent/BRPI0818005A2/pt not_active IP Right Cessation
- 2008-10-16 TW TW097139728A patent/TW200927129A/zh unknown
- 2008-10-16 CL CL2008003057A patent/CL2008003057A1/es unknown
-
2010
- 2010-03-25 IL IL204723A patent/IL204723A0/en unknown
- 2010-03-26 CR CR11341A patent/CR11341A/es not_active Application Discontinuation
- 2010-04-01 ZA ZA2010/02336A patent/ZA201002336B/en unknown
- 2010-04-14 CU CU20100065A patent/CU20100065A7/es unknown
- 2010-04-16 TN TN2010000168A patent/TN2010000168A1/fr unknown
- 2010-04-30 MA MA32802A patent/MA31796B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2008313788A1 (en) | 2009-04-23 |
| JP2011500630A (ja) | 2011-01-06 |
| WO2009050198A2 (fr) | 2009-04-23 |
| IL204723A0 (en) | 2010-11-30 |
| KR20100075925A (ko) | 2010-07-05 |
| CL2008003057A1 (es) | 2009-06-26 |
| TW200927129A (en) | 2009-07-01 |
| AR068879A1 (es) | 2009-12-09 |
| ZA201002336B (en) | 2011-04-28 |
| BRPI0818005A2 (pt) | 2015-04-14 |
| EP2211865A2 (fr) | 2010-08-04 |
| US20090181934A1 (en) | 2009-07-16 |
| TN2010000168A1 (en) | 2011-11-11 |
| PE20091392A1 (es) | 2009-10-14 |
| EA201000617A1 (ru) | 2010-10-29 |
| CU20100065A7 (es) | 2011-10-05 |
| MX2010004252A (es) | 2010-04-30 |
| WO2009050198A3 (fr) | 2009-09-11 |
| CR11341A (es) | 2010-05-06 |
| CN101827596A (zh) | 2010-09-08 |
| CA2702942A1 (fr) | 2009-04-23 |
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