NO20010568L - Substituerte imidazo[1,2a]aziner som selektive COX-2- inhibitorer - Google Patents

Substituerte imidazo[1,2a]aziner som selektive COX-2- inhibitorer

Info

Publication number
NO20010568L
NO20010568L NO20010568A NO20010568A NO20010568L NO 20010568 L NO20010568 L NO 20010568L NO 20010568 A NO20010568 A NO 20010568A NO 20010568 A NO20010568 A NO 20010568A NO 20010568 L NO20010568 L NO 20010568L
Authority
NO
Norway
Prior art keywords
azines
inhibitors
selective cox
substituted imidazo
imidazo
Prior art date
Application number
NO20010568A
Other languages
English (en)
Other versions
NO20010568D0 (no
Inventor
Carles Farrerons Gallemi
Ignacio-Jose Miquel Bono
Ana Maria Fernandez Serrat
Carlos Monserrat Vidal
Carmen Lagunas Arnal
Ferran Gimenez Guasch
Andres Fernandez Garcia
Original Assignee
L V A T Sa Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by L V A T Sa Lab Sa filed Critical L V A T Sa Lab Sa
Publication of NO20010568D0 publication Critical patent/NO20010568D0/no
Publication of NO20010568L publication Critical patent/NO20010568L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20010568A 1998-08-03 2001-02-02 Substituerte imidazo[1,2a]aziner som selektive COX-2- inhibitorer NO20010568L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009801652A ES2140354B1 (es) 1998-08-03 1998-08-03 Imidazo (1,2a) azinas sustituidas como inhibidores selectivos de la cox-2.
PCT/ES1999/000235 WO2000008024A1 (es) 1998-08-03 1999-07-23 IMIDAZO[1,2a]AZINAS SUSTITUIDAS COMO INHIBIDORES SELECTIVOS DE LA COX-2

Publications (2)

Publication Number Publication Date
NO20010568D0 NO20010568D0 (no) 2001-02-02
NO20010568L true NO20010568L (no) 2001-04-02

Family

ID=8304755

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20010568A NO20010568L (no) 1998-08-03 2001-02-02 Substituerte imidazo[1,2a]aziner som selektive COX-2- inhibitorer

Country Status (30)

Country Link
US (1) US6670365B1 (no)
EP (1) EP1104762B1 (no)
JP (1) JP2002522438A (no)
KR (1) KR20010079602A (no)
CN (1) CN1131865C (no)
AP (1) AP2001002082A0 (no)
AT (1) ATE224391T1 (no)
AU (1) AU749770B2 (no)
BG (1) BG105299A (no)
BR (1) BR9912968A (no)
CA (1) CA2339187A1 (no)
CZ (1) CZ291783B6 (no)
DE (1) DE69903046T2 (no)
DK (1) DK1104762T3 (no)
EA (1) EA003399B1 (no)
ES (2) ES2140354B1 (no)
HU (1) HUP0103004A3 (no)
ID (1) ID28539A (no)
IL (1) IL141242A0 (no)
MX (1) MXPA01001332A (no)
NO (1) NO20010568L (no)
NZ (1) NZ510196A (no)
OA (1) OA11592A (no)
PL (1) PL345804A1 (no)
PT (1) PT1104762E (no)
SK (1) SK1662001A3 (no)
TR (1) TR200100359T2 (no)
WO (1) WO2000008024A1 (no)
YU (1) YU7401A (no)
ZA (1) ZA200101632B (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CO5261556A1 (es) 1999-12-08 2003-03-31 Pharmacia Corp Composiciones inhibidoras de ciclooxigenasa-2 que tiene rapido acceso de efecto terapeutico
US8241622B2 (en) * 2001-07-13 2012-08-14 University Of Iowa Research Foundation Adeno-associated virus vectors with intravector heterologous terminal palindromic sequences
US20030100594A1 (en) * 2001-08-10 2003-05-29 Pharmacia Corporation Carbonic anhydrase inhibitor
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
DE10256881A1 (de) * 2002-12-05 2004-06-24 Beiersdorf Ag Neue topische Verwendung von Bis-Arylimidazo[1,2-a]thiolanderivaten
PT1534305E (pt) 2003-05-07 2007-02-28 Osteologix As Tratamento de afecções cartilagineas / osseas com sais de estroncio hidrosoluveis
JP2007500160A (ja) * 2003-07-30 2007-01-11 ラボラトリオス・エセ・ア・エレ・ベ・ア・テ・ソシエダッド・アノニマ 癌の予防および治療のための置換イミダゾピリミジン
WO2007034278A2 (en) * 2005-09-19 2007-03-29 Pfizer Products Inc. Fused imidazole derivatives as c3a receptor antagonists
EP1971867A2 (en) * 2005-12-30 2008-09-24 University of Iowa Research Foundation Method of identifying compounds useful to treat neuronal degenerative diseases
WO2007096764A2 (en) * 2006-02-27 2007-08-30 Glenmark Pharmaceuticals S.A. Bicyclic heteroaryl derivatives as cannabinoid receptor modulators
CA2704436C (en) * 2007-11-14 2016-01-05 Ortho-Mcneil-Janssen Pharmaceuticals, Inc. Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
AU2009300318A1 (en) * 2008-10-01 2010-04-08 Synta Pharmaceuticals Corp. Compounds for inflammation and immune-related uses
GB201321732D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
WO2017139381A1 (en) 2016-02-08 2017-08-17 University Of Iowa Research Foundation Methods to produce chimeric adeno-associated virus/bocavirus parvovirus
WO2017155973A1 (en) 2016-03-07 2017-09-14 University Of Iowa Research Foundation Aav-mediated expression using a synthetic promoter and enhancer
US12173305B2 (en) 2016-05-26 2024-12-24 University Of Iowa Research Foundation cis and trans requirements for terminal resolution of human bocavirus 1
US11142775B2 (en) 2017-01-13 2021-10-12 University Of Iowa Research Foundation Bocaparvovirus small noncoding RNA and uses thereof
IL305573A (en) 2021-03-15 2023-10-01 Saul Yedgar HYALURONIC ACID-CONJUGATED DIPALMITOYL PHOSPHATIDYL ETHANOLAMINE IN COMBINATION WITH NON-STEROIDAL ANTI-INFLAMMATORY DRUGS (NSAIDs) FOR TREATING OR ALLEVIATING INFLAMMATORY DISEASES

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2785133A (en) * 1954-03-26 1957-03-12 Gen Aniline & Film Corp Compositions for a method of whitening fine fabrics
US3455924A (en) * 1967-02-08 1969-07-15 Upjohn Co Dianisylimidazoles
JPH06504779A (ja) * 1990-12-13 1994-06-02 スミスクライン・ビーチャム・コーポレイション 新規ｃｓａｉｄｓ
WO1993019066A1 (fr) * 1992-03-17 1993-09-30 Nippon Shinyaku Co., Ltd. Derive de l'imidazopyridine et medicament
US5620999A (en) 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
NZ304886A (en) * 1995-04-04 1998-11-25 Glaxo Group Ltd Imidazo [1,2a] pyridine derivatives, preparation and pharmaceutical compositions thereof
UA57002C2 (uk) * 1995-10-13 2003-06-16 Мерк Фросст Кенада Енд Ко./Мерк Фросст Кенада Енд Сі. Похідне (метилсульфоніл)феніл-2-(5н)-фуранону, фармацевтична композиція та спосіб лікування

Also Published As

Publication number Publication date
IL141242A0 (en) 2002-03-10
HK1037629A1 (en) 2002-02-15
EP1104762B1 (en) 2002-09-18
SK1662001A3 (en) 2001-08-06
ES2182546T3 (es) 2003-03-01
KR20010079602A (ko) 2001-08-22
US6670365B1 (en) 2003-12-30
MXPA01001332A (es) 2002-11-29
WO2000008024A1 (es) 2000-02-17
AU749770B2 (en) 2002-07-04
CN1321157A (zh) 2001-11-07
YU7401A (sh) 2003-10-31
EA200100212A1 (ru) 2001-08-27
NO20010568D0 (no) 2001-02-02
DK1104762T3 (da) 2002-10-21
EP1104762A1 (en) 2001-06-06
ATE224391T1 (de) 2002-10-15
TR200100359T2 (tr) 2001-06-21
JP2002522438A (ja) 2002-07-23
CN1131865C (zh) 2003-12-24
ES2140354A1 (es) 2000-02-16
PT1104762E (pt) 2002-11-29
ES2140354B1 (es) 2000-11-01
HUP0103004A3 (en) 2003-03-28
OA11592A (en) 2004-07-30
PL345804A1 (en) 2002-01-02
ZA200101632B (en) 2001-08-30
BR9912968A (pt) 2001-05-08
ID28539A (id) 2001-05-31
DE69903046D1 (de) 2002-10-24
EA003399B1 (ru) 2003-04-24
HUP0103004A2 (hu) 2002-01-28
AU4782499A (en) 2000-02-28
CA2339187A1 (en) 2000-02-17
AP2001002082A0 (en) 2001-03-31
BG105299A (en) 2001-11-30
DE69903046T2 (de) 2003-05-22
CZ2001433A3 (cs) 2001-08-15
CZ291783B6 (cs) 2003-05-14
NZ510196A (en) 2002-09-27

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