MA31902B1 - Oxazolidinones pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque - Google Patents

Oxazolidinones pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque

Info

Publication number
MA31902B1
MA31902B1 MA32895A MA32895A MA31902B1 MA 31902 B1 MA31902 B1 MA 31902B1 MA 32895 A MA32895 A MA 32895A MA 32895 A MA32895 A MA 32895A MA 31902 B1 MA31902 B1 MA 31902B1
Authority
MA
Morocco
Prior art keywords
heart failure
prophylaxis
treatment
oxazolidinones
disorders associated
Prior art date
Application number
MA32895A
Other languages
Arabic (ar)
English (en)
Inventor
Harald Kallabis
Wolfgang Thielemann
Elisabeth Perzborn
Susanne Röhrig
Dagmar Kubitza
Theodore Spiro
Lloyd Haskell
Jeet Mahal
Original Assignee
Bayer Schering Pharma Ag
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag, Janssen Pharmaceutica Nv filed Critical Bayer Schering Pharma Ag
Publication of MA31902B1 publication Critical patent/MA31902B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La présente invention concerne l'utilisation d'inhibiteurs sélectifs du facteur xa de coagulation, notamment des oxazolidinones de formule (i), pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque et/ou de troubles associés à l'insuffisance cardiaque ainsi que leur utilisation pour la préparation de médicaments pharmaceutiques pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque et/ou de troubles associés à l'insuffisance cardiaque.
MA32895A 2007-12-11 2010-06-08 Oxazolidinones pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque MA31902B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US740607P 2007-12-11 2007-12-11
PCT/EP2008/010211 WO2009074249A1 (fr) 2007-12-11 2008-12-03 Oxazolidinones pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque

Publications (1)

Publication Number Publication Date
MA31902B1 true MA31902B1 (fr) 2010-12-01

Family

ID=40404481

Family Applications (1)

Application Number Title Priority Date Filing Date
MA32895A MA31902B1 (fr) 2007-12-11 2010-06-08 Oxazolidinones pour le traitement et/ou la prophylaxie de l'insuffisance cardiaque

Country Status (18)

Country Link
US (1) US20110003804A1 (fr)
EP (1) EP2229173A1 (fr)
JP (1) JP2011506363A (fr)
KR (1) KR20110010689A (fr)
CN (1) CN101896185A (fr)
AU (1) AU2008335922A1 (fr)
BR (1) BRPI0820964A2 (fr)
CA (1) CA2708418C (fr)
DO (1) DOP2010000156A (fr)
IL (1) IL205675A (fr)
MA (1) MA31902B1 (fr)
MX (1) MX2010005545A (fr)
NZ (1) NZ586002A (fr)
RU (2) RU2494740C2 (fr)
SV (1) SV2010003578A (fr)
TN (1) TN2010000266A1 (fr)
UA (1) UA99638C2 (fr)
WO (1) WO2009074249A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2905760T3 (es) * 2009-07-31 2022-04-12 Krka D D Novo Mesto Procedimientos para la cristalización del rivaroxabán
CN103626749A (zh) * 2012-08-21 2014-03-12 苏州泽璟生物制药有限公司 取代的噁唑烷酮化合物和包含该化合物的药物组合物及其用途
JP2020524283A (ja) * 2017-06-20 2020-08-13 アンスティチュ ナショナル ドゥ ラ サンテ エ ドゥ ラ ルシェルシュ メディカル 急性非代償性心不全(adhf)患者が凝固亢進状態を示すかどうかを同定するための方法
KR102715821B1 (ko) * 2017-11-09 2024-10-10 고쿠리츠 다이가쿠호우징 도쿄이카시카다이가쿠 암 촉진 인자 발현 억제제, 그 유효 성분의 스크리닝 방법, 그 방법에 유용한 발현 카세트, 진단약, 및 진단 방법
JP6574041B2 (ja) * 2017-12-15 2019-09-11 エルメッド株式会社 リバーロキサバン含有医薬組成物
PE20211267A1 (es) 2019-08-30 2021-07-19 Astrazeneca Ab Metodos de tratamiento de la insuficiencia cardiaca con fraccion de eyeccion reducida con dapagliflozina

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0610265B1 (fr) * 1991-11-01 1996-12-27 PHARMACIA & UPJOHN COMPANY Aryl- et heteroarylphenyloxazolidinones substituees, utilisees comme agents antibacteriens
DK0623615T3 (da) * 1993-05-01 1999-12-13 Merck Patent Gmbh Adhæsionsreceptor-antagonister
DE19962924A1 (de) * 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
DE10129725A1 (de) * 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
TW200812619A (en) * 2006-04-06 2008-03-16 Schering Corp TRA combination therapies

Also Published As

Publication number Publication date
KR20110010689A (ko) 2011-02-07
CN101896185A (zh) 2010-11-24
IL205675A (en) 2013-10-31
AU2008335922A1 (en) 2009-06-18
CA2708418A1 (fr) 2009-06-18
DOP2010000156A (es) 2011-02-15
UA99638C2 (ru) 2012-09-10
TN2010000266A1 (en) 2011-11-11
JP2011506363A (ja) 2011-03-03
RU2010128442A (ru) 2012-01-20
CA2708418C (fr) 2013-11-12
IL205675A0 (en) 2010-11-30
EP2229173A1 (fr) 2010-09-22
RU2494740C2 (ru) 2013-10-10
MX2010005545A (es) 2010-07-30
NZ586002A (en) 2012-06-29
RU2013134140A (ru) 2015-01-27
WO2009074249A1 (fr) 2009-06-18
SV2010003578A (es) 2011-02-21
US20110003804A1 (en) 2011-01-06
BRPI0820964A2 (pt) 2015-07-14

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