MA42913A - Pyridazinones et leur utilisation dans le traitement du cancer - Google Patents
Pyridazinones et leur utilisation dans le traitement du cancerInfo
- Publication number
- MA42913A MA42913A MA042913A MA42913A MA42913A MA 42913 A MA42913 A MA 42913A MA 042913 A MA042913 A MA 042913A MA 42913 A MA42913 A MA 42913A MA 42913 A MA42913 A MA 42913A
- Authority
- MA
- Morocco
- Prior art keywords
- pyridazinones
- cancer
- treatment
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 title 1
- 201000011510 cancer Diseases 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1514015.5A GB201514015D0 (en) | 2015-08-07 | 2015-08-07 | Novel pyridazinones and their use in the treatment of cancer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA42913A true MA42913A (fr) | 2018-08-01 |
Family
ID=54200420
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA042913A MA42913A (fr) | 2015-08-07 | 2016-08-05 | Pyridazinones et leur utilisation dans le traitement du cancer |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US11110089B2 (fr) |
| EP (1) | EP3331878A1 (fr) |
| GB (1) | GB201514015D0 (fr) |
| MA (1) | MA42913A (fr) |
| WO (1) | WO2017027357A1 (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG11202007535VA (en) * | 2018-02-12 | 2020-09-29 | Cinda Pharma Ab | Thioredoxin reductase inhibitors for use in the treatment of cancer |
| CN112996795B (zh) | 2018-09-18 | 2024-11-12 | 尼坎治疗公司 | 作为src同源-2磷酸酶抑制剂的稠合的三环衍生物 |
| EP4076448A4 (fr) | 2019-12-20 | 2024-03-27 | Tenaya Therapeutics, Inc. | Oxadiazoles fluoroalkylés et leurs utilisations |
| EP4333841A1 (fr) | 2021-05-04 | 2024-03-13 | Tenaya Therapeutics, Inc. | 2-fluoroalkyl-1,3,4-oxadiazol-5-yl-thiazol, inhibiteurs de hdac6 pour utilisation dans le traitement des maladies métaboliques et de l'icfep |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4939140A (en) | 1985-11-07 | 1990-07-03 | Pfizer Inc. | Heterocyclic oxophthalazinyl acetic acids |
| JP5423679B2 (ja) * | 2007-10-31 | 2014-02-19 | 日産化学工業株式会社 | ピリダジノン化合物及びp2x7受容体阻害剤 |
| DE102007061963A1 (de) * | 2007-12-21 | 2009-06-25 | Merck Patent Gmbh | Pyridazinonderivate |
| AU2012382373A1 (en) | 2012-06-12 | 2014-12-11 | Abbvie Inc. | Pyridinone and pyridazinone derivatives |
| CN103864769B (zh) * | 2012-12-14 | 2016-11-02 | 上海工程技术大学 | 一种噁二唑化合物及其制备方法 |
| KR20170092634A (ko) | 2014-12-05 | 2017-08-11 | 에이엔2에이치 디스커버리 리미티드 | 파킨 리가제 활성화 방법 및 조성물 |
-
2015
- 2015-08-07 GB GBGB1514015.5A patent/GB201514015D0/en not_active Ceased
-
2016
- 2016-08-05 WO PCT/US2016/045729 patent/WO2017027357A1/fr not_active Ceased
- 2016-08-05 EP EP16751125.2A patent/EP3331878A1/fr not_active Withdrawn
- 2016-08-05 US US15/750,817 patent/US11110089B2/en not_active Expired - Fee Related
- 2016-08-05 MA MA042913A patent/MA42913A/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB201514015D0 (en) | 2015-09-23 |
| EP3331878A1 (fr) | 2018-06-13 |
| WO2017027357A8 (fr) | 2017-04-20 |
| US11110089B2 (en) | 2021-09-07 |
| US20200113897A1 (en) | 2020-04-16 |
| WO2017027357A1 (fr) | 2017-02-16 |
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