MA43169A - Composés hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-gamma - Google Patents
Composés hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-gammaInfo
- Publication number
- MA43169A MA43169A MA043169A MA43169A MA43169A MA 43169 A MA43169 A MA 43169A MA 043169 A MA043169 A MA 043169A MA 43169 A MA43169 A MA 43169A MA 43169 A MA43169 A MA 43169A
- Authority
- MA
- Morocco
- Prior art keywords
- pi3k
- compounds used
- heterocyclic compounds
- gamma inhibitors
- gamma
- Prior art date
Links
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Transplantation (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562252050P | 2015-11-06 | 2015-11-06 | |
| PCT/US2016/060468 WO2017079519A1 (fr) | 2015-11-06 | 2016-11-04 | Composés hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-gamma |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MA43169A true MA43169A (fr) | 2018-09-12 |
| MA43169B1 MA43169B1 (fr) | 2022-05-31 |
Family
ID=57460598
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA43169A MA43169B1 (fr) | 2015-11-06 | 2016-11-04 | Composés héterocycliques en tant qu' inhibiteurs pi3k-gamma |
Country Status (19)
| Country | Link |
|---|---|
| US (4) | US10065963B2 (fr) |
| EP (2) | EP4086259A1 (fr) |
| JP (1) | JP6854817B2 (fr) |
| AR (1) | AR106595A1 (fr) |
| CY (1) | CY1125245T1 (fr) |
| DK (1) | DK3371190T3 (fr) |
| ES (1) | ES2915550T3 (fr) |
| HR (1) | HRP20220599T1 (fr) |
| HU (1) | HUE059324T2 (fr) |
| LT (1) | LT3371190T (fr) |
| MA (1) | MA43169B1 (fr) |
| MD (1) | MD3371190T2 (fr) |
| PL (1) | PL3371190T3 (fr) |
| PT (1) | PT3371190T (fr) |
| RS (1) | RS63359B1 (fr) |
| SI (1) | SI3371190T1 (fr) |
| SM (1) | SMT202200250T1 (fr) |
| TW (2) | TWI744256B (fr) |
| WO (1) | WO2017079519A1 (fr) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2966581A1 (fr) | 2014-11-06 | 2016-05-12 | Lysosomal Therapeutics Inc. | Pyrrolo[1,2-a]pyrimidines substituees et leur utilisation dans le traitement de troubles medicaux |
| US20170333435A1 (en) | 2014-11-06 | 2017-11-23 | Lysosomal Therapeutics Inc. | Substituted imidazo[1,5-a]pyrimidines and their use in the treatment of medical disorders |
| HRP20240644T1 (hr) | 2014-11-06 | 2024-08-02 | Bial-R&D Investments, S.A. | Supstituirani pirazolo(1,5-a)pirimidini i njihova uporaba u liječenju medicinskih poremećaja |
| US9586949B2 (en) | 2015-02-09 | 2017-03-07 | Incyte Corporation | Aza-heteroaryl compounds as PI3K-gamma inhibitors |
| EP4086259A1 (fr) | 2015-11-06 | 2022-11-09 | Incyte Corporation | Composés hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-gamma |
| WO2017120194A1 (fr) | 2016-01-05 | 2017-07-13 | Incyte Corporation | Pyridine et utilisation de composés de la pyridimine comme inhibiteurs de pi3k-gamma |
| WO2017144633A1 (fr) * | 2016-02-25 | 2017-08-31 | Asceneuron S. A. | Inhibiteurs de glycosidases |
| US11124516B2 (en) | 2016-04-06 | 2021-09-21 | BIAL-BioTech Investments, Inc. | Pyrrolo[1,2-A]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders |
| JP7046827B2 (ja) | 2016-04-06 | 2022-04-04 | リソソーマル・セラピューティクス・インコーポレイテッド | イミダゾ[1,5-a]ピリミジニルカルボキサミド化合物および医学的障害の処置におけるその使用 |
| SG11201808830YA (en) | 2016-04-06 | 2018-11-29 | Lysosomal Therapeutics Inc | Pyrazolo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders |
| JP7164774B2 (ja) | 2016-05-05 | 2022-11-02 | ビアル-アール・アンド・ディ・インベストメンツ・ソシエダーデ・アノニマ | 置換イミダゾ[1,2-b]ピリダジン、置換イミダゾ[1,5-b]ピリダジン、関連化合物、および医学的障害の治療におけるその使用 |
| WO2017192931A1 (fr) | 2016-05-05 | 2017-11-09 | Lysosomal Therapeutics Inc. | Imidazo[1,2-a]pyridines substituées, imidazo[1,2-a]pyrazines substituées, composés apparentés et leur utilisation dans le traitement de troubles médicaux |
| WO2017223414A1 (fr) | 2016-06-24 | 2017-12-28 | Incyte Corporation | Composants hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-y |
| TWI795381B (zh) | 2016-12-21 | 2023-03-11 | 比利時商健生藥品公司 | 作為malt1抑制劑之吡唑衍生物 |
| BR112020001695A2 (pt) * | 2017-07-28 | 2020-07-21 | Turning Point Therapeutics, Inc. | compostos macrocíclicos e usos dos mesmos |
| IL295978B2 (en) | 2017-10-18 | 2024-01-01 | Incyte Corp | Condensed imidazole derivatives substituted by tertiary hydroxy groups as pi3k-gamma inhibitors |
| WO2019120212A1 (fr) * | 2017-12-19 | 2019-06-27 | 基石药业(苏州)有限公司 | Inhibiteur d'ido |
| CR20250050A (es) | 2018-09-05 | 2025-03-19 | Incyte Corp | Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165) |
| CN113874021B (zh) | 2019-03-26 | 2024-07-09 | 温缇克斯生物科学公司 | Tyk2假激酶配体 |
| EP3953345B1 (fr) | 2019-04-11 | 2023-04-05 | Janssen Pharmaceutica NV | Dérivés de pyridines comme inhibiteurs de malt1 |
| AU2020288610A1 (en) | 2019-06-04 | 2022-01-27 | Arcus Biosciences, Inc. | 2,3,5-trisubstituted pyrazolo[1,5-a]pyrimidine compounds |
| AU2020289537A1 (en) * | 2019-06-06 | 2021-11-25 | Aligos Therapeutics, Inc. | Heterocyclic compounds |
| AU2020378345A1 (en) | 2019-11-08 | 2022-06-02 | Ventyx Biosciences, Inc. | TYK2 pseudokinase ligands |
| CN116348453B (zh) * | 2021-04-25 | 2025-07-04 | 烨辉医药科技(上海)有限公司 | 杂芳族甲酰胺化合物及其用途 |
| WO2025146216A1 (fr) * | 2024-01-05 | 2025-07-10 | 成都赜灵生物医药科技有限公司 | Composés d'amide fusionné à n-hétérocycle à six chaînons et à cinq chaînons et leur utilisation |
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| TW201406761A (zh) | 2012-05-18 | 2014-02-16 | Incyte Corp | 做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物 |
| JP6217629B2 (ja) | 2012-05-31 | 2017-10-25 | 住友化学株式会社 | 縮合複素環化合物 |
| BR112015000675B1 (pt) | 2012-07-13 | 2022-07-12 | UCB Biopharma SRL | Derivados de imidazopiridina como moduladores da atividade de tnf |
| AU2013337824B2 (en) | 2012-11-01 | 2018-03-08 | Incyte Holdings Corporation | Tricyclic fused thiophene derivatives as JAK inhibitors |
| TWI736135B (zh) | 2013-03-01 | 2021-08-11 | 美商英塞特控股公司 | 吡唑并嘧啶衍生物治療PI3Kδ相關病症之用途 |
| WO2014149207A2 (fr) | 2013-03-15 | 2014-09-25 | Dow Agrosciences Llc | Compositions insecticides à base de benzimidazole et procédés apparentés |
| EP2976077A4 (fr) | 2013-03-22 | 2016-11-30 | Scripps Research Inst | Benzimidazoles substitués en tant que modulateurs d'un récepteur de nociceptine |
| EP2994142A4 (fr) | 2013-05-08 | 2017-03-29 | Colorado Seminary, Which Owns and Operates The University of Denver | Agents antibiotiques et antiparasitaires qui modulent la fructose 1,6-bisphosphate aldolase de classe ii |
| SMT202100040T1 (it) | 2013-05-17 | 2021-03-15 | Incyte Corp | Derivati di bipirazolo come inibitori di jak |
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| EP2930048A1 (fr) | 2014-04-10 | 2015-10-14 | Johnson Controls Automotive Electronics SAS | Dispositif d'affichage tête haute projetant des informations visuelles sur un écran |
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| WO2016054491A1 (fr) * | 2014-10-03 | 2016-04-07 | Infinity Pharmaceuticals, Inc. | Composés hétérocycliques et leurs utilisations |
| MA40933A (fr) | 2014-11-11 | 2017-09-19 | Piqur Therapeutics Ag | Difluorométhyl-aminopyridines et difluorométhyl-aminopyrimidines |
| US9586949B2 (en) | 2015-02-09 | 2017-03-07 | Incyte Corporation | Aza-heteroaryl compounds as PI3K-gamma inhibitors |
| EP4086259A1 (fr) | 2015-11-06 | 2022-11-09 | Incyte Corporation | Composés hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-gamma |
| WO2017120194A1 (fr) | 2016-01-05 | 2017-07-13 | Incyte Corporation | Pyridine et utilisation de composés de la pyridimine comme inhibiteurs de pi3k-gamma |
| WO2017223414A1 (fr) | 2016-06-24 | 2017-12-28 | Incyte Corporation | Composants hétérocycliques utilisés en tant qu'inhibiteurs de pi3k-y |
-
2016
- 2016-11-04 EP EP22162035.4A patent/EP4086259A1/fr not_active Withdrawn
- 2016-11-04 MA MA43169A patent/MA43169B1/fr unknown
- 2016-11-04 LT LTEPPCT/US2016/060468T patent/LT3371190T/lt unknown
- 2016-11-04 PL PL16805238.9T patent/PL3371190T3/pl unknown
- 2016-11-04 JP JP2018523015A patent/JP6854817B2/ja not_active Expired - Fee Related
- 2016-11-04 DK DK16805238.9T patent/DK3371190T3/da active
- 2016-11-04 SM SM20220250T patent/SMT202200250T1/it unknown
- 2016-11-04 SI SI201631549T patent/SI3371190T1/sl unknown
- 2016-11-04 MD MDE20180887T patent/MD3371190T2/ro unknown
- 2016-11-04 AR ARP160103370A patent/AR106595A1/es unknown
- 2016-11-04 ES ES16805238T patent/ES2915550T3/es active Active
- 2016-11-04 HU HUE16805238A patent/HUE059324T2/hu unknown
- 2016-11-04 WO PCT/US2016/060468 patent/WO2017079519A1/fr not_active Ceased
- 2016-11-04 HR HRP20220599TT patent/HRP20220599T1/hr unknown
- 2016-11-04 TW TW105136055A patent/TWI744256B/zh active
- 2016-11-04 EP EP16805238.9A patent/EP3371190B1/fr active Active
- 2016-11-04 PT PT168052389T patent/PT3371190T/pt unknown
- 2016-11-04 TW TW110136698A patent/TWI824309B/zh active
- 2016-11-04 US US15/343,375 patent/US10065963B2/en active Active
- 2016-11-04 RS RS20220521A patent/RS63359B1/sr unknown
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2018
- 2018-07-25 US US16/045,358 patent/US10472368B2/en active Active
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2019
- 2019-10-01 US US16/589,523 patent/US11091491B2/en not_active Expired - Fee Related
-
2021
- 2021-06-24 US US17/356,984 patent/US11773102B2/en active Active
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2022
- 2022-06-10 CY CY20221100410T patent/CY1125245T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK3371190T3 (da) | 2022-05-23 |
| MD3371190T2 (ro) | 2022-09-30 |
| HUE059324T2 (hu) | 2022-11-28 |
| EP3371190B1 (fr) | 2022-03-30 |
| RS63359B1 (sr) | 2022-07-29 |
| US10472368B2 (en) | 2019-11-12 |
| CY1125245T1 (el) | 2025-03-28 |
| TWI744256B (zh) | 2021-11-01 |
| JP2018532760A (ja) | 2018-11-08 |
| AR106595A1 (es) | 2018-01-31 |
| MA43169B1 (fr) | 2022-05-31 |
| US20230009843A1 (en) | 2023-01-12 |
| TWI824309B (zh) | 2023-12-01 |
| HRP20220599T1 (hr) | 2022-06-24 |
| US20200031837A1 (en) | 2020-01-30 |
| US10065963B2 (en) | 2018-09-04 |
| PT3371190T (pt) | 2022-07-08 |
| SMT202200250T1 (it) | 2022-07-21 |
| JP6854817B2 (ja) | 2021-04-07 |
| ES2915550T3 (es) | 2022-06-23 |
| EP3371190A1 (fr) | 2018-09-12 |
| TW202204362A (zh) | 2022-02-01 |
| LT3371190T (lt) | 2022-08-10 |
| US20170129899A1 (en) | 2017-05-11 |
| US11773102B2 (en) | 2023-10-03 |
| US20190062336A1 (en) | 2019-02-28 |
| PL3371190T3 (pl) | 2022-11-07 |
| TW201726679A (zh) | 2017-08-01 |
| US11091491B2 (en) | 2021-08-17 |
| EP4086259A1 (fr) | 2022-11-09 |
| SI3371190T1 (sl) | 2022-08-31 |
| WO2017079519A1 (fr) | 2017-05-11 |
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