MA42242A - Inhibiteurs de la tyrosine kinase - Google Patents

Inhibiteurs de la tyrosine kinase

Info

Publication number
MA42242A
MA42242A MA042242A MA42242A MA42242A MA 42242 A MA42242 A MA 42242A MA 042242 A MA042242 A MA 042242A MA 42242 A MA42242 A MA 42242A MA 42242 A MA42242 A MA 42242A
Authority
MA
Morocco
Prior art keywords
tyrosine kinase
kinase inhibitors
inhibitors
tyrosine
kinase
Prior art date
Application number
MA042242A
Other languages
English (en)
Inventor
David Goldstein
Timothy D Owens
Original Assignee
Principia Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Principia Biopharma Inc filed Critical Principia Biopharma Inc
Publication of MA42242A publication Critical patent/MA42242A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA042242A 2015-06-24 2016-06-23 Inhibiteurs de la tyrosine kinase MA42242A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562183969P 2015-06-24 2015-06-24
US201562271715P 2015-12-28 2015-12-28

Publications (1)

Publication Number Publication Date
MA42242A true MA42242A (fr) 2018-05-02

Family

ID=56292979

Family Applications (1)

Application Number Title Priority Date Filing Date
MA042242A MA42242A (fr) 2015-06-24 2016-06-23 Inhibiteurs de la tyrosine kinase

Country Status (5)

Country Link
US (2) US20180305350A1 (fr)
EP (1) EP3313839A1 (fr)
MA (1) MA42242A (fr)
TW (1) TW201718572A (fr)
WO (1) WO2016210165A1 (fr)

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JP7891740B2 (ja) * 2020-03-30 2026-07-17 イエール ユニバーシティ チロシンキナーゼ阻害剤の小児用製剤
CN113527300B (zh) * 2020-06-04 2023-02-03 广州百霆医药科技有限公司 布鲁顿酪氨酸蛋白激酶抑制剂
CN116018345A (zh) * 2020-07-16 2023-04-25 株式会社棱镜生物实验室 新的杂环化合物
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CN115073468B (zh) * 2021-03-15 2023-12-22 药雅科技(上海)有限公司 咪唑并吡嗪类btk抑制剂的制备及用途
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US20190345159A1 (en) 2019-11-14
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US20180305350A1 (en) 2018-10-25
WO2016210165A1 (fr) 2016-12-29
US11155544B2 (en) 2021-10-26

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