MA52337A - Nouveaux analogues d'oxaborole et utilisations de ces derniers - Google Patents
Nouveaux analogues d'oxaborole et utilisations de ces derniersInfo
- Publication number
- MA52337A MA52337A MA052337A MA52337A MA52337A MA 52337 A MA52337 A MA 52337A MA 052337 A MA052337 A MA 052337A MA 52337 A MA52337 A MA 52337A MA 52337 A MA52337 A MA 52337A
- Authority
- MA
- Morocco
- Prior art keywords
- oxaborole
- analogues
- latest
- new
- oxaborole analogues
- Prior art date
Links
- OHENQANLQNOMAO-UHFFFAOYSA-N oxaborole Chemical class O1B=CC=C1 OHENQANLQNOMAO-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762465294P | 2017-03-01 | 2017-03-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA52337A true MA52337A (fr) | 2021-03-03 |
Family
ID=63370509
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA052337A MA52337A (fr) | 2017-03-01 | 2018-03-01 | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
Country Status (4)
| Country | Link |
|---|---|
| US (2) | US10961261B2 (fr) |
| EP (1) | EP3609504A4 (fr) |
| MA (1) | MA52337A (fr) |
| WO (1) | WO2018160845A1 (fr) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| NZ745681A (en) | 2016-03-07 | 2022-05-27 | Agrofresh Inc | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| EP3609504A4 (fr) | 2017-03-01 | 2021-03-03 | Anacor Pharmaceuticals, Inc. | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
| US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
| KR20250005365A (ko) | 2022-04-28 | 2025-01-09 | 니혼노야쿠가부시키가이샤 | 옥심기를 갖는 함질소 복소환 화합물 및 상기 화합물을 함유하는 농원예용 제초제 및 이들의 사용방법 |
| TR2023001878A1 (tr) * | 2023-02-20 | 2024-08-21 | Univ Yeditepe | Borun nöronal kaynakli lei̇shmani̇asi̇s hastaliğinin tedavi̇si̇ i̇çi̇n kullanimi |
| CN118724752B (zh) * | 2023-03-29 | 2025-11-28 | 重庆博腾制药科技股份有限公司 | 一种酪氨酸激酶抑制剂中间体、制备方法及其应用 |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA05006685A (es) | 2002-12-18 | 2005-12-14 | Anacor Pharmaceuticals Inc | Antibioticos que contienen complejos de acido borinico y metodos de uso. |
| US7465836B2 (en) | 2003-06-16 | 2008-12-16 | Anacor Pharmaceuticals, Inc. | Hydrolytically-resistant boron-containing therapeutics and methods of use |
| AR049915A1 (es) | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Compuestos con contenido de boro y metodos de uso de los mismos |
| ATE447960T1 (de) | 2004-06-14 | 2009-11-15 | Anacor Pharmaceuticals Inc | Antivirale verwendung von borinsäurekomplexen |
| HRP20150710T1 (hr) | 2006-02-16 | 2015-08-14 | Anacor Pharmaceuticals, Inc. | Male molekule koje sadrže bor kao protu-upalni agensi |
| BRPI0711155A2 (pt) | 2006-05-02 | 2011-08-23 | Anacor Pharmaceuticals Inc | terapêuticos contendo boro resistentes hidroliticamente e métodos de uso |
| WO2007146965A2 (fr) | 2006-06-12 | 2007-12-21 | Anacor Pharmaceuticals, Inc. | Composés destinés au traitement d'une maladie périodontale |
| JO3396B1 (ar) | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
| EP2187893A4 (fr) | 2008-03-06 | 2012-02-22 | Anacor Pharmaceuticals Inc | Petites molécules contenant du bore utilisées en tant qu'agents anti-inflammatoires |
| JP2011515359A (ja) * | 2008-03-18 | 2011-05-19 | グラクソ グループ リミテッド | 治療用トリアゾールアミド誘導体 |
| US20100256092A1 (en) | 2008-05-12 | 2010-10-07 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2010027975A1 (fr) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore |
| WO2010045503A1 (fr) | 2008-10-15 | 2010-04-22 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore en tant qu’agents antiprotozoaires |
| WO2010045505A1 (fr) | 2008-10-15 | 2010-04-22 | Anacor Pharmaceuticals, Inc | Petites molécules contenant du bore en tant qu’agents antiprotozoaires |
| CN102256494A (zh) | 2008-12-17 | 2011-11-23 | 阿纳科制药公司 | (s)-3-氨甲基-7-(3-羟基-丙氧基)-3h-苯并[c][1,2]氧杂硼杂环戊-1-醇的多晶型物 |
| JP2013500974A (ja) | 2009-07-28 | 2013-01-10 | アナコール ファーマシューティカルズ,インコーポレイテッド | 三置換ホウ素含有分子 |
| US9440994B2 (en) * | 2009-08-14 | 2016-09-13 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules as antiprotozoal agents |
| WO2011022337A1 (fr) | 2009-08-19 | 2011-02-24 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore en tant qu'agents anti-protozoaires |
| WO2011037731A1 (fr) | 2009-09-25 | 2011-03-31 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore |
| US9346834B2 (en) | 2009-10-20 | 2016-05-24 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| WO2011060199A1 (fr) | 2009-11-11 | 2011-05-19 | Anacor Pharmaceuticals, Inc. | Petites molecules contenant du bore |
| WO2011094450A1 (fr) | 2010-01-27 | 2011-08-04 | Anacor Pharmaceuticals, Inc | Petites molecules contenant du bore |
| US8623911B2 (en) | 2010-03-19 | 2014-01-07 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agent |
| PT3251678T (pt) | 2010-09-07 | 2021-11-22 | Anacor Pharmaceuticals Inc | Derivados de benzoxaborol para tratamento de infeções bacterianas |
| WO2012145734A1 (fr) * | 2011-04-22 | 2012-10-26 | The Ohio State University | Compositions antileshmaniennes et ses méthodes d'utilisation |
| AR088668A1 (es) | 2011-11-21 | 2014-06-25 | Lilly Co Eli | Moleculas pequeñas que contienen boro |
| AR088669A1 (es) | 2011-11-21 | 2014-06-25 | Lilly Co Eli | Derivados de dihidrodibenzo[c][1,2]oxaborol y dihidroisoxazol utiles para el control de ectoparasitos |
| WO2014078802A1 (fr) | 2012-11-19 | 2014-05-22 | Irm Llc | Composés et compositions pour le traitement de maladies parasitaires |
| AP2015008638A0 (en) * | 2013-02-01 | 2015-08-31 | Anacor Pharmaceuticals Inc | Boron-containing small molecules as antiprotozoal agents |
| WO2015013318A1 (fr) | 2013-07-22 | 2015-01-29 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore |
| EP3609504A4 (fr) | 2017-03-01 | 2021-03-03 | Anacor Pharmaceuticals, Inc. | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
-
2018
- 2018-03-01 EP EP18761407.8A patent/EP3609504A4/fr active Pending
- 2018-03-01 WO PCT/US2018/020464 patent/WO2018160845A1/fr not_active Ceased
- 2018-03-01 US US16/489,824 patent/US10961261B2/en active Active
- 2018-03-01 MA MA052337A patent/MA52337A/fr unknown
-
2021
- 2021-02-11 US US17/173,884 patent/US11691992B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP3609504A4 (fr) | 2021-03-03 |
| EP3609504A1 (fr) | 2020-02-19 |
| US11691992B2 (en) | 2023-07-04 |
| US10961261B2 (en) | 2021-03-30 |
| US20210253605A1 (en) | 2021-08-19 |
| US20200024289A1 (en) | 2020-01-23 |
| WO2018160845A1 (fr) | 2018-09-07 |
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