DK1104762T3 - Substituerede imidazo[1,2a]aziner som selektive COX-2-inhibitorer - Google Patents

Substituerede imidazo[1,2a]aziner som selektive COX-2-inhibitorer

Info

Publication number: DK1104762T3
Authority: DK; Denmark
Prior art keywords: azines; inhibitors; selective cox; substituted imidazo; imidazo
Prior art date: 1998-08-03

Application number

DK99931266T

Other languages

English (en)

Inventor

Gallemi Carles Farrerons

Bono Ignacio-Jose Miquel

Serrat Ana Maria Fernandez

Vidal Carlos Monserrat

Arnal Carmen Lagunas

Guasch Ferran Gimenez

Garcia Andres Fernandez

Original Assignee

S A L V A T Lab Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-08-03

Filing date

1999-07-23

Publication date

2002-10-21

1999-07-23 Application filed by S A L V A T Lab Sa filed Critical S A L V A T Lab Sa

2002-10-21 Application granted granted Critical

2002-10-21 Publication of DK1104762T3 publication Critical patent/DK1104762T3/da

Links

229940111134 coxibs Drugs 0.000 title 1
239000003255 cyclooxygenase 2 inhibitor Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

DK99931266T 1998-08-03 1999-07-23 Substituerede imidazo[1,2a]aziner som selektive COX-2-inhibitorer DK1104762T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ES009801652A ES2140354B1 (es)	1998-08-03	1998-08-03	Imidazo (1,2a) azinas sustituidas como inhibidores selectivos de la cox-2.
PCT/ES1999/000235 WO2000008024A1 (es)	1998-08-03	1999-07-23	IMIDAZO[1,2a]AZINAS SUSTITUIDAS COMO INHIBIDORES SELECTIVOS DE LA COX-2

Publications (1)

Publication Number	Publication Date
DK1104762T3 true DK1104762T3 (da)	2002-10-21

Family

ID=8304755

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK99931266T DK1104762T3 (da)	1998-08-03	1999-07-23	Substituerede imidazo[1,2a]aziner som selektive COX-2-inhibitorer

Country Status (30)

Country	Link
US (1)	US6670365B1 (da)
EP (1)	EP1104762B1 (da)
JP (1)	JP2002522438A (da)
KR (1)	KR20010079602A (da)
CN (1)	CN1131865C (da)
AP (1)	AP2001002082A0 (da)
AT (1)	ATE224391T1 (da)
AU (1)	AU749770B2 (da)
BG (1)	BG105299A (da)
BR (1)	BR9912968A (da)
CA (1)	CA2339187A1 (da)
CZ (1)	CZ291783B6 (da)
DE (1)	DE69903046T2 (da)
DK (1)	DK1104762T3 (da)
EA (1)	EA003399B1 (da)
ES (2)	ES2140354B1 (da)
HU (1)	HUP0103004A3 (da)
ID (1)	ID28539A (da)
IL (1)	IL141242A0 (da)
MX (1)	MXPA01001332A (da)
NO (1)	NO20010568L (da)
NZ (1)	NZ510196A (da)
OA (1)	OA11592A (da)
PL (1)	PL345804A1 (da)
PT (1)	PT1104762E (da)
SK (1)	SK1662001A3 (da)
TR (1)	TR200100359T2 (da)
WO (1)	WO2000008024A1 (da)
YU (1)	YU7401A (da)
ZA (1)	ZA200101632B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CO5261556A1 (es)	1999-12-08	2003-03-31	Pharmacia Corp	Composiciones inhibidoras de ciclooxigenasa-2 que tiene rapido acceso de efecto terapeutico
US8241622B2 (en) *	2001-07-13	2012-08-14	University Of Iowa Research Foundation	Adeno-associated virus vectors with intravector heterologous terminal palindromic sequences
US20030100594A1 (en) *	2001-08-10	2003-05-29	Pharmacia Corporation	Carbonic anhydrase inhibitor
DE10247271A1 (de) *	2002-10-10	2004-08-26	Grünenthal GmbH	Substituierte C-Imidazo[1,2-a]pyridin-3-yle
DE10256881A1 (de) *	2002-12-05	2004-06-24	Beiersdorf Ag	Neue topische Verwendung von Bis-Arylimidazo[1,2-a]thiolanderivaten
PT1534305E (pt)	2003-05-07	2007-02-28	Osteologix As	Tratamento de afecções cartilagineas / osseas com sais de estroncio hidrosoluveis
JP2007500160A (ja) *	2003-07-30	2007-01-11	ラボラトリオス・エセ・ア・エレ・ベ・ア・テ・ソシエダッド・アノニマ	癌の予防および治療のための置換イミダゾピリミジン
WO2007034278A2 (en) *	2005-09-19	2007-03-29	Pfizer Products Inc.	Fused imidazole derivatives as c3a receptor antagonists
EP1971867A2 (en) *	2005-12-30	2008-09-24	University of Iowa Research Foundation	Method of identifying compounds useful to treat neuronal degenerative diseases
WO2007096764A2 (en) *	2006-02-27	2007-08-30	Glenmark Pharmaceuticals S.A.	Bicyclic heteroaryl derivatives as cannabinoid receptor modulators
CA2704436C (en) *	2007-11-14	2016-01-05	Ortho-Mcneil-Janssen Pharmaceuticals, Inc.	Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
AU2009300318A1 (en) *	2008-10-01	2010-04-08	Synta Pharmaceuticals Corp.	Compounds for inflammation and immune-related uses
GB201321732D0 (en) *	2013-12-09	2014-01-22	Ucb Pharma Sa	Therapeutic agents
WO2017139381A1 (en)	2016-02-08	2017-08-17	University Of Iowa Research Foundation	Methods to produce chimeric adeno-associated virus/bocavirus parvovirus
WO2017155973A1 (en)	2016-03-07	2017-09-14	University Of Iowa Research Foundation	Aav-mediated expression using a synthetic promoter and enhancer
US12173305B2 (en)	2016-05-26	2024-12-24	University Of Iowa Research Foundation	cis and trans requirements for terminal resolution of human bocavirus 1
US11142775B2 (en)	2017-01-13	2021-10-12	University Of Iowa Research Foundation	Bocaparvovirus small noncoding RNA and uses thereof
IL305573A (en)	2021-03-15	2023-10-01	Saul Yedgar	HYALURONIC ACID-CONJUGATED DIPALMITOYL PHOSPHATIDYL ETHANOLAMINE IN COMBINATION WITH NON-STEROIDAL ANTI-INFLAMMATORY DRUGS (NSAIDs) FOR TREATING OR ALLEVIATING INFLAMMATORY DISEASES

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2785133A (en) *	1954-03-26	1957-03-12	Gen Aniline & Film Corp	Compositions for a method of whitening fine fabrics
US3455924A (en) *	1967-02-08	1969-07-15	Upjohn Co	Dianisylimidazoles
JPH06504779A (ja) *	1990-12-13	1994-06-02	スミスクライン・ビーチャム・コーポレイション	新規ｃｓａｉｄｓ
WO1993019066A1 (fr) *	1992-03-17	1993-09-30	Nippon Shinyaku Co., Ltd.	Derive de l'imidazopyridine et medicament
US5620999A (en)	1994-07-28	1997-04-15	Weier; Richard M.	Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
NZ304886A (en) *	1995-04-04	1998-11-25	Glaxo Group Ltd	Imidazo [1,2a] pyridine derivatives, preparation and pharmaceutical compositions thereof
UA57002C2 (uk) *	1995-10-13	2003-06-16	Мерк Фросст Кенада Енд Ко./Мерк Фросст Кенада Енд Сі.	Похідне (метилсульфоніл)феніл-2-(5н)-фуранону, фармацевтична композиція та спосіб лікування

1998
- 1998-08-03 ES ES009801652A patent/ES2140354B1/es not_active Expired - Lifetime
1999
- 1999-07-23 AT AT99931266T patent/ATE224391T1/de not_active IP Right Cessation
- 1999-07-23 PL PL99345804A patent/PL345804A1/xx not_active IP Right Cessation
- 1999-07-23 IL IL14124299A patent/IL141242A0/xx unknown
- 1999-07-23 MX MXPA01001332A patent/MXPA01001332A/es unknown
- 1999-07-23 AP APAP/P/2001/002082A patent/AP2001002082A0/en unknown
- 1999-07-23 ID IDW20010517A patent/ID28539A/id unknown
- 1999-07-23 DE DE69903046T patent/DE69903046T2/de not_active Expired - Fee Related
- 1999-07-23 CA CA002339187A patent/CA2339187A1/en not_active Abandoned
- 1999-07-23 KR KR1020017001453A patent/KR20010079602A/ko not_active Ceased
- 1999-07-23 SK SK166-2001A patent/SK1662001A3/sk unknown
- 1999-07-23 YU YU7401A patent/YU7401A/sh unknown
- 1999-07-23 WO PCT/ES1999/000235 patent/WO2000008024A1/es not_active Ceased
- 1999-07-23 OA OA1200100033A patent/OA11592A/en unknown
- 1999-07-23 CN CN998116750A patent/CN1131865C/zh not_active Expired - Fee Related
- 1999-07-23 JP JP2000563657A patent/JP2002522438A/ja active Pending
- 1999-07-23 PT PT99931266T patent/PT1104762E/pt unknown
- 1999-07-23 NZ NZ510196A patent/NZ510196A/xx unknown
- 1999-07-23 HU HU0103004A patent/HUP0103004A3/hu unknown
- 1999-07-23 AU AU47824/99A patent/AU749770B2/en not_active Ceased
- 1999-07-23 BR BR9912968-0A patent/BR9912968A/pt not_active IP Right Cessation
- 1999-07-23 ES ES99931266T patent/ES2182546T3/es not_active Expired - Lifetime
- 1999-07-23 DK DK99931266T patent/DK1104762T3/da active
- 1999-07-23 CZ CZ2001433A patent/CZ291783B6/cs not_active IP Right Cessation
- 1999-07-23 US US09/762,146 patent/US6670365B1/en not_active Expired - Fee Related
- 1999-07-23 EP EP99931266A patent/EP1104762B1/en not_active Expired - Lifetime
- 1999-07-23 TR TR2001/00359T patent/TR200100359T2/xx unknown
- 1999-07-23 EA EA200100212A patent/EA003399B1/ru not_active IP Right Cessation
2001
- 2001-02-02 NO NO20010568A patent/NO20010568L/no not_active Application Discontinuation
- 2001-02-27 ZA ZA200101632A patent/ZA200101632B/en unknown
- 2001-02-28 BG BG105299A patent/BG105299A/xx unknown

Also Published As

Publication number	Publication date
IL141242A0 (en)	2002-03-10
HK1037629A1 (en)	2002-02-15
EP1104762B1 (en)	2002-09-18
SK1662001A3 (en)	2001-08-06
ES2182546T3 (es)	2003-03-01
KR20010079602A (ko)	2001-08-22
US6670365B1 (en)	2003-12-30
MXPA01001332A (es)	2002-11-29
WO2000008024A1 (es)	2000-02-17
AU749770B2 (en)	2002-07-04
CN1321157A (zh)	2001-11-07
YU7401A (sh)	2003-10-31
EA200100212A1 (ru)	2001-08-27
NO20010568D0 (no)	2001-02-02
EP1104762A1 (en)	2001-06-06
ATE224391T1 (de)	2002-10-15
TR200100359T2 (tr)	2001-06-21
JP2002522438A (ja)	2002-07-23
CN1131865C (zh)	2003-12-24
ES2140354A1 (es)	2000-02-16
PT1104762E (pt)	2002-11-29
ES2140354B1 (es)	2000-11-01
HUP0103004A3 (en)	2003-03-28
OA11592A (en)	2004-07-30
PL345804A1 (en)	2002-01-02
ZA200101632B (en)	2001-08-30
BR9912968A (pt)	2001-05-08
ID28539A (id)	2001-05-31
NO20010568L (no)	2001-04-02
DE69903046D1 (de)	2002-10-24
EA003399B1 (ru)	2003-04-24
HUP0103004A2 (hu)	2002-01-28
AU4782499A (en)	2000-02-28
CA2339187A1 (en)	2000-02-17
AP2001002082A0 (en)	2001-03-31
BG105299A (en)	2001-11-30
DE69903046T2 (de)	2003-05-22
CZ2001433A3 (cs)	2001-08-15
CZ291783B6 (cs)	2003-05-14
NZ510196A (en)	2002-09-27

Publication	Publication Date	Title
NO20012156D0 (no)	2001-05-02	Pyrazolopyridinderivater som selektive COX-2 inhibitorer
DK2253620T3 (da)	2014-03-31	Substituerede 3-cyanoquinoliner som protein-tyrosinkinase-inhibitorer
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DE69933287D1 (de)	2006-11-02	12,13-modifizierte epothilon-derivate
IS5722A (is)	2000-11-21	Pýróló [2,3-dl]pírimídín efnasambönd
NO20010568L (no)	2001-04-02	Substituerte imidazo[1,2a]aziner som selektive COX-2- inhibitorer
NO20010684D0 (no)	2001-02-09	Substituert 1,8-Naphthyridin-4(1H)-on som fosfodiesterase 4 inhibitorer
DK0946512T3 (da)	2004-01-12	6-Phenylpyridyl-2-aminderivater, der er nyttige som NOS-inhibitorer
NO20003451D0 (no)	2000-07-04	2,3-substituerte indolforbindelser som cox-2 inhibitorer
NO20010331L (no)	2001-03-20	Ftalazinderivater som fosfodiesterase 4-inhibitorer
ATE204279T1 (de)	2001-09-15	Diaza-spiro(3,5)nonan-derivate
EE200000447A (et)	2001-12-17	1,3,4-oksadiasolooni derivaadid
DK1075471T3 (da)	2005-01-17	Idolylderivater som serotonerge midler
NO20021846D0 (no)	2002-04-19	Imidazolderivater som fosfodiesterase VII-inhibitorer
DK1073651T3 (da)	2003-01-27	Indolylderivater som serotonerge midler
DK0944601T3 (da)	2003-06-10	Heterocykliske quanidinylaminoforbindelser som alfa-2-adrenoceptoragonister
DK1115708T3 (da)	2004-08-02	Aminoalkyl-3,4-dihydriquinolinderivater som NO-synthaseinhibitorer
FI980053A0 (fi)	1998-01-14	Anordning foer utformande av fiberbollar av laongstraeckta fibrer som foeljer med enluftstroem
DE59909590D1 (de)	2004-07-01	Azidfreie, gaserzeugende zusammensetzung
NO20011309D0 (no)	2001-03-15	Benzotieno [3,2-c]pyridiner som<alfa>2-antagonister
SI1104762T1 (en)	2002-12-31	Substituted imidazo(1,2a)azines as selective inhibitors of cox-2
ES1044951Y (es)	2000-12-16	Tabique perfeccionado.
FI980755A0 (fi)	1998-04-02	Foerfarande foer montering/faestande av vaermeisoleringsskivor som vaermeisolering i en byggnad
ES1040348Y (es)	1999-08-16	Portabrocas.
FI980722A0 (fi)	1998-03-31	Motions-, rehabiliterings-, sport- och lagspelredskap som staerker baolens muskler