NO20001404L - Nye stereoselektive fremgangsmÕter for fremstilling av gabapentinanaloger - Google Patents

Nye stereoselektive fremgangsmÕter for fremstilling av gabapentinanaloger

Info

Publication number
NO20001404L
NO20001404L NO20001404A NO20001404A NO20001404L NO 20001404 L NO20001404 L NO 20001404L NO 20001404 A NO20001404 A NO 20001404A NO 20001404 A NO20001404 A NO 20001404A NO 20001404 L NO20001404 L NO 20001404L
Authority
NO
Norway
Prior art keywords
preparation
stereoselective methods
new stereoselective
gabapentin
gabapentin analogs
Prior art date
Application number
NO20001404A
Other languages
English (en)
Other versions
NO20001404D0 (no
NO326227B1 (no
Inventor
Justin Stephen Bryans
Andrew Ian Morrell
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of NO20001404D0 publication Critical patent/NO20001404D0/no
Publication of NO20001404L publication Critical patent/NO20001404L/no
Publication of NO326227B1 publication Critical patent/NO326227B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Silicates, Zeolites, And Molecular Sieves (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
NO20001404A 1997-09-18 2000-03-17 Nye stereoselektive fremgangsmater for fremstilling av gabapentinanaloger NO326227B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5920497P 1997-09-18 1997-09-18
PCT/US1998/016652 WO1999014184A1 (en) 1997-09-18 1998-08-11 Novel stereoselective processes for the preparation of gabapentin analogues

Publications (3)

Publication Number Publication Date
NO20001404D0 NO20001404D0 (no) 2000-03-17
NO20001404L true NO20001404L (no) 2000-03-17
NO326227B1 NO326227B1 (no) 2008-10-20

Family

ID=22021467

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20001404A NO326227B1 (no) 1997-09-18 2000-03-17 Nye stereoselektive fremgangsmater for fremstilling av gabapentinanaloger

Country Status (20)

Country Link
US (1) US6465689B1 (no)
EP (1) EP1015415B1 (no)
JP (1) JP3878809B2 (no)
KR (1) KR100563894B1 (no)
AT (1) ATE239695T1 (no)
AU (1) AU752444B2 (no)
BR (1) BR9812351A (no)
CA (1) CA2295993C (no)
DE (1) DE69814420T2 (no)
DK (1) DK1015415T3 (no)
ES (1) ES2197493T3 (no)
HU (1) HUP0004582A3 (no)
IL (2) IL133782A0 (no)
IS (1) IS2198B (no)
NO (1) NO326227B1 (no)
NZ (1) NZ502786A (no)
PL (1) PL192180B1 (no)
PT (1) PT1015415E (no)
WO (1) WO1999014184A1 (no)
ZA (1) ZA988508B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10203122A1 (de) * 2002-01-25 2003-07-31 Gruenenthal Gmbh Verfahren zur Herstellung von substituierten Acrylsäureestern bzw. deren Einsatz zur Herstellung von substituierten gamma-Aminosäuren
US7439387B2 (en) 2003-04-21 2008-10-21 Matrix Laboratories Ltd. Process for the preparation of Gabapentin form-II
US20050187295A1 (en) * 2004-02-19 2005-08-25 Surendra Kalyan Processes for the preparation of gabapentin
WO2005087709A1 (en) 2004-03-17 2005-09-22 Hikal Limited 4-t-butylgabapentin and its synthesis
US7632864B2 (en) 2004-03-17 2009-12-15 Hikal Ltd. Gabapentin analogues and process thereof
US7442834B2 (en) 2006-06-12 2008-10-28 Zhejiang Chiral Medicine Chemicals Co., Ltd. Process suitable for industrial scale production of gabapentin
WO2013190357A1 (en) * 2012-06-18 2013-12-27 Hikal Limited A process for the preparation of gabapentin

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3928182A1 (de) 1989-08-25 1991-02-28 Goedecke Ag Verfahren zur herstellung von gabapentin
DE69712877T2 (de) 1996-02-07 2002-11-14 Warner-Lambert Co., Morris Plains Zyklischaminosäure als pharmazeutische mittel
EA001214B1 (ru) 1996-03-14 2000-12-25 Варнер-Ламберт Компани Новые мостиковые циклические аминокислоты как фармацевтически применимые вещества

Also Published As

Publication number Publication date
AU8779198A (en) 1999-04-05
CA2295993C (en) 2004-05-04
NZ502786A (en) 2002-05-31
WO1999014184A1 (en) 1999-03-25
IS5355A (is) 2000-05-22
EP1015415A1 (en) 2000-07-05
ES2197493T3 (es) 2004-01-01
KR100563894B1 (ko) 2006-03-24
NO20001404D0 (no) 2000-03-17
DE69814420T2 (de) 2003-11-27
DE69814420D1 (de) 2003-06-12
ATE239695T1 (de) 2003-05-15
PT1015415E (pt) 2003-09-30
PL192180B1 (pl) 2006-09-29
IL133782A (en) 2006-12-31
KR20010024079A (ko) 2001-03-26
US6465689B1 (en) 2002-10-15
BR9812351A (pt) 2000-09-19
CA2295993A1 (en) 1999-03-25
ZA988508B (en) 1999-03-30
IL133782A0 (en) 2001-04-30
IS2198B (is) 2007-02-15
HUP0004582A2 (hu) 2001-05-28
NO326227B1 (no) 2008-10-20
HUP0004582A3 (en) 2002-01-28
DK1015415T3 (da) 2003-07-21
JP3878809B2 (ja) 2007-02-07
PL339296A1 (en) 2000-12-04
AU752444B2 (en) 2002-09-19
JP2001516738A (ja) 2001-10-02
EP1015415B1 (en) 2003-05-07

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