MA33806B1 - Inhibiteurs du virus de l'hepatite c - Google Patents

Inhibiteurs du virus de l'hepatite c

Info

Publication number
MA33806B1
MA33806B1 MA34944A MA34944A MA33806B1 MA 33806 B1 MA33806 B1 MA 33806B1 MA 34944 A MA34944 A MA 34944A MA 34944 A MA34944 A MA 34944A MA 33806 B1 MA33806 B1 MA 33806B1
Authority
MA
Morocco
Prior art keywords
hepatitis
inhibitors
compounds
treatment
methods
Prior art date
Application number
MA34944A
Other languages
Arabic (ar)
English (en)
Inventor
Makonen Belema
Jeffrey Lee Romine
Van N Nguyen
Gan Wang
Omar D Lopez
Laurent Denis R St
Qi Chen
John A Bender
Zhong Yang
Piyasena Hewawasam
Ningning Xu
Nicholas A Meanwell
John A Easter
bao-ning Su
Michael J Smith
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43479603&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA33806(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of MA33806B1 publication Critical patent/MA33806B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19—Cytokines; Lymphokines; Interferons
    • A61K38/21—Interferons [IFN]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La présente invention porte sur des composés, des compositions et des procédés pour le traitement d'une infection par le virus de l'hépatite c (vhc). L'invention porte également sur des compositions pharmaceutiques contenant de tels composés et sur des procédés d'utilisation de ces composés dans le traitement d'une infection par le vhc.
MA34944A 2009-12-16 2012-06-06 Inhibiteurs du virus de l'hepatite c MA33806B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28694209P 2009-12-16 2009-12-16
US12/957,512 US8377980B2 (en) 2009-12-16 2010-12-01 Hepatitis C virus inhibitors
PCT/US2010/060077 WO2011075439A1 (fr) 2009-12-16 2010-12-13 Inhibiteurs du virus de l'hépatite c

Publications (1)

Publication Number Publication Date
MA33806B1 true MA33806B1 (fr) 2012-12-03

Family

ID=43479603

Family Applications (1)

Application Number Title Priority Date Filing Date
MA34944A MA33806B1 (fr) 2009-12-16 2012-06-06 Inhibiteurs du virus de l'hepatite c

Country Status (21)

Country Link
US (1) US8377980B2 (fr)
EP (1) EP2513091B1 (fr)
JP (1) JP5785189B2 (fr)
KR (1) KR20120107991A (fr)
CN (1) CN102741242B (fr)
AR (1) AR079634A1 (fr)
AU (1) AU2010332034B2 (fr)
BR (1) BR112012014677A2 (fr)
CA (1) CA2784662A1 (fr)
CL (1) CL2012001637A1 (fr)
CO (1) CO6561788A2 (fr)
EA (1) EA020815B1 (fr)
MA (1) MA33806B1 (fr)
MX (1) MX2012006635A (fr)
NZ (1) NZ601220A (fr)
PE (1) PE20121479A1 (fr)
PH (1) PH12012500979A1 (fr)
SG (1) SG181700A1 (fr)
TN (1) TN2012000264A1 (fr)
TW (1) TWI487702B (fr)
WO (1) WO2011075439A1 (fr)

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US20190127365A1 (en) 2017-11-01 2019-05-02 Merck Sharp & Dohme Corp. Inhibitors of hepatitis c virus replication
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EP2513091B1 (fr) 2017-04-12
TN2012000264A1 (en) 2013-12-12
CA2784662A1 (fr) 2011-06-23
KR20120107991A (ko) 2012-10-04
EP2513091A1 (fr) 2012-10-24
MX2012006635A (es) 2012-06-21
US8377980B2 (en) 2013-02-19
JP2013514359A (ja) 2013-04-25
WO2011075439A1 (fr) 2011-06-23
AU2010332034A1 (en) 2012-08-02
NZ601220A (en) 2014-07-25
AU2010332034B2 (en) 2016-04-14
PH12012500979A1 (en) 2014-09-05
BR112012014677A2 (pt) 2015-09-15
TW201130825A (en) 2011-09-16
CO6561788A2 (es) 2012-11-15
TWI487702B (zh) 2015-06-11
CL2012001637A1 (es) 2012-10-12
US20110286961A1 (en) 2011-11-24
EA020815B1 (ru) 2015-01-30
CN102741242A (zh) 2012-10-17
PE20121479A1 (es) 2012-11-07
EA201270656A1 (ru) 2012-11-30
JP5785189B2 (ja) 2015-09-24
CN102741242B (zh) 2015-07-01
SG181700A1 (en) 2012-07-30

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