MC1394A1 - Nouveaux derives de l'imidazole - Google Patents

Nouveaux derives de l'imidazole

Info

Publication number
MC1394A1
MC1394A1 MC811517A MC1517A MC1394A1 MC 1394 A1 MC1394 A1 MC 1394A1 MC 811517 A MC811517 A MC 811517A MC 1517 A MC1517 A MC 1517A MC 1394 A1 MC1394 A1 MC 1394A1
Authority
MC
Monaco
Prior art keywords
formula
compound
butyl
tert
imidazole
Prior art date
Application number
MC811517A
Other languages
English (en)
French (fr)
Inventor
Romano Derungs
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1394A1 publication Critical patent/MC1394A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Fats And Perfumes (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Epoxy Resins (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
MC811517A 1980-06-05 1981-06-03 Nouveaux derives de l'imidazole MC1394A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH434780 1980-06-05

Publications (1)

Publication Number Publication Date
MC1394A1 true MC1394A1 (fr) 1982-04-27

Family

ID=4274400

Family Applications (1)

Application Number Title Priority Date Filing Date
MC811517A MC1394A1 (fr) 1980-06-05 1981-06-03 Nouveaux derives de l'imidazole

Country Status (22)

Country Link
US (1) US4582844A (cs)
EP (1) EP0041652B1 (cs)
JP (1) JPS5731667A (cs)
KR (1) KR850000126B1 (cs)
AT (1) ATE6369T1 (cs)
AU (1) AU7111581A (cs)
BR (1) BR8103553A (cs)
CA (1) CA1161847A (cs)
CS (1) CS220340B2 (cs)
DE (1) DE3162356D1 (cs)
DK (1) DK193181A (cs)
ES (1) ES502777A0 (cs)
FI (1) FI811527L (cs)
GR (1) GR77076B (cs)
IL (1) IL63009A0 (cs)
MC (1) MC1394A1 (cs)
NO (1) NO811908L (cs)
NZ (1) NZ197248A (cs)
PH (1) PH15876A (cs)
PT (1) PT73143B (cs)
ZA (1) ZA813644B (cs)
ZW (1) ZW10781A1 (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4501892A (en) * 1982-07-28 1985-02-26 The Upjohn Company Pyridyl benzenediols
IT1193608B (it) * 1983-01-21 1988-07-21 Pierrel Spa Derivati di arilossipropanolamina,procedimento per la loro preparazione composizioni farmaceutiche che li contengono e loro impiego terapeutico
US4790775A (en) * 1988-02-09 1988-12-13 E. I. Du Pont De Nemours And Company Transition connector
US8182528B2 (en) 2003-12-23 2012-05-22 Sadra Medical, Inc. Locking heart valve anchor
JP6064653B2 (ja) * 2013-02-15 2017-01-25 東洋インキScホールディングス株式会社 蛍光材料、蛍光性樹脂組成物および化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE585555A (cs) * 1960-03-31
US3473901A (en) * 1963-02-08 1969-10-21 Rohm & Haas Fuel compositions
CH496710A (de) * 1967-12-16 1970-09-30 Basf Ag Verfahren zur Herstellung von substituierten Imidazolen
DD99787A1 (cs) * 1969-06-23 1973-08-20
US3707475A (en) * 1970-11-16 1972-12-26 Pfizer Antiinflammatory imidazoles
DE2701372A1 (de) * 1977-01-14 1978-07-20 Veba Chemie Ag Verfahren zur herstellung cyclischer amidine
DE2733466A1 (de) * 1977-07-25 1979-02-22 Basf Ag Verfahren zur herstellung von imidazolen

Also Published As

Publication number Publication date
AU7111581A (en) 1981-12-10
KR850000126B1 (ko) 1985-02-27
JPS5731667A (en) 1982-02-20
CA1161847A (en) 1984-02-07
DK193181A (da) 1981-12-06
NZ197248A (en) 1984-07-31
NO811908L (no) 1981-12-07
PT73143A (en) 1981-07-01
EP0041652A1 (de) 1981-12-16
EP0041652B1 (de) 1984-02-22
FI811527A7 (fi) 1981-12-06
IL63009A0 (en) 1981-09-13
DE3162356D1 (en) 1984-03-29
ES8300755A1 (es) 1982-11-16
ES502777A0 (es) 1982-11-16
KR830006229A (ko) 1983-09-20
PT73143B (en) 1983-05-11
US4582844A (en) 1986-04-15
BR8103553A (pt) 1982-03-02
GR77076B (cs) 1984-09-06
ZW10781A1 (en) 1981-12-30
CS220340B2 (en) 1983-03-25
FI811527L (fi) 1981-12-06
ATE6369T1 (de) 1984-03-15
ZA813644B (en) 1982-06-30
PH15876A (en) 1983-04-13

Similar Documents

Publication Publication Date Title
MC1241A1 (fr) Derives de l'imidazole et leur preparation et preparation de medicaments contenant ces substances
FR2501686A1 (fr) Nouveaux derives de 3,4-dihydro-5h-2,3-benzodiazepine, procede pour les preparer et medicaments les contenant
FR2561647A1 (fr) Derives de 1-(hydroxymethyl)-1,6,7,11b-tetrahydro-2h,4h-(1,3)-oxazino- ou -thiazino(4,3,a)isoquinoleine, procede pour leur preparation et compositions pharmaceutiques les contenant
MC1769A1 (fr) Diphenaylpiperidines n-substituees
FR2468601A1 (fr) Nouveaux derives de flavanne utiles notamment comme anticonvulsivants
FR2756560A1 (fr) Nouveaux derives de l'imidazoline, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
MC1332A1 (fr) Nouveaux derives de quinazoline et preparations pharmaceutiques
MC1394A1 (fr) Nouveaux derives de l'imidazole
EP0002978B1 (fr) Dérivés de thiazolidinedione-2,4, leur préparation et leur application en thérapeutique
US4061769A (en) Method and composition for treating hypertension
FR2602771A1 (fr) Nouveaux derives de la benzyl-4 piperazine, leur preparation et les compositions pharmaceutiques qui les contiennent
CA2000247A1 (fr) Derives de methyl-4 ¬(phenyl-4 piperazinyl-1)-2 ethyl -5| thiazole, leur procede de preparation et les compositions pharmaceutiques, en contenant
FR2669030A1 (fr) Nouveaux derives d'imidazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
EP0196943B1 (fr) Nouveaux dérivés 8-thiotétrahydroquinoléines et leurs sels
FR2528846A1 (fr) Nouveau derive de la pyrazolo (1,5-a) pyridine, sa preparation et les compositions pharmaceutiques qui le contiennent
JPS62283967A (ja) ド−パミン−β−ヒドロキシラ−ゼ抑制剤
MC593A1 (fr) Nouveaux benzène sulfonyl-semicarbazides et leur préparation
FR2516510A1 (fr) Derives de la (trimethoxy-3,4,5-cinnamoyl)-1-aminocarbonylethyl-4-piperazine substituee utilisables en pharmacie et procede pour leur preparation
EP0037777B1 (fr) Procédé de préparation de cycloalcoyl propanol amines utiles comme médicaments
WO1991017984A1 (fr) Derives d'(alkylthio-3 propyl)-3 benzothiazoline, leur preparation et les medicaments les contenant
MC1393A1 (fr) Nouveaux derives de l'imidazole
FR2551756A1 (fr) Derives de 4,7-dihydropyrazolo (3,4-b)pyridine et composition pharmaceutique a action anti-hypertensive et de vasodilatation coronaire les renfermant
CH625249A5 (en) Process for the preparation of imidazothiazole derivatives
EP0033432B1 (fr) Composition thérapeutique à base d'imidazoles destinée notamment au traitement des thromboses, nouveaux imidazoles et leur procédé de préparation
FR2551753A2 (fr) Benzotriazine-1,2,3-ones-4, procede de preparation et medicaments les contenant

Legal Events

Date Code Title Description
YP Annual fee paid