MA56930B1 - L'inhibiteur de vmat2 valbenazine pour son utilisation dans une méthode de traitement d'un trouble neurologique ou psychiatrique chez des patients présentant une insuffisance rénale grave - Google Patents

L'inhibiteur de vmat2 valbenazine pour son utilisation dans une méthode de traitement d'un trouble neurologique ou psychiatrique chez des patients présentant une insuffisance rénale grave

Info

Publication number
MA56930B1
MA56930B1 MA56930A MA56930A MA56930B1 MA 56930 B1 MA56930 B1 MA 56930B1 MA 56930 A MA56930 A MA 56930A MA 56930 A MA56930 A MA 56930A MA 56930 B1 MA56930 B1 MA 56930B1
Authority
MA
Morocco
Prior art keywords
valbenazine
neurological
patients
treating
severe renal
Prior art date
Application number
MA56930A
Other languages
English (en)
Inventor
Gordon Raphael LOEWEN
Sha Rosa Luo
Original Assignee
Neurocrine Biosciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=72292706&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA56930(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Neurocrine Biosciences, Inc. filed Critical Neurocrine Biosciences, Inc.
Publication of MA56930B1 publication Critical patent/MA56930B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

L'invention concerne un procédé d'administration d'un inhibiteur du transporteur de monoamine vésiculaire 2 (VMAT2) à un sujet en ayant besoin, le sujet présentant une insuffisance rénale sévère.
MA56930A 2019-08-23 2020-08-21 L'inhibiteur de vmat2 valbenazine pour son utilisation dans une méthode de traitement d'un trouble neurologique ou psychiatrique chez des patients présentant une insuffisance rénale grave MA56930B1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201962890697P 2019-08-23 2019-08-23
US202063028754P 2020-05-22 2020-05-22
EP20764910.4A EP4017494B1 (fr) 2019-08-23 2020-08-21 L'inhibiteur de vmat2 valbenazine pour son utilisation dans une méthode de traitement d'un trouble neurologique ou psychiatrique chez des patients présentant une insuffisance rénale grave
PCT/US2020/047392 WO2021041208A1 (fr) 2019-08-23 2020-08-21 Procédés d'administration de certains inhibiteurs de vmat2 à des patients présentant une insuffisance rénale grave

Publications (1)

Publication Number Publication Date
MA56930B1 true MA56930B1 (fr) 2025-10-31

Family

ID=72292706

Family Applications (1)

Application Number Title Priority Date Filing Date
MA56930A MA56930B1 (fr) 2019-08-23 2020-08-21 L'inhibiteur de vmat2 valbenazine pour son utilisation dans une méthode de traitement d'un trouble neurologique ou psychiatrique chez des patients présentant une insuffisance rénale grave

Country Status (26)

Country Link
US (1) US10940141B1 (fr)
EP (2) EP4652986A3 (fr)
JP (2) JP7603662B2 (fr)
KR (1) KR20220051239A (fr)
CN (1) CN114679906A (fr)
AU (2) AU2020336017B2 (fr)
BR (1) BR112022002834A2 (fr)
CA (1) CA3149033A1 (fr)
DK (1) DK4017494T3 (fr)
ES (1) ES3040583T3 (fr)
FI (1) FI4017494T3 (fr)
HR (1) HRP20251281T1 (fr)
HU (1) HUE073484T2 (fr)
IL (1) IL290686B2 (fr)
JO (1) JOP20220040A1 (fr)
LT (1) LT4017494T (fr)
MA (1) MA56930B1 (fr)
MD (1) MD4017494T2 (fr)
MX (1) MX2022000559A (fr)
PH (1) PH12022550385A1 (fr)
PT (1) PT4017494T (fr)
RS (1) RS67194B1 (fr)
SI (1) SI4017494T1 (fr)
SM (1) SMT202500480T1 (fr)
TW (1) TWI894161B (fr)
WO (1) WO2021041208A1 (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3051830A1 (fr) 2017-01-27 2018-08-02 Neurocrine Bioscienes, Inc. Methodes d'administration de certains inhibiteurs de vmat2
CA3076000A1 (fr) 2017-09-21 2019-03-28 Neurocrine Biosciences, Inc. Formulation de valbenazine a dosage eleve et compositions, procedes et kits associes
JP2021502959A (ja) 2017-10-10 2021-02-04 ニューロクライン バイオサイエンシーズ，インコーポレイテッド 特定のｖｍａｔ２インヒビターを投与するための方法
MA53239A (fr) 2018-08-15 2022-05-04 Neurocrine Biosciences Inc Procédés d'administration de certains inhibiteurs de vmat2
WO2022221551A1 (fr) * 2021-04-15 2022-10-20 Neurocrine Biosciences, Inc. Méthodes d'administration de certains inhibiteurs de vmat2
BR112023021257A2 (pt) * 2021-04-15 2023-12-12 Neurocrine Biosciences Inc Métodos para a administração combinada de deutetrabenzina e um cyp2d6
CA3220946A1 (fr) 2021-06-30 2023-01-05 Angel S. Angelov Valbenazine destinee a etre utilisee dans le traitement complementaire de la schizophrenie
BR112023026160A2 (pt) 2021-06-30 2024-03-05 Neurocrine Biosciences Inc Valbenazina para uso no tratamento de discinesia devido à paralisia cerebral
EP4489754A1 (fr) 2022-03-07 2025-01-15 Neurocrine Biosciences, Inc. Valbénazine, inhibiteur de vmat2, en tant que base libre d'un tosylate ou d'un sel de ditosylate, destinée à être utilisée dans le traitement de la chorée associée à la maladie de huntington
WO2025038959A1 (fr) 2023-08-17 2025-02-20 Neurocrine Biosciences, Inc. Méthodes d'administration de certains inhibiteurs de vmat2
TW202521119A (zh) 2023-08-17 2025-06-01 美商紐羅克里生物科學有限公司 用於投與特定vmat2抑制劑之方法
WO2025096823A1 (fr) 2023-11-01 2025-05-08 Neurocrine Biosciences, Inc. Amélioration, maintien ou réduction du déclin de la fonction motrice associé à la maladie de huntington en utilisant de la valbénazine
WO2025188830A1 (fr) 2024-03-06 2025-09-12 Neurocrine Biosciences, Inc. Méthodes d'administration de certains inhibiteurs de vmat2

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