MA51224A - Composés de sulfonamide et leur utilisation - Google Patents

Composés de sulfonamide et leur utilisation

Info

Publication number
MA51224A
MA51224A MA051224A MA51224A MA51224A MA 51224 A MA51224 A MA 51224A MA 051224 A MA051224 A MA 051224A MA 51224 A MA51224 A MA 51224A MA 51224 A MA51224 A MA 51224A
Authority
MA
Morocco
Prior art keywords
sulfonamide compounds
sulfonamide
compounds
Prior art date
Application number
MA051224A
Other languages
English (en)
Inventor
Nathan Gignac
Hiroyuki Nakamura
Jing Teng
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of MA51224A publication Critical patent/MA51224A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/1131,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C63/00Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
    • C07C63/04Monocyclic monocarboxylic acids
    • C07C63/06Benzoic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MA051224A 2017-11-29 2018-11-28 Composés de sulfonamide et leur utilisation MA51224A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762592023P 2017-11-29 2017-11-29

Publications (1)

Publication Number Publication Date
MA51224A true MA51224A (fr) 2020-10-07

Family

ID=66665441

Family Applications (1)

Application Number Title Priority Date Filing Date
MA051224A MA51224A (fr) 2017-11-29 2018-11-28 Composés de sulfonamide et leur utilisation

Country Status (15)

Country Link
US (2) US12344588B2 (fr)
EP (1) EP3717462B1 (fr)
JP (1) JP6846574B2 (fr)
KR (1) KR102480074B1 (fr)
CN (1) CN111386260B (fr)
AU (1) AU2018377036B2 (fr)
CA (1) CA3084030C (fr)
ES (1) ES2969901T3 (fr)
MA (1) MA51224A (fr)
MX (1) MX2020005478A (fr)
MY (1) MY201832A (fr)
PH (1) PH12020550703A1 (fr)
SG (1) SG11202004877UA (fr)
TW (1) TWI762743B (fr)
WO (1) WO2019106579A1 (fr)

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* Cited by examiner, † Cited by third party
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AU2017275209C1 (en) 2016-05-31 2020-01-23 Taiho Pharmaceutical Co., Ltd. Sulfonamide compound or salt thereof
US11439623B2 (en) 2017-04-04 2022-09-13 Case Western Reserve University Method of modulating ribonucleotide reductase
AU2018377036B2 (en) 2017-11-29 2022-04-14 Taiho Pharmaceutical Co., Ltd. Sulfonamide compounds and use thereof
WO2022187200A1 (fr) * 2021-03-02 2022-09-09 Boundless Bio, Inc. Inhibiteurs de ribonucléotide réductase (rnr) et leurs utilisations
WO2023043938A1 (fr) * 2021-09-17 2023-03-23 Boundless Bio, Inc. Inhibiteurs de ribonucléotide réductase (rnr) de sulfamide et leurs utilisations
TW202328121A (zh) * 2021-09-17 2023-07-16 美商無界生物公司 環狀磺醯胺核糖核苷酸還原酶(rnr)抑制劑及其用途
JP2025531147A (ja) * 2022-09-13 2025-09-19 バウンドレス バイオ,インク. 環状スルホンアミドリボヌクレオチドレダクターゼ(rnr)阻害剤およびその使用
WO2025240847A1 (fr) 2024-05-17 2025-11-20 Revolution Medicines, Inc. Inhibiteurs de ras
WO2025255438A1 (fr) 2024-06-07 2025-12-11 Revolution Medicines, Inc. Procédés de traitement d'une maladie ou d'un trouble lié à la protéine ras
WO2025265060A1 (fr) 2024-06-21 2025-12-26 Revolution Medicines, Inc. Compositions thérapeutiques et procédés de gestion d'effets liés au traitement
WO2026006747A1 (fr) 2024-06-28 2026-01-02 Revolution Medicines, Inc. Inhibiteurs de ras
WO2026015825A1 (fr) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Utilisation d'un inhibiteur de ras pour traiter le cancer du pancréas
WO2026015790A1 (fr) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Méthodes de traitement d'une maladie ou d'un trouble lié à ras
WO2026015801A1 (fr) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Méthodes de traitement d'une maladie ou d'un trouble liés à ras
WO2026015796A1 (fr) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Méthodes de traitement d'une maladie ou d'un trouble lié à ras
WO2026050446A1 (fr) 2024-08-29 2026-03-05 Revolution Medicines, Inc. Inhibiteurs de ras
WO2026072904A2 (fr) 2024-09-26 2026-04-02 Revolution Medicines, Inc. Compositions et méthodes de traitement du cancer du poumon
WO2026090116A2 (fr) 2024-10-21 2026-04-30 Revolution Medicines, Inc. Inhibiteurs de ras
WO2026090245A1 (fr) 2024-10-22 2026-04-30 Revolution Medicines, Inc. Utilisation d'inhibiteurs ras pour traiter un cancer
US20260108528A1 (en) 2024-10-22 2026-04-23 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder

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GB9721437D0 (en) 1997-10-10 1997-12-10 Glaxo Group Ltd Heteroaromatic compounds and their use in medicine
ZA991029B (en) * 1998-02-09 1999-09-30 Rhone Poulenc Rorer Pharma Composition and methods for treatment of hiv infections.
AU1182300A (en) * 1998-11-17 2000-06-05 Fuji Photo Film Co., Ltd. Bisaryl compounds and cancer remedies containing the same
AU6894400A (en) * 1999-08-06 2001-03-05 Enzon Pharmaceuticals Inc. Composition and methods for treatment of HIV infection
CA2407799A1 (fr) 2000-05-02 2001-11-08 Sugen, Inc. Derives d'acide acetique (2-oxindole-3-ylidenyl) et leur utilisation comme inhibiteurs de la proteine kinase
EP1313742A1 (fr) 2000-08-31 2003-05-28 Dr. Reddy's Laboratories Ltd. Procede de preparation d'hydrates d'olanzapine et de conversion de ceux-ci en formes cristallines d'olanzapine
PT1537878E (pt) 2002-07-03 2010-11-18 Ono Pharmaceutical Co Composições de imunopotenciação
US20060128783A1 (en) 2002-08-09 2006-06-15 Dinsmore Christopher J Tyrosine kinase inhibitors
RU2383536C2 (ru) 2004-08-04 2010-03-10 Тайсо Фармасьютикал Ко., Лтд. Производное триазола
MY142304A (en) 2005-01-31 2010-11-15 Taiho Pharmaceutical Co Ltd Novel pyrimidine nucleoside compound or salt thereof
TW200736234A (en) * 2006-01-17 2007-10-01 Astrazeneca Ab Chemical compounds
ES2458615T3 (es) * 2006-02-03 2014-05-06 Taisho Pharmaceutical Co., Ltd. Derivado de triazol
KR20100031528A (ko) 2007-06-01 2010-03-22 더 트러스티즈 오브 프린스턴 유니버시티 숙주세포 대사경로의 조절을 통한 바이러스 감염 치료
JP2012508215A (ja) 2008-11-11 2012-04-05 ノバルティス アーゲー 有機化合物
AU2015203322B2 (en) 2009-07-20 2016-09-29 Bristol-Myers Squibb Company Combination of anti-ctla4 antibody with diverse therapeutic regimens for the synergistic treatment of proliferative diseases
EP2552453A2 (fr) 2010-03-30 2013-02-06 Clavis Pharma ASA Procédés d'amélioration du cancer
AU2015210750B2 (en) 2014-01-31 2020-08-20 Children's Medical Center Corporation Antibody molecules to TIM-3 and uses thereof
WO2015138920A1 (fr) 2014-03-14 2015-09-17 Novartis Ag Molécules d'anticorps anti-lag-3 et leurs utilisations
WO2016040882A1 (fr) 2014-09-13 2016-03-17 Novartis Ag Polythérapie par les inhibiteurs de l'egfr
GB201420239D0 (en) 2014-11-14 2014-12-31 Bergenbio As Biomarker
TWI623316B (zh) 2015-12-22 2018-05-11 Taiho Pharmaceutical Co Ltd Antitumor effect enhancer derived from pyrrolopyrimidine compound
US11883404B2 (en) 2016-03-04 2024-01-30 Taiho Pharmaceuticals Co., Ltd. Preparation and composition for treatment of malignant tumors
EP3424505A4 (fr) 2016-03-04 2019-10-16 Taiho Pharmaceutical Co., Ltd. Préparation et composition de traitement de tumeurs malignes
US10889555B2 (en) * 2016-05-31 2021-01-12 Taiho Pharmaceutical Co., Ltd. Sulfonamide compound or salt thereof
AU2017275209C1 (en) 2016-05-31 2020-01-23 Taiho Pharmaceutical Co., Ltd. Sulfonamide compound or salt thereof
US20200405697A1 (en) 2017-11-29 2020-12-31 Taiho Pharmaceutical Co., Ltd. Antitumor Agent
AU2018377036B2 (en) 2017-11-29 2022-04-14 Taiho Pharmaceutical Co., Ltd. Sulfonamide compounds and use thereof
KR20220011562A (ko) 2018-04-25 2022-01-28 안나 마트너 급성 골수성 백혈병에서의 재발 위험 감소 및 생존 연장을 위한 방법 및 조성물

Also Published As

Publication number Publication date
SG11202004877UA (en) 2020-06-29
CA3084030C (fr) 2023-03-21
ES2969901T3 (es) 2024-05-23
AU2018377036A1 (en) 2020-06-18
TW201925182A (zh) 2019-07-01
CA3084030A1 (fr) 2019-06-06
WO2019106579A1 (fr) 2019-06-06
US20200361883A1 (en) 2020-11-19
EP3717462B1 (fr) 2024-01-03
EP3717462A1 (fr) 2020-10-07
CN111386260B (zh) 2024-04-30
BR112020010148A2 (pt) 2020-10-13
RU2020121153A3 (fr) 2021-12-29
KR20200096261A (ko) 2020-08-11
RU2020121153A (ru) 2021-12-29
KR102480074B1 (ko) 2022-12-21
EP3717462A4 (fr) 2021-07-21
PH12020550703A1 (en) 2021-04-26
JP2021504432A (ja) 2021-02-15
MY201832A (en) 2024-03-19
MX2020005478A (es) 2020-08-27
JP6846574B2 (ja) 2021-03-24
TWI762743B (zh) 2022-05-01
US20250223270A1 (en) 2025-07-10
CN111386260A (zh) 2020-07-07
AU2018377036B2 (en) 2022-04-14
US12344588B2 (en) 2025-07-01

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