MA37438A1 - Procédés de traitement du cancer utilisant des inhibiteurs de la kinase aurora - Google Patents
Procédés de traitement du cancer utilisant des inhibiteurs de la kinase auroraInfo
- Publication number
- MA37438A1 MA37438A1 MA37438A MA37438A MA37438A1 MA 37438 A1 MA37438 A1 MA 37438A1 MA 37438 A MA37438 A MA 37438A MA 37438 A MA37438 A MA 37438A MA 37438 A1 MA37438 A1 MA 37438A1
- Authority
- MA
- Morocco
- Prior art keywords
- kinase inhibitors
- cancer treatment
- treatment methods
- aurora kinase
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention concerne des procédés pour le traitement de divers troubles prolifératifs cellulaires. L'invention concerne en particulier des procédés pour le traitement de divers troubles prolifératifs cellulaires par administration d'un inhibiteur sélectif de la kinase aurora a en combinaison avec une chimiothérapie à base de taxane, tel que le paclitaxel ou le docétaxel.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261613258P | 2012-03-20 | 2012-03-20 | |
| PCT/US2013/032962 WO2013142491A1 (fr) | 2012-03-20 | 2013-03-19 | Procédés de traitement du cancer utilisant des inhibiteurs de la kinase aurora |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA37438A1 true MA37438A1 (fr) | 2016-05-31 |
Family
ID=48048255
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA37438A MA37438A1 (fr) | 2012-03-20 | 2013-03-19 | Procédés de traitement du cancer utilisant des inhibiteurs de la kinase aurora |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US20130303519A1 (fr) |
| EP (1) | EP2827855B1 (fr) |
| JP (1) | JP6373252B2 (fr) |
| KR (1) | KR102128866B1 (fr) |
| CN (1) | CN104271129A (fr) |
| AU (1) | AU2013235275B2 (fr) |
| CA (1) | CA2868024A1 (fr) |
| EA (1) | EA036434B1 (fr) |
| ES (1) | ES2746946T3 (fr) |
| GE (2) | GEAP201813599A (fr) |
| IL (1) | IL234686B (fr) |
| IN (1) | IN2014DN08477A (fr) |
| JO (1) | JO3630B1 (fr) |
| MA (1) | MA37438A1 (fr) |
| MX (1) | MX358411B (fr) |
| MY (1) | MY175225A (fr) |
| NZ (1) | NZ700744A (fr) |
| PH (1) | PH12014502109A1 (fr) |
| SG (2) | SG10201607741RA (fr) |
| TN (1) | TN2014000387A1 (fr) |
| TW (1) | TWI649082B (fr) |
| UA (1) | UA117455C2 (fr) |
| WO (1) | WO2013142491A1 (fr) |
| ZA (1) | ZA201407551B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130303519A1 (en) | 2012-03-20 | 2013-11-14 | Millennium Pharmaceuticals, Inc. | Methods of treating cancer using aurora kinase inhibitors |
| EP3236948A4 (fr) * | 2014-12-23 | 2018-10-03 | Millennium Pharmaceuticals, Inc. | Combinaison d'inhibiteurs de raf et d'inhibiteurs de kinases aurora |
| EP3317427B1 (fr) * | 2015-07-02 | 2020-12-23 | Millennium Pharmaceuticals, Inc. | Biomarqueurs de réponse à des inhibiteurs sélectifs d'aurora a kinase |
| CN110833544B (zh) * | 2018-08-17 | 2022-08-09 | 深圳微芯生物科技股份有限公司 | 组蛋白去乙酰化酶抑制剂与蛋白激酶抑制剂之组合及其制药用途 |
Family Cites Families (42)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4099012A (en) | 1975-08-28 | 1978-07-04 | Ciba-Geigy Corporation | 2-pyrazolyl-benzophenones |
| FR2450833A1 (fr) | 1979-02-07 | 1980-10-03 | Hoffmann La Roche | Derives de benzazepine |
| US4481142A (en) | 1979-02-07 | 1984-11-06 | Hoffmann-La Roche Inc. | Pyrimido-2-benzazepines |
| US4469633A (en) | 1980-05-16 | 1984-09-04 | Hoffmann-La Roche Inc. | N-oxides of 5-oxo-1-phenyl-2-benzazepines |
| EP0273697A3 (fr) | 1986-12-30 | 1989-11-29 | Merck & Co. Inc. | 2-Benzazépines à cycles hétérocycliques de 5 et 6 côtés |
| US5166151A (en) | 1988-03-25 | 1992-11-24 | Merck & Co., Inc. | 2-Benzazepines with 5- and 6-membered heterocyclic rings, compositions and medical methods of use thereof |
| US5210082A (en) | 1991-05-16 | 1993-05-11 | Merck & Co., Inc. | 2-benzazepines with 5- and 6-membered heterocyclic rings to treat pain and anxiety disorders |
| US6096331A (en) | 1993-02-22 | 2000-08-01 | Vivorx Pharmaceuticals, Inc. | Methods and compositions useful for administration of chemotherapeutic agents |
| US5747487A (en) | 1993-07-29 | 1998-05-05 | American Cyanamid Company | Tricyclic benzazepine vasopressin antagonists |
| GB9523675D0 (en) | 1995-11-20 | 1996-01-24 | Celltech Therapeutics Ltd | Chemical compounds |
| CA2247453A1 (fr) | 1996-03-08 | 1997-09-12 | Joseph James Lewis | Principes actifs neurologiques derives d'azolobenzazepine |
| US6057329A (en) | 1996-12-23 | 2000-05-02 | Celltech Therapeutics Limited | Fused polycyclic 2-aminopyrimidine derivatives |
| GB9713087D0 (en) | 1997-06-20 | 1997-08-27 | Celltech Therapeutics Ltd | Chemical compounds |
| NZ503601A (en) | 1997-09-29 | 2002-02-01 | Meiji Seika Kaisha | Tricyclic triazolobenzazepine derivatives for use as antiallergic medicaments |
| US6277844B1 (en) | 1998-09-14 | 2001-08-21 | Sydney Spector | Compound for selective treatment of malignant cells by inhibiting cell cycle progression, decreasing Bcl2, and increasing apoptosis |
| WO2000067754A1 (fr) | 1999-05-12 | 2000-11-16 | Nitromed, Inc. | Activateurs nitroses et nitrosyles du canal potassique, compositions et utilisations |
| AP2003002762A0 (en) | 2000-09-15 | 2003-03-31 | Vertex Pharma | Pyrazole compounds useful as protein kinase inhibitors |
| AU2002255452B2 (en) | 2000-12-21 | 2006-06-08 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
| SI20848A (sl) | 2001-03-14 | 2002-10-31 | Lek, Tovarna Farmacevtskih In Kemijskih Izdelkov, D.D. | Farmacevtska formulacija, ki vsebuje atorvastatin kalcij |
| US6686352B2 (en) | 2001-05-18 | 2004-02-03 | Hoffmann-La Roche Inc. | Substituted imidazo [1,5-a] pyrimido [5,4-d] [1] benzazepine derivatives |
| DE10135457A1 (de) | 2001-07-20 | 2003-02-06 | Adc Automotive Dist Control | Optische Sensoranordnung |
| IL159963A0 (en) | 2001-08-09 | 2004-06-20 | Actelion Pharmaceuticals Ltd | Novel benzo-fused heterocycles as endothelin antagonisits |
| CN1897950A (zh) | 2003-10-14 | 2007-01-17 | 惠氏公司 | 稠合芳基和杂芳基衍生物及其使用方法 |
| CA2554271A1 (fr) | 2004-02-10 | 2005-08-25 | Santarus, Inc. | Combinaison d'un inhibiteur de la pompe a protons, d'un tampon et d'un medicament anti-inflammatoire non steroidien |
| EP2261226B1 (fr) | 2004-05-14 | 2015-04-01 | Millennium Pharmaceuticals, Inc. | Procédés pour la préparation d'inhibiteurs de l'aurora kinase |
| WO2006055831A2 (fr) | 2004-11-17 | 2006-05-26 | Miikana Therapeutics, Inc. | Inhibiteurs de kinase |
| EP1836188A1 (fr) | 2004-12-30 | 2007-09-26 | Astex Therapeutics Limited | Derives pyrazoliques modulant l'activite des kinases cdk, gsk et aurora |
| CN101389324A (zh) | 2005-12-23 | 2009-03-18 | 史密丝克莱恩比彻姆公司 | Aurora激酶的氮杂吲哚抑制剂 |
| WO2007080601A1 (fr) | 2006-01-16 | 2007-07-19 | Jubilant Organosys Limited | Formulation pharmaceutique stable d'un compose labile a base d'acide et son procede de preparation |
| AR059838A1 (es) | 2006-03-14 | 2008-04-30 | Ranbaxy Lab Ltd | Formulaciones para dosis estabilizantes de estatina |
| DE102006012301A1 (de) | 2006-03-15 | 2007-09-20 | Cemag-Anlagenbau-Dessau Gmbh | Herstellung von Zementklinker |
| US7718648B2 (en) | 2006-08-09 | 2010-05-18 | Millennium Pharmaceuticals, Inc. | Pyridobenzazepine compounds and methods for inhibiting mitotic progression |
| CN101528237A (zh) | 2006-10-31 | 2009-09-09 | 艾其林医药公司 | 艾夫他滨药物组合物 |
| CL2007003244A1 (es) | 2006-11-16 | 2008-04-04 | Millennium Pharm Inc | Compuestos derivados de pirimido[5,4-d][2]benzazepina; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento del cancer. |
| PE20081891A1 (es) | 2007-03-22 | 2008-12-27 | Opko Health Inc | Formulaciones de comprimidos que contienen sales de 8-[{1-(3,5-bis-(trifluorometil)fenil)-etoxi}-metil]-8-fenil-1,7-diaza-spiro[4.5]decan-2-ona y comprimidos elaborados a partir de estas |
| US20090203671A1 (en) | 2007-11-27 | 2009-08-13 | Abbott Laboratories | Method of treating cancer |
| US20110033461A1 (en) * | 2008-03-12 | 2011-02-10 | Vladimir Ratushny | Combination Therapy for the Treatment of Cancer |
| KR101848095B1 (ko) | 2008-06-26 | 2018-04-11 | 안테리오스, 인코퍼레이티드 | 경피 운반 |
| JO3635B1 (ar) | 2009-05-18 | 2020-08-27 | Millennium Pharm Inc | مركبات صيدلانية صلبة وطرق لانتاجها |
| JO3434B1 (ar) | 2009-07-31 | 2019-10-20 | Millennium Pharm Inc | مركبات صيدلانية لمعالجة السرطان وامراض واضطرابات اخري |
| BR112012020557A8 (pt) | 2010-02-19 | 2018-01-02 | Millennium Pharm Inc | formas cristalinas de 4-{[9-cloro-7-(2-flúor-6-metoifenil)-5h-pirimido[5,4-d][2]benzazepin-2-il]amino}-2-metoxibenzoato de sódio |
| US20130303519A1 (en) | 2012-03-20 | 2013-11-14 | Millennium Pharmaceuticals, Inc. | Methods of treating cancer using aurora kinase inhibitors |
-
2013
- 2013-03-14 US US13/804,570 patent/US20130303519A1/en not_active Abandoned
- 2013-03-18 JO JOP/2013/0075A patent/JO3630B1/ar active
- 2013-03-19 KR KR1020147028776A patent/KR102128866B1/ko active Active
- 2013-03-19 AU AU2013235275A patent/AU2013235275B2/en active Active
- 2013-03-19 JP JP2015501852A patent/JP6373252B2/ja active Active
- 2013-03-19 SG SG10201607741RA patent/SG10201607741RA/en unknown
- 2013-03-19 UA UAA201411324A patent/UA117455C2/uk unknown
- 2013-03-19 MA MA37438A patent/MA37438A1/fr unknown
- 2013-03-19 CA CA2868024A patent/CA2868024A1/fr not_active Abandoned
- 2013-03-19 EP EP13714455.6A patent/EP2827855B1/fr active Active
- 2013-03-19 MY MYPI2014702635A patent/MY175225A/en unknown
- 2013-03-19 ES ES13714455T patent/ES2746946T3/es active Active
- 2013-03-19 EA EA201491727A patent/EA036434B1/ru not_active IP Right Cessation
- 2013-03-19 GE GEAP201813599A patent/GEAP201813599A/en unknown
- 2013-03-19 GE GEAP201313599A patent/GEP20186900B/en unknown
- 2013-03-19 NZ NZ700744A patent/NZ700744A/en not_active IP Right Cessation
- 2013-03-19 WO PCT/US2013/032962 patent/WO2013142491A1/fr not_active Ceased
- 2013-03-19 SG SG11201405621UA patent/SG11201405621UA/en unknown
- 2013-03-19 CN CN201380015806.1A patent/CN104271129A/zh active Pending
- 2013-03-19 IN IN8477DEN2014 patent/IN2014DN08477A/en unknown
- 2013-03-19 MX MX2014011324A patent/MX358411B/es active IP Right Grant
- 2013-03-20 TW TW102109912A patent/TWI649082B/zh active
-
2014
- 2014-09-15 TN TNP2014000387A patent/TN2014000387A1/fr unknown
- 2014-09-16 IL IL234686A patent/IL234686B/en active IP Right Grant
- 2014-09-22 PH PH12014502109A patent/PH12014502109A1/en unknown
- 2014-10-17 ZA ZA2014/07551A patent/ZA201407551B/en unknown
-
2015
- 2015-09-03 US US14/844,270 patent/US10213436B2/en active Active
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