MA37379A1 - Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one - Google Patents

Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one

Info

Publication number
MA37379A1
MA37379A1 MA37379A MA37379A MA37379A1 MA 37379 A1 MA37379 A1 MA 37379A1 MA 37379 A MA37379 A MA 37379A MA 37379 A MA37379 A MA 37379A MA 37379 A1 MA37379 A1 MA 37379A1
Authority
MA
Morocco
Prior art keywords
phenylquinazolin
purin
ylamino
fluoro
propyl
Prior art date
Application number
MA37379A
Other languages
English (en)
Inventor
Ernest Carra
Michael Gerber
Bing Shi
Keiko Sujino
Duong Tran
Fang Wang
Jerry B Evarts
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA37379(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of MA37379A1 publication Critical patent/MA37379A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

Cette invention concerne des polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one, des compositions de ceux-ci, des procédés pour leur préparation et pour leur utilisation.
MA37379A 2012-03-05 2014-09-26 Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one MA37379A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05
PCT/US2013/029157 WO2013134288A1 (fr) 2012-03-05 2013-03-05 Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one

Publications (1)

Publication Number Publication Date
MA37379A1 true MA37379A1 (fr) 2016-11-30

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
MA37379A MA37379A1 (fr) 2012-03-05 2014-09-26 Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one

Country Status (31)

Country Link
US (3) US8865730B2 (fr)
EP (1) EP2834241B1 (fr)
JP (2) JP2015509537A (fr)
KR (1) KR20140133590A (fr)
CN (2) CN106146506A (fr)
AP (1) AP2014007875A0 (fr)
AR (1) AR090253A1 (fr)
AU (1) AU2013203620B2 (fr)
BR (1) BR112014021935A2 (fr)
CA (1) CA2864305C (fr)
CL (1) CL2014002358A1 (fr)
CO (1) CO7071131A2 (fr)
CR (1) CR20140460A (fr)
EA (3) EA201690461A1 (fr)
EC (1) ECSP14020478A (fr)
ES (1) ES2848273T3 (fr)
IN (1) IN2014DN07105A (fr)
MA (1) MA37379A1 (fr)
MD (1) MD20140100A2 (fr)
MX (1) MX2014010656A (fr)
NZ (1) NZ629684A (fr)
PE (1) PE20141792A1 (fr)
PH (1) PH12014501920A1 (fr)
PL (1) PL2834241T3 (fr)
PT (1) PT2834241T (fr)
SG (1) SG11201405446PA (fr)
SI (1) SI2834241T1 (fr)
TW (1) TW201350486A (fr)
UY (1) UY34656A (fr)
WO (1) WO2013134288A1 (fr)
ZA (1) ZA201405870B (fr)

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