MA31796B1 - Composes organiques - Google Patents

Composes organiques

Info

Publication number
MA31796B1
MA31796B1 MA32802A MA32802A MA31796B1 MA 31796 B1 MA31796 B1 MA 31796B1 MA 32802 A MA32802 A MA 32802A MA 32802 A MA32802 A MA 32802A MA 31796 B1 MA31796 B1 MA 31796B1
Authority
MA
Morocco
Prior art keywords
antagonist
inhibitor
component
adrenoreceptor
beta
Prior art date
Application number
MA32802A
Other languages
Arabic (ar)
English (en)
Inventor
Robin Alec Fairhurst
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA31796B1 publication Critical patent/MA31796B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

L'invention concerne un médicament comprenant, séparément ou ensemble :, un composant (a) qui est un agoniste de récepteur d'adénosine a2a tel que défini dans la description; et un composant (b) qui est constitué d'un ou plusieurs composés choisis parmi : (i) un corticostéroïde, (ii) un agoniste d'adrénorécepteur bêta-2, (iii) un agent antimuscarinique, (iv) un antagoniste de a 2b, (v) un antihistaminique, (vi) un inhibiteur de caspase, (vii) un inhibiteur de enac, (viii) un antagoniste de ltb4, (ix) un antagoniste de ltd4, (x) un inhibiteur de sérine protéase, (xi) un inhibiteur de pde4 et (xii) un composé à double action agoniste d'adrénorécepteur bêta-2/antagoniste muscarinique, pour une administration simultanée, séquentielle ou séparée dans le traitement d'une maladie inflammatoire ou d'obstruction des voies aériennes.
MA32802A 2007-10-17 2010-04-30 Composes organiques MA31796B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07118721 2007-10-17
PCT/EP2008/063869 WO2009050198A2 (fr) 2007-10-17 2008-10-15 Composés organiques

Publications (1)

Publication Number Publication Date
MA31796B1 true MA31796B1 (fr) 2010-10-01

Family

ID=39185790

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32802A MA31796B1 (fr) 2007-10-17 2010-04-30 Composes organiques

Country Status (21)

Country Link
US (1) US20090181934A1 (fr)
EP (1) EP2211865A2 (fr)
JP (1) JP2011500630A (fr)
KR (1) KR20100075925A (fr)
CN (1) CN101827596A (fr)
AR (1) AR068879A1 (fr)
AU (1) AU2008313788A1 (fr)
BR (1) BRPI0818005A2 (fr)
CA (1) CA2702942A1 (fr)
CL (1) CL2008003057A1 (fr)
CR (1) CR11341A (fr)
CU (1) CU20100065A7 (fr)
EA (1) EA201000617A1 (fr)
IL (1) IL204723A0 (fr)
MA (1) MA31796B1 (fr)
MX (1) MX2010004252A (fr)
PE (1) PE20091392A1 (fr)
TN (1) TN2010000168A1 (fr)
TW (1) TW200927129A (fr)
WO (1) WO2009050198A2 (fr)
ZA (1) ZA201002336B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0500785D0 (en) 2005-01-14 2005-02-23 Novartis Ag Organic compounds
GB0607944D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
PE20080361A1 (es) 2006-04-21 2008-06-03 Novartis Ag Compuestos derivados de purina como activadores del receptor de adenosina a2a
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607948D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
EP1889846A1 (fr) 2006-07-13 2008-02-20 Novartis AG Dérivés de purine comme agonistes du recepteur A2a
EP1903044A1 (fr) * 2006-09-14 2008-03-26 Novartis AG Derivés de l'adénosine en tant qu' agonistes du récepteur A2A
WO2008055874A1 (fr) * 2006-11-10 2008-05-15 Novartis Ag Dérivés de monoacétate de cyclopentène diol
WO2009050199A1 (fr) * 2007-10-17 2009-04-23 Novartis Ag Dérivés de purine comme ligands des récepteurs a1 à l'adénosine
AU2013251079B2 (en) 2012-04-20 2017-03-23 Ucb Pharma S.A. Methods for treating Parkinson's disease
JOP20210164A1 (ar) 2019-01-11 2023-01-30 Omeros Corp طرق وتركيبات علاج السرطان
WO2026006723A1 (fr) * 2024-06-27 2026-01-02 Anand Rene Réactifs et méthodes pour traiter les céphalées, dont les migraines, ainsi que leurs comorbidités

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
PE20080361A1 (es) * 2006-04-21 2008-06-03 Novartis Ag Compuestos derivados de purina como activadores del receptor de adenosina a2a
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
PE20091392A1 (es) 2009-10-14
WO2009050198A2 (fr) 2009-04-23
JP2011500630A (ja) 2011-01-06
ZA201002336B (en) 2011-04-28
MX2010004252A (es) 2010-04-30
BRPI0818005A2 (pt) 2015-04-14
CU20100065A7 (es) 2011-10-05
AU2008313788A1 (en) 2009-04-23
EP2211865A2 (fr) 2010-08-04
EA201000617A1 (ru) 2010-10-29
US20090181934A1 (en) 2009-07-16
AR068879A1 (es) 2009-12-09
CL2008003057A1 (es) 2009-06-26
KR20100075925A (ko) 2010-07-05
TW200927129A (en) 2009-07-01
CR11341A (es) 2010-05-06
IL204723A0 (en) 2010-11-30
CN101827596A (zh) 2010-09-08
WO2009050198A3 (fr) 2009-09-11
TN2010000168A1 (en) 2011-11-11
CA2702942A1 (fr) 2009-04-23

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