MA31796B1 - Composes organiques - Google Patents

Composes organiques

Info

Publication number
MA31796B1
MA31796B1 MA32802A MA32802A MA31796B1 MA 31796 B1 MA31796 B1 MA 31796B1 MA 32802 A MA32802 A MA 32802A MA 32802 A MA32802 A MA 32802A MA 31796 B1 MA31796 B1 MA 31796B1
Authority
MA
Morocco
Prior art keywords
antagonist
inhibitor
component
adrenoreceptor
beta
Prior art date
Application number
MA32802A
Other languages
Arabic (ar)
English (en)
Inventor
Robin Alec Fairhurst
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA31796B1 publication Critical patent/MA31796B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

L'invention concerne un médicament comprenant, séparément ou ensemble :, un composant (a) qui est un agoniste de récepteur d'adénosine a2a tel que défini dans la description; et un composant (b) qui est constitué d'un ou plusieurs composés choisis parmi : (i) un corticostéroïde, (ii) un agoniste d'adrénorécepteur bêta-2, (iii) un agent antimuscarinique, (iv) un antagoniste de a 2b, (v) un antihistaminique, (vi) un inhibiteur de caspase, (vii) un inhibiteur de enac, (viii) un antagoniste de ltb4, (ix) un antagoniste de ltd4, (x) un inhibiteur de sérine protéase, (xi) un inhibiteur de pde4 et (xii) un composé à double action agoniste d'adrénorécepteur bêta-2/antagoniste muscarinique, pour une administration simultanée, séquentielle ou séparée dans le traitement d'une maladie inflammatoire ou d'obstruction des voies aériennes.
MA32802A 2007-10-17 2010-04-30 Composes organiques MA31796B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07118721 2007-10-17
PCT/EP2008/063869 WO2009050198A2 (fr) 2007-10-17 2008-10-15 Composés organiques

Publications (1)

Publication Number Publication Date
MA31796B1 true MA31796B1 (fr) 2010-10-01

Family

ID=39185790

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32802A MA31796B1 (fr) 2007-10-17 2010-04-30 Composes organiques

Country Status (21)

Country Link
US (1) US20090181934A1 (fr)
EP (1) EP2211865A2 (fr)
JP (1) JP2011500630A (fr)
KR (1) KR20100075925A (fr)
CN (1) CN101827596A (fr)
AR (1) AR068879A1 (fr)
AU (1) AU2008313788A1 (fr)
BR (1) BRPI0818005A2 (fr)
CA (1) CA2702942A1 (fr)
CL (1) CL2008003057A1 (fr)
CR (1) CR11341A (fr)
CU (1) CU20100065A7 (fr)
EA (1) EA201000617A1 (fr)
IL (1) IL204723A0 (fr)
MA (1) MA31796B1 (fr)
MX (1) MX2010004252A (fr)
PE (1) PE20091392A1 (fr)
TN (1) TN2010000168A1 (fr)
TW (1) TW200927129A (fr)
WO (1) WO2009050198A2 (fr)
ZA (1) ZA201002336B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0500785D0 (en) 2005-01-14 2005-02-23 Novartis Ag Organic compounds
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607944D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
HRP20120494T1 (hr) 2006-04-21 2012-08-31 Novartis Ag Derivati purina za uporabu kao agonista adenozin a2a receptora
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607948D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
EP1889846A1 (fr) 2006-07-13 2008-02-20 Novartis AG Dérivés de purine comme agonistes du recepteur A2a
EP1903044A1 (fr) * 2006-09-14 2008-03-26 Novartis AG Derivés de l'adénosine en tant qu' agonistes du récepteur A2A
JP2010508835A (ja) * 2006-11-10 2010-03-25 ノバルティス アーゲー シクロペンテンジオールモノアセテート誘導体
KR20100068286A (ko) * 2007-10-17 2010-06-22 노파르티스 아게 아데노신 ａ1 수용체 리간드로서의 퓨린 유도체
AU2013251079B2 (en) 2012-04-20 2017-03-23 Ucb Pharma S.A. Methods for treating Parkinson's disease
WO2020146795A1 (fr) 2019-01-11 2020-07-16 Omeros Corporation Procédés et compositions pour le traitement du cancer
WO2026006723A1 (fr) * 2024-06-27 2026-01-02 Anand Rene Réactifs et méthodes pour traiter les céphalées, dont les migraines, ainsi que leurs comorbidités
WO2026064126A1 (fr) 2024-09-19 2026-03-26 University Of Rochester Utilisation d'inhibiteurs de gadd34 tels que sephin1 pour le traitement d'une maladie fibrotique des voies respiratoires

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
HRP20120494T1 (hr) * 2006-04-21 2012-08-31 Novartis Ag Derivati purina za uporabu kao agonista adenozin a2a receptora
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
WO2009050198A2 (fr) 2009-04-23
JP2011500630A (ja) 2011-01-06
CA2702942A1 (fr) 2009-04-23
EP2211865A2 (fr) 2010-08-04
AR068879A1 (es) 2009-12-09
MX2010004252A (es) 2010-04-30
WO2009050198A3 (fr) 2009-09-11
CN101827596A (zh) 2010-09-08
CU20100065A7 (es) 2011-10-05
BRPI0818005A2 (pt) 2015-04-14
CR11341A (es) 2010-05-06
CL2008003057A1 (es) 2009-06-26
AU2008313788A1 (en) 2009-04-23
US20090181934A1 (en) 2009-07-16
PE20091392A1 (es) 2009-10-14
TN2010000168A1 (en) 2011-11-11
EA201000617A1 (ru) 2010-10-29
IL204723A0 (en) 2010-11-30
TW200927129A (en) 2009-07-01
ZA201002336B (en) 2011-04-28
KR20100075925A (ko) 2010-07-05

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