NL179585C - Geneesmiddelen met vaatverwijdende en bloeddruk verlagende eigenschappen, op basis van een op de 4-plaats door een via een stikstofatoom gebonden basische groep gesubstitueerd 6-acylaminopyrimidinederivaat, alsmede deze 6-acylaminopyrimidinederivaten zelf. - Google Patents

Geneesmiddelen met vaatverwijdende en bloeddruk verlagende eigenschappen, op basis van een op de 4-plaats door een via een stikstofatoom gebonden basische groep gesubstitueerd 6-acylaminopyrimidinederivaat, alsmede deze 6-acylaminopyrimidinederivaten zelf.

Info

Publication number
NL179585C
NL179585C NLAANVRAGE7801288,A NL7801288A NL179585C NL 179585 C NL179585 C NL 179585C NL 7801288 A NL7801288 A NL 7801288A NL 179585 C NL179585 C NL 179585C
Authority
NL
Netherlands
Prior art keywords
acylaminopyrimidinederivaten
acylaminopyrimidinederivaat
vasodilating
yourself
medicines
Prior art date
Application number
NLAANVRAGE7801288,A
Other languages
English (en)
Dutch (nl)
Other versions
NL7801288A (nl
NL179585B (nl
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AT73877A external-priority patent/AT351036B/de
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NL7801288A publication Critical patent/NL7801288A/xx
Publication of NL179585B publication Critical patent/NL179585B/xx
Application granted granted Critical
Publication of NL179585C publication Critical patent/NL179585C/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NLAANVRAGE7801288,A 1977-02-04 1978-02-03 Geneesmiddelen met vaatverwijdende en bloeddruk verlagende eigenschappen, op basis van een op de 4-plaats door een via een stikstofatoom gebonden basische groep gesubstitueerd 6-acylaminopyrimidinederivaat, alsmede deze 6-acylaminopyrimidinederivaten zelf. NL179585C (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT73877A AT351036B (de) 1977-02-04 1977-02-04 Verfahren zur herstellung von neuen oxadiazolopyrimidinderivaten und von deren salzen
LU7778639A LU78639A1 (de) 1977-02-04 1977-12-05

Publications (3)

Publication Number Publication Date
NL7801288A NL7801288A (nl) 1978-08-08
NL179585B NL179585B (nl) 1986-05-01
NL179585C true NL179585C (nl) 1986-10-01

Family

ID=25593772

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7801288,A NL179585C (nl) 1977-02-04 1978-02-03 Geneesmiddelen met vaatverwijdende en bloeddruk verlagende eigenschappen, op basis van een op de 4-plaats door een via een stikstofatoom gebonden basische groep gesubstitueerd 6-acylaminopyrimidinederivaat, alsmede deze 6-acylaminopyrimidinederivaten zelf.

Country Status (22)

Country Link
US (1) US4150132A (de)
JP (1) JPS6024794B2 (de)
AR (1) AR223642A1 (de)
CA (1) CA1092108A (de)
CH (1) CH638215A5 (de)
DE (1) DE2804518C2 (de)
DK (1) DK50878A (de)
ES (2) ES466589A1 (de)
FI (1) FI62309C (de)
FR (2) FR2379538A1 (de)
GB (2) GB1563887A (de)
GR (1) GR72280B (de)
IE (1) IE46318B1 (de)
IL (2) IL53925A (de)
IT (1) IT1092334B (de)
MC (1) MC1183A1 (de)
NL (1) NL179585C (de)
NO (2) NO780396L (de)
NZ (1) NZ186334A (de)
PH (3) PH13962A (de)
PT (1) PT67614B (de)
SE (1) SE7801311L (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1103245A (en) * 1978-07-21 1981-06-16 Jean-Claude Muller Process for the manufacture of novel oxadiazolopyrimidine derivatives
NZ190915A (en) * 1978-07-31 1984-07-31 Hoffmann La Roche Oxadiazolotriazine derivatives and pharmaceutical compositions
US4307093A (en) * 1980-06-23 1981-12-22 The Upjohn Company Animal feed and process
DK148826C (da) * 1980-12-19 1986-03-24 Hoffmann La Roche Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade
CA1179344A (en) * 1981-07-15 1984-12-11 Jean-Claude Muller Process for the preparation of 6-¬3,6-dihydro-1(2h)- pyridyl| pyrimidine-3-oxides
CH649291A5 (de) * 1982-03-16 1985-05-15 Hoffmann La Roche Dicarbamate.
EP0187854A4 (de) * 1984-07-13 1987-01-22 Gail S Bazzano Substituierte pyrimidinoxide, einsetzbar zur haarwachsanregung.
JPH04249875A (ja) * 1991-01-08 1992-09-04 Yazaki Corp 電線を端子化するための成形用電極及び端子化電線

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3382248A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-4, 5-di(substituted amino)-1, 2-dihydro-1-hydroxy-2-iminopyrimidines
CA1020558A (en) * 1971-04-07 1977-11-08 Richard C. Thomas (Jr.) 6-amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidines
DE2118261A1 (de) * 1971-04-15 1972-11-02 C.H. Boehringer Sohn, 6507 Ingelheim Neue N-haltige Bicyclen, deren Säureadditionssalze sowie Verfahren zu deren Herstellung
BE786028A (fr) * 1971-07-08 1973-01-08 Boehringer Sohn Ingelheim 2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
BE790008A (fr) * 1971-10-15 1973-04-12 Fmc Corp Nouveaux composes herbicides
DE2210633C2 (de) * 1972-03-06 1983-09-22 Bayer Ag, 5090 Leverkusen Kondensierte Pyridinderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE2252122A1 (de) * 1972-10-24 1974-04-25 Hoechst Ag Oxazolo-chinazoline und verfahren zu ihrer herstellung
DE2253555A1 (de) * 1972-11-02 1974-05-09 Hoechst Ag Oxazolo-pyrimidine und verfahren zu ihrer herstellung
US3901928A (en) * 1973-01-10 1975-08-26 Robert Henry Hesse 1' ,3' -dihydroxy steroid-5-enes method of preparing same and their use for preparing 1' -hydroxy-25-hydrogen vitamin d compounds

Also Published As

Publication number Publication date
NZ186334A (en) 1980-05-08
PH13962A (en) 1980-11-12
FR2379538B1 (de) 1980-05-16
NL7801288A (nl) 1978-08-08
JPS5398992A (en) 1978-08-29
NL179585B (nl) 1986-05-01
JPS6024794B2 (ja) 1985-06-14
ES472875A1 (es) 1979-02-16
CA1092108A (en) 1980-12-23
ES466589A1 (es) 1978-10-01
IE46318B1 (en) 1983-05-04
IT7819786A0 (it) 1978-01-30
DE2804518C2 (de) 1985-12-19
FI780343A7 (fi) 1978-08-05
NO780396L (no) 1978-08-07
FR2379538A1 (fr) 1978-09-01
US4150132A (en) 1979-04-17
FI62309C (fi) 1982-12-10
DK50878A (da) 1978-08-05
GB1563888A (en) 1980-04-02
MC1183A1 (fr) 1978-12-22
FI62309B (fi) 1982-08-31
CH638215A5 (de) 1983-09-15
FR2383941A1 (fr) 1978-10-13
IL53925A (en) 1981-06-29
PT67614B (en) 1980-03-03
IT1092334B (it) 1985-07-06
IL53925A0 (en) 1978-04-30
GB1563887A (en) 1980-04-02
PH15009A (en) 1982-05-10
PT67614A (en) 1978-03-01
AR223642A1 (es) 1981-09-15
GR72280B (de) 1983-10-13
DE2804518A1 (de) 1978-08-17
NO803160L (no) 1978-08-07
IE780197L (en) 1978-08-04
IL59627A0 (en) 1980-06-30
SE7801311L (sv) 1978-08-05
FR2383941B1 (de) 1980-07-25
PH14637A (en) 1981-10-12

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Legal Events

Date Code Title Description
BB A search report has been drawn up
BX A request for additional search has been filed
BY An additional search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
BK Erratum

Free format text: IN PAT.BUL.9/86,PAGE 984:ON LINE 11 AFTER OOSTENRIJK (AT) SHOULD BE ADDED: LUXEMBURG (LU)

SNR Assignments of patents or rights arising from examined patent applications

Owner name: F. HOFFMANN-LA ROCHE AG

V1 Lapsed because of non-payment of the annual fee